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上海药物研究所 [12]
长春应用化学研究所 [9]
复旦大学上海医学院 [7]
上海中医药大学 [7]
北京大学 [6]
山东大学 [6]
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期刊论文 [116]
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Identification of phosphodiesterase-4 as the therapeutic target of arctigenin in alleviating psoriatic skin inflammation
期刊论文
JOURNAL OF ADVANCED RESEARCH, 2021, 卷号: 33, 页码: 241-251
作者:
Li, Heng
;
Zhang, Xianglei
;
Xiang, Caigui
;
Feng, Chunlan
;
Fan, Chen
收藏
  |  
浏览/下载:86/0
  |  
提交时间:2021/11/04
PDE4
Arctigenin
Psoriasis
Inflammation
MALDI-MS imaging of lipids and small molecules in rat brain tissue based on graphene oxide film pre-coated matrix
期刊论文
INTERNATIONAL JOURNAL OF MASS SPECTROMETRY, 2021, 卷号: 464, 页码: 8
作者:
Xu, Yang
;
Deng, Yingzhi
;
Ye, Rongrong
;
Gong, Can
;
Liu, Zhaoxin
收藏
  |  
浏览/下载:61/0
  |  
提交时间:2021/06/11
Single-layer graphene oxide film
Matrix-assisted laser desorption ionization-mass spectrometry imaging
Phospholipids
Pre-coated matrix
Inhibition of PDE4 by apremilast attenuates skin fibrosis through directly suppressing activation of M1 and T cells
期刊论文
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 11
作者:
Lu, Qiu-kai
;
Fan, Chen
;
Xiang, Cai-gui
;
Wu, Bing
;
Lu, Hui-min
收藏
  |  
浏览/下载:57/0
  |  
提交时间:2021/06/11
PDE4
apremilast
skin fibrosis
macrophages
Design, synthesis, and biological evaluation of tetrahydroisoquinolines derivatives as novel, selective PDE4 inhibitors for antipsoriasis treatment
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 211, 页码: 20
作者:
Zhang, Rui
;
Li, Heng
;
Zhang, Xianglei
;
Li, Jian
;
Su, Haixia
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2021/05/24
PDE4 inhibitors
Tetrahydroisoquinoline
Antipsoriasis
Small molecules targeting the innate immune cGAS-STING-TBK1 signaling pathway
期刊论文
ACTA PHARMACEUTICA SINICA B, 2020, 卷号: 10, 期号: 12, 页码: 2272-2298
作者:
Ding, Chunyong
;
Song, Zilan
;
Shen, Ancheng
;
Chen, Tingting
;
Zhang, Ao
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2021/05/24
Immunotherapy
Anti-tumor
cGAS
STING
TBK1
Small molecule modulators
Discovery of a potent and selective adenylyl cyclase type 8 agonist by docking-based virtual screening
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2020, 卷号: 30, 期号: 2, 页码: 7
作者:
Weng, Zhiying
;
Xu, Guowei
;
Chen, Dingyuan
;
Yang, Yaqing
;
Song, Gao
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2020/03/18
Adenylyl cyclases
Homology modeling
Consensus scoring
Molecular dynamics simulation
Virtual screening
Biological evaluation
Identification of functional lncRNAs based on competing endogenous RNA network in osteoblast differentiation
期刊论文
JOURNAL OF CELLULAR PHYSIOLOGY, 2019, 页码: 13
作者:
Hong, Shuai
;
Hu, Supei
;
Kang, Zhengyang
;
Liu, Zhiguo
;
Yang, Weibin
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  |  
浏览/下载:80/0
  |  
提交时间:2019/12/10
ceRNA
feedback loops
lncRNA
osteoblast differentiation
Ligand-induced activation of ERK1/2 signaling by constitutively active G(s)-coupled 5-HT receptors
期刊论文
ACTA PHARMACOLOGICA SINICA, 2019, 卷号: 40, 期号: 9, 页码: 1157-1167
作者:
Liu, Ping
;
Yin, Yu-ling
;
Wang, Ting
;
Hou, Li
;
Wang, Xiao-xi
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2020/07/01
5-HT4R
5-HT6R
5-HT7AR
5-HT
ERK1/2
G(s)
beta-arrestin
Fyn
Src
cAMP-modulated biomimetic ionic nanochannels based on a smart polymer
期刊论文
JOURNAL OF MATERIALS CHEMISTRY B, 2019, 卷号: 7, 期号: 23, 页码: 3710-3715
作者:
Chen, Zhixiang
;
Sun, Taolei
;
Qing, Guangyan
收藏
  |  
浏览/下载:70/0
  |  
提交时间:2019/12/02
Pulsed electromagnetic fields promote bone formation by activating the sAC-cAMP-PKA-CREB signaling pathway
期刊论文
JOURNAL OF CELLULAR PHYSIOLOGY, 2019, 卷号: 234, 期号: 3, 页码: 2807-2821
作者:
Wang, Yuan-Yuan
;
Pu, Xiu-Ying
;
Shi, Wen-Gui
;
Fang, Qing-Qing
;
Chen, Xin-Ru
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2019/11/15
bone formation
cAMP
osteoblast
PEMFs
soluble AC
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