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Zebrafish (Danio rerio) TR beta- and TTR-based electrochemical biosensors: Construction and application for the evaluation of thyroid-disrupting activity of bisphenols
期刊论文
ENVIRONMENTAL POLLUTION, 2023, 卷号: 330, 页码: 9
作者:
Li, Yuejiao
;
Zhang, Zhenzhong
;
Wang, Jun
;
Shan, Yeqi
;
Tian, Hua
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2023/12/07
Thyroid-disrupting chemicals
Thyroid hormone receptor beta
Transthyretin
In vitro screening Assay
Electrochemical biosensor
Integrated strategy for the screening of cyclooxygenase-2 inhibitors from triterpenoid saponins in Clematis tangutica
期刊论文
PHYTOCHEMICAL ANALYSIS, 2023, 卷号: 34, 期号: 6, 页码: 692
作者:
Wei, Yangfei
;
Chen, Tao
;
Wang, Shuo
;
Shen, Cheng
;
Song, Zhibo
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2023/12/01
The discovery of a novel series of potential ERR alpha inverse agonists based on p-nitrobenzenesulfonamide template for triple-negative breast cancer in vivo
期刊论文
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 2022, 卷号: 37, 期号: 1, 页码: 125-134
作者:
Gao, Zhipei
;
Wang, Tianxiao
;
Li, Rui
;
Du, Yongli
;
Lv, Han
收藏
  |  
浏览/下载:39/0
  |  
提交时间:2022/01/18
ERR alpha
TNBC
p-Nitrobenzenesulfonamide
inverse agonist
Distinct binding kinetics of E-, P- and L-selectins to CD44
期刊论文
FEBS JOURNAL, 2021, 页码: 18
作者:
Li LD(李林达)
;
Ding QH(丁奇寒)
;
Zhou J(周瑾)
;
Wu Y(武亿)
;
Zhang MK(张明坤)
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  |  
浏览/下载:49/0
  |  
提交时间:2022/01/12
binding epitope
binding kinetics
CD44
selectin
Multiple-Tissue and Multilevel Analysis on Differentially Expressed Genes and Differentially Correlated Gene Pairs for HFpEF
期刊论文
FRONTIERS IN GENETICS, 2021, 卷号: 12, 页码: 14
作者:
Zhou, Guofeng
;
Sun, Shaoyan
;
Yuan, Qiuyue
;
Zhang, Run
;
Jiang, Ping
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  |  
浏览/下载:47/0
  |  
提交时间:2021/10/26
heart failure with preserved ejection fraction
differentially expressed genes
differentially correlated gene pairs
differential network
molecular docking
Discovery of Novel Allosteric Modulators Targeting an Extra-Helical Binding Site of GLP-1R Using Structure- and Ligand-Based Virtual Screening
期刊论文
BIOMOLECULES, 2021, 卷号: 11, 期号: 7, 页码: 14
作者:
Zhou, Qingtong
;
Guo, Wanjing
;
Dai, Antao
;
Cai, Xiaoqing
;
Vass, Marton
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  |  
浏览/下载:41/0
  |  
提交时间:2021/08/17
GLP-1R
virtual screening
allosteric modulator
drug discovery
molecular docking
Design, synthesis and pharmacological evaluation of tricyclic derivatives as selective RXFP4 agonists
期刊论文
BIOORGANIC CHEMISTRY, 2021, 卷号: 110, 页码: 17
作者:
Lin, Lin
;
Lin, Guangyao
;
Zhou, Qingtong
;
Bathgate, Ross A. D.
;
Gong, Grace Qun
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  |  
浏览/下载:31/0
  |  
提交时间:2021/08/17
Synthesis
Structure-activity relationship
Relaxin family peptide receptor 4
Selective agonist
Molecular docking
CSConv2d: A 2-D Structural Convolution Neural Network with a Channel and Spatial Attention Mechanism for Protein-Ligand Binding Affinity Prediction
期刊论文
BIOMOLECULES, 2021, 卷号: 11, 期号: 5, 页码: 9
作者:
Wang, Xun
;
Liu, Dayan
;
Zhu, Jinfu
;
Rodriguez-Paton, Alfonso
;
Song, Tao
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2021/12/01
protein-ligand binding affinity
2-D structural CNN
spatial attention mechanism
Ligand-based approach for predicting drug targets and for virtual screening against COVID-19
期刊论文
BRIEFINGS IN BIOINFORMATICS, 2021, 卷号: 22, 期号: 2, 页码: 1053-1064
作者:
Yang, Yanqing
;
Zhu, Zhengdan
;
Wang, Xiaoyu
;
Zhang, Xinben
;
Mu, Kaijie
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2021/11/16
D3Similarity
COVID-19
target prediction
database
virtual screening
Discovery of a new inhibitor targeting PD-L1 for cancer immunotherapy
期刊论文
NEOPLASIA, 2021, 卷号: 23, 期号: 3, 页码: 281-293
作者:
Wang, Fengling
;
Ye, Wenling
;
Wang, Shuang
;
He, Yongxing
;
Zhong, Haiyang
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  |  
浏览/下载:33/0
  |  
提交时间:2021/12/10
PD-1
PD-L1
Inhibitor
APBC
Cancer immunotherapy
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