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科研机构
上海药物研究所 [15]
北京大学 [2]
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南海海洋研究所 [1]
中国科学院大学 [1]
武汉植物园 [1]
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期刊论文 [24]
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P300/CBP inhibition sensitizes mantle cell lymphoma to PI3K delta inhibitor idelalisib
期刊论文
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 13
作者:
Zhou, Xiao-ru
;
Li, Xiao
;
Liao, Li-ping
;
Han, Jie
;
Huang, Jing
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2021/06/11
mantle cell lymphoma
idelalisib
drug resistance
P300
CBP
synergistic drug action
PI3Kδ
epigenetics
P300/CBP inhibition sensitizes mantle cell lymphoma to PI3K delta inhibitor idelalisib
期刊论文
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 13
作者:
Zhou, Xiao-ru
;
Li, Xiao
;
Liao, Li-ping
;
Han, Jie
;
Huang, Jing
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2021/06/11
mantle cell lymphoma
idelalisib
drug resistance
P300
CBP
synergistic drug action
PI3Kδ
epigenetics
A novel virtual screening procedure identifies Pralatrexate as inhibitor of SARS-CoV-2 RdRp and it reduces viral replication in vitro
期刊论文
PLOS COMPUTATIONAL BIOLOGY, 2020, 卷号: 16, 期号: 12, 页码: 20
作者:
Zhang, Haiping
;
Yang, Yang
;
Li, Junxin
;
Wang, Min
;
Saravanan, Konda Mani
收藏
  |  
浏览/下载:38/0
  |  
提交时间:2021/12/01
Identification of SARS-CoV-2 entry inhibitors among already approved drugs
期刊论文
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 7
作者:
Yang, Li
;
Pei, Rong-juan
;
Li, Heng
;
Ma, Xin-na
;
Zhou, Yu
收藏
  |  
浏览/下载:41/0
  |  
提交时间:2020/12/24
COVID-19
SARS-CoV-2
virus entry inhibitors
high throughput screening assay
approved drug library
histamine receptor antagonists
clemastine
USP28 and USP25 are downregulated by Vismodegib in vitro and in colorectal cancer cell lines
期刊论文
FEBS JOURNAL, 2020, 页码: 18
作者:
Wang, Hui
;
Meng, Qian
;
Ding, Yiluan
;
Xiong, Muya
;
Zhu, Mengying
收藏
  |  
浏览/下载:84/0
  |  
提交时间:2020/12/24
colorectal cancer
HDX-MS
inhibitor
USP25
USP28
Vismodegib
Deep Learning Based Drug Screening for Novel Coronavirus 2019-nCov
期刊论文
INTERDISCIPLINARY SCIENCES-COMPUTATIONAL LIFE SCIENCES, 2020, 页码: 9
作者:
Zhang, Haiping
;
Saravanan, Konda Mani
;
Yang, Yang
;
Hossain, Md Tofazzal
;
Li, Junxin
收藏
  |  
浏览/下载:163/0
  |  
提交时间:2020/12/10
Coronavirus
Deep learning
Drug screening
Homology modeling
3C-like protease
Nitazoxanide, an anti-parasitic drug, efficiently ameliorates learning and memory impairments in AD model mice
期刊论文
ACTA PHARMACOLOGICA SINICA, 2019, 卷号: 40, 期号: 10, 页码: 1279-1291
作者:
Fan, Lei
;
Qiu, Xiao-xia
;
Zhu, Zhi-yuan
;
Lv, Jian-lu
;
Lu, Jian
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2020/07/01
Alzheimer's disease
nitazoxanide
autophagy
inflammation
APP/PS1 transgenic mice
Sodium chloride (NaCl) potentiates digoxin-induced anti-tumor activity in small cell lung cancer
期刊论文
CANCER BIOLOGY & THERAPY, 2019, 卷号: 20, 期号: 1, 页码: 52-64
作者:
Deng, Ke
;
Shen, Jiawei
;
Wang, Wei
;
Li, Ming
;
Li, Hong
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2020/03/31
small cell lung cancer
digoxin
NaCl
cardiac glycosides
ATP1A1
PDE3A inhibitor anagrelide activates death signaling pathway genes and synergizes with cell death-inducing cytokines to selectively inhibit cancer cell growth
期刊论文
AMERICAN JOURNAL OF CANCER RESEARCH, 2019, 卷号: 9, 期号: 9, 页码: 1905-+
作者:
An, Ran
;
Liu, Jueyu
;
He, Jing
;
Wang, Fei
;
Zhang, Qing
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2020/07/01
Anagrelide
PDE3A
SLFN12
cancer
cytokine
Screening and Identification of Lassa Virus Entry Inhibitors from an FDA-Approved Drug Library
期刊论文
JOURNAL OF VIROLOGY, 2018, 卷号: 92, 期号: 16, 页码: 14
作者:
Xiao, Gengfu
;
Wang, Wei
;
Liu, Yang
;
Zhang, Guangshun
;
Wang, Shaobo
收藏
  |  
浏览/下载:68/0
  |  
提交时间:2018/12/29
Lassa virus (LASV)
glycoprotein complex (GPC)
lacidipine
phenothrin
membrane fusion
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