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科研机构
山东大学 [11]
内容类型
期刊论文 [11]
发表日期
2015 [11]
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共11条,第1-10条
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发表日期:2015
专题:山东大学
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Design, Synthesis, and Antitumor Evaluation of Novel Histone Deacetylase Inhibitors Equipped with a Phenylsulfonylfuroxan Module as a Nitric Oxide Donor
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2015, 卷号: 58, 期号: 10, 页码: 4325-4338
作者:
Duan, Wenwen
;
Li, Jin
;
Inks, Elizabeth S.
;
Chou, C. James
;
Jia, Yuping
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2019/12/17
Development of 3-hydroxycinnamamide-based HDAC inhibitors with potent in vitro and in vivo anti-tumor activity
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2015, 卷号: 89, 页码: 628-637
作者:
Li, Xiaoyang
;
Hou, Jinning
;
Li, Xiaoguang
;
Jiang, Yuqi
;
Liu, Xueliang
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2019/12/17
HDACs
HDACIs
Anti-tumor drugs
Antiproliferative activity
In vivo
oral activity
Synthesis and biological evaluation of novel histone deacetylases inhibitors with nitric oxide releasing activity
期刊论文
Bioorganic and medicinal chemistry, 2015, 卷号: 23, 期号: 15, 页码: 4481-4488
作者:
Duan, Wenwen
;
Hou, Jinning
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2019/12/17
HDAC inhibitor
Nitric oxide
Benzofuroxan
Multifunctional drugs
Epigenetic
Enhanced anticancer activity of 5-FU in combination with Bestatin: Evidence in human tumor-derived cell lines and an H22 tumor-bearing mouse
期刊论文
Drug discoveries & therapeutics, 2015, 卷号: 9, 期号: 1
作者:
Li, Jin
;
Wang, Xuejian
;
Hou, Jinning
;
Huang, Yongxue
;
Zhang, Yingjie
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2019/12/17
Trend of Histone Deacetylase Inhibitors in Cancer Therapy: Isoform Selectivity or Multitargeted Strategy
期刊论文
Medicinal research reviews, 2015, 卷号: 35, 期号: 1, 页码: 63-84
作者:
Zhang, Lei
;
Han, Yantao
;
Jiang, Qixiao
;
Wang, Chunbo
;
Chen, Xuehong
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2019/12/17
histone deacetylase
inhibitors
selectivity
multitargeted
bifunctional molecule
Development of N-hydroxybenzamide derivatives with indole-containing cap group as histone deacetylases inhibitors
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2015, 卷号: 23, 期号: 19, 页码: 6258-6270
作者:
Li, Xiaoyang
;
Wu, Jingde
;
Li, Xiaoguang
;
Mu, Weiwei
;
Liu, Xueliang
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2019/12/17
HDACs
HDACIs
HDAC inhibitory activity
Antiproliferative activity
Class I and class IIa cellular activity
Design, synthesis, and antitumor evaluation of histone deacetylase inhibitors with L-phenylglycine scaffold
期刊论文
DRUG DESIGN DEVELOPMENT AND THERAPY, 2015, 卷号: 9, 页码: 5553-5567
作者:
Zhang, Yingjie
;
Li, Xiaoguang
;
Hou, Jinning
;
Huang, Yongxue
;
Xu, Wenfang
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2019/12/17
phenylglycine
histone deacetylases
inhibitor
antitumor
Enhancing the Sensitivity of Pharmacophore-Based Virtual Screening by Incorporating Customized ZBG Features: A Case Study Using Histone Deacetylase 8
期刊论文
Journal of chemical information and modeling, 2015, 卷号: 55, 期号: 4, 页码: 861-871
作者:
Hou, Xuben
;
Du, Jintong
;
Liu, Renshuai
;
Zhou, Yi
;
Li, Minyong
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2019/12/17
Design, synthesis and preliminary biological evaluation of indoline-2,3-dione derivatives as novel HDAC inhibitors
期刊论文
Bioorganic and medicinal chemistry, 2015, 卷号: 23, 期号: 15, 页码: 4728-4736
作者:
Jin, Kang
;
Li, Shanshan
;
Li, Xiaoguang
;
Zhang, Jian
;
Xu, Wenfang
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2019/12/17
Indoline-2
3-dione derivatives
HDAC inhibitors
Synthesis
Biological evaluation
QSAR
Design, Synthesis, and Preliminary Activity Evaluation of Novel Pyrimidine Derivatives as Acid Pump Antagonists
期刊论文
Chemical biology and drug design, 2015, 卷号: 85, 期号: 3, 页码: 306-314
作者:
Song, Weiguo
;
Zhang, Xiaopan
;
Li, Shutao
;
Xu, Wenfang
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2019/12/17
acid pump antagonists
bioisosterism
gastric antisecretory activity
pyrimidine derivatives
synthesis
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