×
验证码:
换一张
忘记密码?
记住我
CORC
首页
科研机构
检索
知识图谱
申请加入
托管服务
登录
注册
在结果中检索
科研机构
山东大学 [78]
吉林大学白求恩第一... [52]
化学研究所 [28]
上海药物研究所 [28]
兰州大学 [22]
福建物质结构研究所 [22]
更多...
内容类型
期刊论文 [410]
专利 [56]
会议论文 [8]
学位论文 [8]
无文献类型 [2]
其他 [1]
更多...
发表日期
2021 [3]
2019 [17]
2018 [27]
2017 [16]
2016 [24]
2015 [22]
更多...
学科主题
chemistry [16]
crystallog... [7]
Pharmacolo... [4]
Chemistry [3]
有机氟化学 [3]
物理化学 [3]
更多...
×
知识图谱
CORC
开始提交
已提交作品
待认领作品
已认领作品
未提交全文
收藏管理
QQ客服
官方微博
反馈留言
浏览/检索结果:
共485条,第1-10条
帮助
已选(
0
)
清除
条数/页:
5
10
15
20
25
30
35
40
45
50
55
60
65
70
75
80
85
90
95
100
排序方式:
请选择
作者升序
作者降序
题名升序
题名降序
发表日期升序
发表日期降序
提交时间升序
提交时间降序
Design, synthesis, and biological evaluation of 4-benzoylamino-1H-pyrazole-3-carboxamide derivatives as potent CDK2 inhibitors
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 215, 页码: 12
作者:
Lin, Tingting
;
Li, Jiacheng
;
Liu, Liping
;
Li, Yuanqing
;
Jiang, Hualiang
收藏
  |  
浏览/下载:70/0
  |  
提交时间:2021/05/24
CDK2 inhibitor
Selectivity
Anti-proliferative potency
Synthetic Studies toward DNA-Encoded Heterocycles Based on the On-DNA Formation of alpha,beta-Unsaturated Ketones
期刊论文
ORGANIC LETTERS, 2021, 卷号: 23, 期号: 3, 页码: 908-913
作者:
Liu, Sixiu
;
Qi, Jingjing
;
Lu, Weiwei
;
Wang, Xuan
;
Lu, Xiaojie
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2021/05/24
A Novel Fluorescent Probe Based on Pyrazole-Pyrazoline for Fe (III) Ions Recognition
期刊论文
Journal of Fluorescence, 2021, 卷号: 31, 期号: 1, 页码: 29-38
作者:
Zhang, Ying-Peng
;
Li, Xiang-Fang
;
Yang, Yun-Shang
;
Wang, Jing-Li
;
Zhao, Yu-Chen
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2021/03/02
Binding energy
Fluorescence
Fluorescence spectroscopy
Metal ions
Metals
Probes
Uranium metallography
Vanadium metallography
Fluorescence intensities
Fluorescent probes
Selective recognition
Selectivity and sensitivity
Sensing mechanism
Tetra-hydrofuran
Theoretical calculations
UV absorption spectrum
fDiscovery of pyrazole-thiophene derivatives as highly Potent, orally active Akt inhibitors
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 180, 页码: 72-85
作者:
Zhan, Wenhu
;
Che, Jinxin
;
Xu, Lei
;
Wu, Yizhe
;
Hu, Xiaobei
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2020/07/01
Pyrazole-thiophene derivatives
Akt inhibitor
Antitumor
Pd-Catalyzed intramolecular C-H activation and C-S formation to synthesize pyrazolo[5,1-b]benzothiazoles without an additional oxidant
期刊论文
ORGANIC CHEMISTRY FRONTIERS, 2019, 卷号: 6, 期号: 18, 页码: 3234-3237
作者:
Peng, Yingyuan
;
He, Qian
;
Zhang, Xiaofei
;
Yang, Chunhao
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2020/07/01
Discovery of 1,3-diphenyl-1H-pyrazole derivatives containing rhodanine-3-alkanoic acid groups as potential PTP1B inhibitors
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2019, 卷号: 29, 期号: 10, 页码: 1187-1193
作者:
Sun, Liangpeng
;
Wang, Peipei
;
Xu, Lili
;
Gao, Lixin
;
Li, Jia
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2020/07/01
PTP1B inhibitor
1,3-Diphenyl-1H-pyrazole
Rhodanine-3-alkanoic acid
Design, synthesis and structure-activity relationship optimization of phenanthridine derivatives as new Wnt/beta-catenin signalling pathway agonists
期刊论文
BIOORGANIC CHEMISTRY, 2019, 卷号: 84, 页码: 285-294
作者:
Chen, Duo-zhi
;
Yang, Bi-juan
;
He, Xiao-li
;
Fan, Shi-rui
;
Cai, Jie-yun
收藏
  |  
浏览/下载:113/0
  |  
提交时间:2019/03/18
Wnt/beta-catenin signalling pathway agonist
Phenanthridine derivatives
Structural optimization
Structure-activity relationships (SARs)
Synthesis, biological evaluation and molecular docking of benzimidazole grafted benzsulfamide-containing pyrazole ring derivatives as novel tubulin polymerization inhibitors
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2019, 卷号: 27, 期号: 3
作者:
Shi, Tian-Qi
;
Wang, Yan-Ting
;
Liu, Chang-Hong
;
Zhu, Hai-Liang
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2019/12/05
Benzimidazole
Benzsulfamide
Pyrazole
Tubulin
Inhibition
Apoptosis
Molecular docking
Discovery of novel bacterial FabH inhibitors (Pyrazol-Benzimidazole amide derivatives): Design, synthesis, bioassay, molecular docking and crystal structure determination
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 171
作者:
Wang, Yan-Ting
;
Shi, Tian-Qi
;
Fu, Jie
;
Zhu, Hai-Liang
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2019/12/05
FabH
Inhibitor
Pyrazole
Antibacterial
Molecule docking
Synthesis and bioevaluation of diarylpyrazoles as antiproliferative agents
期刊论文
European Journal of Medicinal Chemistry, 2019
作者:
Chao Wang
;
Shuang Yang
;
Jianan Du
;
Jia Ni
;
Yue Wu
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2019/12/13
CA-4
Tubulin
Pyrazole
Colchicine
binding
site
©版权所有 ©2017 CSpace - Powered by
CSpace