CORC

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Repressing MYC by targeting BET synergizes with selective inhibition of PI3K alpha against B cell lymphoma 期刊论文
CANCER LETTERS, 2022, 卷号: 524, 页码: 206-218
作者:  Chen, Zi-qi;  Cao, Zhe-rui;  Wang, Yi;  Zhang, Xi;  Xu, Lan
收藏  |  浏览/下载:53/0  |  提交时间:2021/12/16
CYH33  MYC  P300  BET  B cell lymphoma  PI3K  
W2476 represses TXNIP transcription via dephosphorylation of FOXO1 at Ser319 期刊论文
CHEMICAL BIOLOGY & DRUG DESIGN, 2021, 页码: 11
作者:  Zhong, Li;  Liu, Qing;  Liu, Qiaofeng;  Zhang, Shikai;  Cao, Yongbing
收藏  |  浏览/下载:21/0  |  提交时间:2021/05/24
SL010110, a lead compound, inhibits gluconeogenesis via SIRT2-p300-mediated PEPCK1 degradation and improves glucose homeostasis in diabetic mice 期刊论文
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 13
作者:  Ren, Yu-ran;  Ye, Yang-liang;  Feng, Ying;  Xu, Ti-fei;  Shen, Yu
收藏  |  浏览/下载:22/0  |  提交时间:2021/05/24
Design, synthesis, and biological evaluation of a new class of histone acetyltransferase p300 inhibitors (vol 180, pg 171, 2019) 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 186, 页码: 2
作者:  Liu, Ruiqi;  Zhang, Zhuqing;  Yang, Hong;  Zhou, Kaixin;  Geng, Meiyu
收藏  |  浏览/下载:14/0  |  提交时间:2020/07/01
Design, synthesis, and biological evaluation of a new class of histone acetyltransferase p300 inhibitors 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 180, 页码: 171-190
作者:  Liu, Ruiqi;  Zhang, Zhuqing;  Yang, Hong;  Zhou, Kaixin;  Geng, Meiyu
收藏  |  浏览/下载:8/0  |  提交时间:2020/07/01
Laminar shear stress alters endothelial KCa2.3 expression in H9c2 cells partially via regulating the PI3K/Akt/p300 axis 期刊论文
INTERNATIONAL JOURNAL OF MOLECULAR MEDICINE, 2019, 卷号: 43, 期号: 3
作者:  Li, Guojian;  Yang, Qionghui;  Yang, Yong;  Yang, Guokai;  Wan, Jia
收藏  |  浏览/下载:17/0  |  提交时间:2019/12/04
Functional Studies of Transcriptional Cofactors via Microinjection-Mediated Gene Editing in Xenopus. 期刊论文
Methods in molecular biology, 2019, 卷号: 1874, 页码: 507-524
作者:  Shibata Yuki;  Bao Lingyu;  Fu Liezhen;  Shi Bingyin;  Shi Yun-Bo
收藏  |  浏览/下载:23/0  |  提交时间:2019/11/19
Garcinol inhibits esophageal cancer metastasis by suppressing the p300 and TGF-β1 signaling pathways. 期刊论文
Acta pharmacologica Sinica, 2019
作者:  Wang Jing;  Wu Man;  Zheng Dan;  Zhang Hong;  Lv Yue
收藏  |  浏览/下载:8/0  |  提交时间:2019/12/05
MicroRNA-377 exerts a potent suppressive role in osteosarcoma through the involvement of the histone acetyltransferase 1-mediated Wnt axis 期刊论文
JOURNAL OF CELLULAR PHYSIOLOGY, 2019, 卷号: 234, 期号: 12
作者:  Li, Fang;  Xia, Peng;  Gu, Rui;  Zhang, Wei;  Shao, Liwei
收藏  |  浏览/下载:4/0  |  提交时间:2019/12/05
Cucurbit[8]uril-assisted peptide assembly for feasible electrochemical assay of histone acetyltransferase activity 期刊论文
ANALYTICAL AND BIOANALYTICAL CHEMISTRY, 2019, 卷号: 411, 页码: 387-393
作者:  Miao, Xiangyang[1];  Wang, Yang[2];  Gu, Zhun[3];  Mao, Dongsheng[4];  Ning, Limin[5]
收藏  |  浏览/下载:32/0  |  提交时间:2019/04/22


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