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上海药物研究所 [64]
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期刊论文 [64]
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2021 [1]
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Rh-Catalyzed C-H alkylation enabling modular synthesis of CF3-substituted benzannulated macrocyclic inhibitors of B cell responses dagger
期刊论文
ORGANIC & BIOMOLECULAR CHEMISTRY, 2021, 页码: 6
作者:
Sun, Tao
;
He, Shijun
;
Xu, Zhongliang
;
Zuo, Jianping
;
Yu, Yang
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2021/05/24
Structure-based design, synthesis and bioactivity evaluation of macrocyclic inhibitors of mutant isocitrate dehydrogenase 2 (IDH2) displaying activity in acute myeloid leukemia cells
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 203, 页码: 19
作者:
Che, Jinxin
;
Huang, Feng
;
Zhang, Mengmeng
;
Xu, Gaoya
;
Qu, Bingxue
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2020/12/21
Metabolic pathways
Isocitrate dehydrogenase 2
Conformational restriction
Macrocyclic derivatives
Inhibitors
Structure-based design, synthesis and bioactivity evaluation of macrocyclic inhibitors of mutant isocitrate dehydrogenase 2 (IDH2) displaying activity in acute myeloid leukemia cells
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 203, 页码: 19
作者:
Che, Jinxin
;
Huang, Feng
;
Zhang, Mengmeng
;
Xu, Gaoya
;
Qu, Bingxue
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2020/12/21
Metabolic pathways
Isocitrate dehydrogenase 2
Conformational restriction
Macrocyclic derivatives
Inhibitors
Quantum Mechanical-NMR-Aided Configuration and Conformation of Two Unreported Macrocycles Isolated from the Soft Coral Lobophytum sp.: Energy Calculations versus Coupling Constants
期刊论文
ORGANIC LETTERS, 2020, 卷号: 22, 期号: 11, 页码: 4093-4096
作者:
Li, Song-Wei
;
Cuadrado, Cristina
;
Yao, Li-Gong
;
Daranas, Antonio Hernandez
;
Guo, Yue-Wei
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  |  
浏览/下载:27/0
  |  
提交时间:2020/12/24
Pd-Catalyzed Decarboxylative Olefination: Stereoselective Synthesis of Polysubstituted Butadienes and Macrocyclic P-glycoprotein Inhibitors
期刊论文
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2020, 卷号: 142, 期号: 22, 页码: 9982-9992
作者:
Song, Bichao
;
Xie, Peipei
;
Li, Yingzi
;
Hao, Jiping
;
Wang, Lu
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2020/12/24
A modular biomimetic strategy for the synthesis of macrolide P-glycoprotein inhibitors via Rh-catalyzed C-H activation
期刊论文
NATURE COMMUNICATIONS, 2020, 卷号: 11, 期号: 1, 页码: 8
作者:
Chen, Lu
;
Quan, Haitian
;
Xu, Zhongliang
;
Wang, Hao
;
Xia, Yuanzhi
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  |  
浏览/下载:17/0
  |  
提交时间:2020/12/24
Rhodium(III)-Catalyzed C-H Alkenylation: Access to Maleimide-Decorated Tryptophan and Tryptophan-Containing Peptides
期刊论文
ORGANIC LETTERS, 2020, 卷号: 22, 期号: 4, 页码: 1535-1541
作者:
Peng, Jingjing
;
Li, Chunpu
;
Khamrakulov, Mirzadavlat
;
Wang, Jiang
;
Liu, Hong
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  |  
浏览/下载:20/0
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提交时间:2020/07/01
Conformation of the Macrocyclic Drug Lorlatinib in Polar and Nonpolar Environments: A MD Simulation and NMR Study
期刊论文
ACS OMEGA, 2019, 卷号: 4, 期号: 26, 页码: 22245-22250
作者:
Peng, Cheng
;
Atilaw, Yoseph
;
Wang, Jinan
;
Xu, Zhijian
;
Poongavanam, Vasanthanathan
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  |  
浏览/下载:23/0
  |  
提交时间:2020/07/01
Exploration of novel macrocyclic dipeptide N-benzyl amides as proteasome inhibitors
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 164, 页码: 423-439
作者:
Yu, Jianjun
;
Liu, Jieyu
;
Li, Daqiang
;
Xu, Lei
;
Hong, Duidui
收藏
  |  
浏览/下载:0/0
  |  
提交时间:2020/07/01
Proteasome inhibitors
Macrocyclic dipeptides
N-Benzyl amides
Metabolic stability
The value of universally available raw NMR data for transparency, reproducibility, and integrity in natural product research
期刊论文
NATURAL PRODUCT REPORTS, 2019, 卷号: 36, 期号: 1, 页码: 35-107
作者:
McAlpine, James B.
;
Chen, Shao-Nong
;
Kutateladze, Andrei
;
MacMillan, John B.
;
Appendino, Giovanni
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  |  
浏览/下载:25/0
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提交时间:2020/07/01
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