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科研机构
上海药物研究所 [45]
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期刊论文 [44]
会议论文 [1]
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2021 [4]
2020 [3]
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A General Set of DNA-Compatible Reactions for Preparing DNA-Tagged Multisubstituted Pyrroles
期刊论文
BIOCONJUGATE CHEMISTRY, 2021, 卷号: 32, 期号: 11, 页码: 2290-2294
作者:
Qi, Jingjing
;
Liu, Sixiu
;
Seydimemet, Mengnisa
;
Wang, Xuan
;
Lu, Xiaojie
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2022/01/04
Synthesis and Evaluation of 3-(Indol-3-yl)-4-(Pyrazolo[3,4-c]Pyridazin-3-yl)-Maleimides as Potent Mutant Isocitrate Dehydrogenase-1 Inhibitors
期刊论文
PHARMACEUTICAL CHEMISTRY JOURNAL, 2021, 卷号: 55, 期号: 7, 页码: 655-664
作者:
Xu, Jianghong
;
Hu, Yuanyuan
;
Liu, Xiaoqi
;
Gao, Anhui
;
Gao, Lixin
收藏
  |  
浏览/下载:34/0
  |  
提交时间:2021/12/01
IDH1-R132H inhibitors
synthesis
biological activity
docking
3-(indol-3-yl)-4-(pyrazolo-[3
4-c]pyridazin-3-yl)-maleimides
Blood Pyrrole-DNA Adducts Define the Early Tumorigenic Risk in Patients with Pyrrolizidine Alkaloid-Induced Liver Injury
期刊论文
ENVIRONMENTAL SCIENCE & TECHNOLOGY LETTERS, 2021, 卷号: 8, 期号: 7, 页码: 551-557
作者:
He, Yisheng
;
Zhang, Wei
;
Ma, Jiang
;
Xia, Qingsu
;
Song, Zijing
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2021/08/17
Synthetic Studies toward DNA-Encoded Heterocycles Based on the On-DNA Formation of alpha,beta-Unsaturated Ketones
期刊论文
ORGANIC LETTERS, 2021, 卷号: 23, 期号: 3, 页码: 908-913
作者:
Liu, Sixiu
;
Qi, Jingjing
;
Lu, Weiwei
;
Wang, Xuan
;
Lu, Xiaojie
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2021/05/24
Clinical application of pyrrole-hemoglobin adducts as a biomarker of pyrrolizidine alkaloid exposure in humans
期刊论文
ARCHIVES OF TOXICOLOGY, 2020, 页码: 7
作者:
Ma, Jiang
;
Zhang, Wei
;
He, Yisheng
;
Zhu, Lin
;
Zhang, Chunyuan
收藏
  |  
浏览/下载:41/0
  |  
提交时间:2020/12/24
Pyrrolizidine alkaloids
Liver injury
Diagnostic biomarkers
Pyrrole-hemoglobin adducts
Pyrrole-plasma protein adducts
Tu-San-Qi (Gynura japonica): the culprit behind pyrrolizidine alkaloid-induced liver injury in China
期刊论文
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 11
作者:
Zhu, Lin
;
Zhang, Chun-yuan
;
Li, Dong-ping
;
Chen, Hu-biao
;
Ma, Jiang
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2020/12/24
herb-induced liver injury
hepatic sinusoidal obstruction syndrome
pyrrolizidine alkaloids
Tu-San-Qi
Gynura japonica
Copper-mediated C-H thiolation of (hetero)arenes using weakly coordinating directing group
期刊论文
TETRAHEDRON LETTERS, 2020, 卷号: 61, 期号: 28, 页码: 4
作者:
Wu, Peng
;
Cheng, Tai-Jin
;
Lin, Hai-Xia
;
Xu, Hui
;
Dai, Hui-Xiong
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2020/12/24
Copper catalyst
C-H activation
Weakly coordinating directing group
Thiolation
Pyrrole-Hemoglobin Adducts, a More Feasible Potential Biomarker of Pyrrolizidine Alkaloid Exposure
期刊论文
CHEMICAL RESEARCH IN TOXICOLOGY, 2019, 卷号: 32, 期号: 6, 页码: 1027-1039
作者:
Ma, Jiang
;
Ruan, Jianqing
;
Chen, Xinmeng
;
Li, Dongping
;
Yao, Sheng
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2020/07/01
Gold-catalyzed Rapid Construction of Nitrogen-containing Heterocyclic Compound Library with Scaffold Diversity and Molecular Complexity
期刊论文
ADVANCED SYNTHESIS & CATALYSIS, 2019, 卷号: 361, 期号: 6, 页码: 1419-1440
作者:
Qiao, Jin
;
Jia, Xiuwen
;
Li, Pinyi
;
Liu, Xiaoyan
;
Zhao, Jingwei
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2020/07/01
Alkynes
Amines
Cascade reaction
Compound library
Gold
Scaffold diversity
Green and Facile Assembly of Diverse Fused N-Heterocycles Using Gold-Catalyzed Cascade Reactions in Water
期刊论文
MOLECULES, 2019, 卷号: 24, 期号: 5, 页码: 30
作者:
Jia, Xiuwen
;
Li, Pinyi
;
Liu, Xiaoyan
;
Lin, Jiafu
;
Chu, Yiwen
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2020/07/01
amine nucleophiles
alkynoic acids
cascade reaction
gold catalysis
fused N-heterocycles
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