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上海药物研究所 [5]
西北高原生物研究所 [1]
海洋研究所 [1]
合肥物质科学研究院 [1]
西安光学精密机械研究... [1]
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期刊论文 [9]
发表日期
2021 [9]
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Internal Wave Imprints on Temperature Fluctuations as Revealed by Rapid-Sampling Deep Profiling Floats
期刊论文
JOURNAL OF GEOPHYSICAL RESEARCH-OCEANS, 2021, 卷号: 126, 期号: 12, 页码: 20
作者:
Gao, Zhiyuan
;
Chen, Zhaohui
;
Huang, Xiaodong
;
Xu, Zhenhua
;
Yang, Haiyuan
收藏
  |  
浏览/下载:40/0
  |  
提交时间:2022/02/18
internal wave
temperature fluctuations
deep floats
deep ocean
Classification of Pneumonia Images Based on Improved VGG19 Convolutional Neural Network (Invited)
期刊论文
Guangzi Xuebao/Acta Photonica Sinica, 2021, 卷号: 50, 期号: 10
作者:
Xiong, Feng
;
He, Di
;
Liu, Yujie
;
Qi, Meijie
;
Gao, Peng
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2021/12/13
Pneumonia image classification
Convolution neural network
Deep learning
VGG19
Support vector machine
eXtreme Gradient Boosting
Rational Design and Development of Novel CDK9 Inhibitors for the Treatment of Acute Myeloid Leukemia
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 19, 页码: 14647-14663
作者:
Han, Xu
;
Song, Ning
;
Saidahmatov, Abdusaid
;
Wang, Peipei
;
Wang, Yong
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  |  
浏览/下载:17/0
  |  
提交时间:2021/12/16
Synthesis and Evaluation of 3-(Indol-3-yl)-4-(Pyrazolo[3,4-c]Pyridazin-3-yl)-Maleimides as Potent Mutant Isocitrate Dehydrogenase-1 Inhibitors
期刊论文
PHARMACEUTICAL CHEMISTRY JOURNAL, 2021, 卷号: 55, 期号: 7, 页码: 655-664
作者:
Xu, Jianghong
;
Hu, Yuanyuan
;
Liu, Xiaoqi
;
Gao, Anhui
;
Gao, Lixin
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  |  
浏览/下载:37/0
  |  
提交时间:2021/12/01
IDH1-R132H inhibitors
synthesis
biological activity
docking
3-(indol-3-yl)-4-(pyrazolo-[3
4-c]pyridazin-3-yl)-maleimides
Synthesis and Protein Tyrosine Phosphatase 1B (PTP1B) Inhibitory Activity Evaluation of Novel N-Acylhydrazone Derivatives Containing Carbazole and Aromatic Ring/Aromatic Fused Heterocycle
期刊论文
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2021, 卷号: 41, 期号: 9, 页码: 3593-3607
作者:
Li Yingjun
;
Lin Ledi
;
Liu Jihong
;
Gao Lixin
;
Sheng Li
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  |  
浏览/下载:19/0
  |  
提交时间:2021/12/01
PTP1B inhibitor
carbazole
N-actylhydrazone
synthesis
molecular docking
Synthesis of 5-Phenyl-1,3,4-thiadiazole Derivatives and Their Biochemical Evaluation against Src Homology 2 Domain-Containing Protein Tyrosine Phosphatase 1 (SHP1)
期刊论文
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2021, 卷号: 41, 期号: 8, 页码: 3097-3105
作者:
Yu Lijie
;
Feng Bo
;
Wang Zhijia
;
Gao Lixin
;
Zhang Chun
收藏
  |  
浏览/下载:242/0
  |  
提交时间:2021/11/04
5-phenyl-1,3,4-thiadiazole derivatives
Src homology 2 domain-containing protein tyrosine phosphatase 1 (SHP1)
inhibitors
structure-activity relationships
Synthesis and Protein Tyrosine Phosphatase 1B (PTP1B) Inhibitory Activity Evaluation of Novel Arylaminoacetylhydrazone Derivatives Containing Carbazole Moiety
期刊论文
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2021, 卷号: 41, 期号: 8, 页码: 3157-3170
作者:
Li Yingjun
;
Lin Ledi
;
Jin Kun
;
Gao Lixin
;
Sheng Li
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2021/11/04
protein tyrosine phosphatase 1B (PTP1B) inhibitor
carbazole
arylaminoacetylhydrazone
synthesis
molecular docking
Guidelines for the use and interpretation of assays for monitoring autophagy (4th edition)
期刊论文
AUTOPHAGY, 2021, 卷号: 17
作者:
Klionsky, Daniel J.
;
Abdel-Aziz, Amal Kamal
;
Abdelfatah, Sara
;
Abdellatif, Mahmoud
;
Abdoli, Asghar
收藏
  |  
浏览/下载:268/0
  |  
提交时间:2021/05/31
Autophagosome
cancer
flux
LC3
lysosome
macroautophagy
neurodegeneration
phagophore
stress
vacuole
Structure and immunomodulatory activity of a water-soluble alpha-glucan from Hirsutella sinensis mycelia
期刊论文
INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES, 2021, 卷号: 189
作者:
Rong, Lin
;
Li, Guoqiang
;
Zhang, Yuxia
;
Xiao, Yuancan
;
Qiao, Yajun
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2021/11/18
Hirsutella sinensis
alpha-Glucan
Structure
Immunomodulatory activity
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