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Design, synthesis, and biological evaluation of 4-benzoylamino-1H-pyrazole-3-carboxamide derivatives as potent CDK2 inhibitors 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 215, 页码: 12
作者:  Lin, Tingting;  Li, Jiacheng;  Liu, Liping;  Li, Yuanqing;  Jiang, Hualiang
收藏  |  浏览/下载:70/0  |  提交时间:2021/05/24
Synthetic Studies toward DNA-Encoded Heterocycles Based on the On-DNA Formation of alpha,beta-Unsaturated Ketones 期刊论文
ORGANIC LETTERS, 2021, 卷号: 23, 期号: 3, 页码: 908-913
作者:  Liu, Sixiu;  Qi, Jingjing;  Lu, Weiwei;  Wang, Xuan;  Lu, Xiaojie
收藏  |  浏览/下载:11/0  |  提交时间:2021/05/24
A Novel Fluorescent Probe Based on Pyrazole-Pyrazoline for Fe (III) Ions Recognition 期刊论文
Journal of Fluorescence, 2021, 卷号: 31, 期号: 1, 页码: 29-38
作者:  Zhang, Ying-Peng;  Li, Xiang-Fang;  Yang, Yun-Shang;  Wang, Jing-Li;  Zhao, Yu-Chen
收藏  |  浏览/下载:5/0  |  提交时间:2021/03/02
fDiscovery of pyrazole-thiophene derivatives as highly Potent, orally active Akt inhibitors 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 180, 页码: 72-85
作者:  Zhan, Wenhu;  Che, Jinxin;  Xu, Lei;  Wu, Yizhe;  Hu, Xiaobei
收藏  |  浏览/下载:15/0  |  提交时间:2020/07/01
Pd-Catalyzed intramolecular C-H activation and C-S formation to synthesize pyrazolo[5,1-b]benzothiazoles without an additional oxidant 期刊论文
ORGANIC CHEMISTRY FRONTIERS, 2019, 卷号: 6, 期号: 18, 页码: 3234-3237
作者:  Peng, Yingyuan;  He, Qian;  Zhang, Xiaofei;  Yang, Chunhao
收藏  |  浏览/下载:1/0  |  提交时间:2020/07/01
Discovery of 1,3-diphenyl-1H-pyrazole derivatives containing rhodanine-3-alkanoic acid groups as potential PTP1B inhibitors 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2019, 卷号: 29, 期号: 10, 页码: 1187-1193
作者:  Sun, Liangpeng;  Wang, Peipei;  Xu, Lili;  Gao, Lixin;  Li, Jia
收藏  |  浏览/下载:4/0  |  提交时间:2020/07/01
Design, synthesis and structure-activity relationship optimization of phenanthridine derivatives as new Wnt/beta-catenin signalling pathway agonists 期刊论文
BIOORGANIC CHEMISTRY, 2019, 卷号: 84, 页码: 285-294
作者:  Chen, Duo-zhi;  Yang, Bi-juan;  He, Xiao-li;  Fan, Shi-rui;  Cai, Jie-yun
收藏  |  浏览/下载:113/0  |  提交时间:2019/03/18
Synthesis, biological evaluation and molecular docking of benzimidazole grafted benzsulfamide-containing pyrazole ring derivatives as novel tubulin polymerization inhibitors 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2019, 卷号: 27, 期号: 3
作者:  Shi, Tian-Qi;  Wang, Yan-Ting;  Liu, Chang-Hong;  Zhu, Hai-Liang
收藏  |  浏览/下载:8/0  |  提交时间:2019/12/05
Discovery of novel bacterial FabH inhibitors (Pyrazol-Benzimidazole amide derivatives): Design, synthesis, bioassay, molecular docking and crystal structure determination 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 171
作者:  Wang, Yan-Ting;  Shi, Tian-Qi;  Fu, Jie;  Zhu, Hai-Liang
收藏  |  浏览/下载:14/0  |  提交时间:2019/12/05
Synthesis and bioevaluation of diarylpyrazoles as antiproliferative agents 期刊论文
European Journal of Medicinal Chemistry, 2019
作者:  Chao Wang;  Shuang Yang;  Jianan Du;  Jia Ni;  Yue Wu
收藏  |  浏览/下载:7/0  |  提交时间:2019/12/13


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