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科研机构
上海药物研究所 [119]
内容类型
期刊论文 [119]
发表日期
2019 [119]
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共119条,第1-10条
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发表日期:2019
专题:上海药物研究所
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Discovery of a Highly Selective and Potent kappa Opioid Receptor Agonist from N-Cyclopropylmethyl-7 alpha-phenyl-6,14-endoethanotetrahydronorthebaines with Reduced Central Nervous System (CNS) Side Effects Navigated by the Message-Address Concept
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 24, 页码: 11054-11070
作者:
Xiao, Li
;
Wang, Yujun
;
Zhang, Mumei
;
Wu, Weiwei
;
Kong, Linghui
收藏
  |  
浏览/下载:92/0
  |  
提交时间:2020/07/01
Imaging Tumorous Methylglyoxal by an Activatable Near-Infrared Fluorescent Probe for Monitoring Glyoxalase 1 Activity
期刊论文
ANALYTICAL CHEMISTRY, 2019, 卷号: 91, 期号: 24, 页码: 15577-15584
作者:
Ding, Chunyong
;
Wang, Fengyang
;
Dang, Yijing
;
Xu, Zhiai
;
Li, Lingling
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2020/07/01
DZ2002 ameliorates fibrosis, inflammation, and vasculopathy in experimental systemic sclerosis models
期刊论文
ARTHRITIS RESEARCH & THERAPY, 2019, 卷号: 21, 期号: 1, 页码: 15
作者:
Zhang, Zongwang
;
Wu, Yanwei
;
Wu, Bing
;
Qi, Qing
;
Li, Heng
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2020/07/01
Systemic sclerosis
SAHH inhibitor
Fibrosis
Inflammation
Vasculopathy
TGF-beta
Structure elucidation and anti-tumor activity in vivo of a polysaccharide from spores of Ganoderma lucidum (Fr.) Karst
期刊论文
INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES, 2019, 卷号: 141, 页码: 693-699
作者:
Fu, Youli
;
Shi, Lei
;
Ding, Kan
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2020/07/01
Polysaccharide
Anti-tumor activity
beta-Glucan
Structure
Ganoderma lucidum
Metabolic Evaluation of MYCN-Amplified Neuroblastoma by 4-[F-18]FGln PET Imaging
期刊论文
MOLECULAR IMAGING AND BIOLOGY, 2019, 卷号: 21, 期号: 6, 页码: 1117-1126
作者:
Li, Chao
;
Huang, Shuo
;
Guo, Jun
;
Wang, Cheng
;
Huang, Zhichao
收藏
  |  
浏览/下载:38/0
  |  
提交时间:2020/07/01
Glutamine
PET
MYCN
ASCT2
Neuroblastoma
Design, synthesis, and biological evaluation of thieno[3,2-d]pyrimidine derivatives as potential simplified phosphatidylinositol 3-kinase alpha inhibitors
期刊论文
CHEMICAL BIOLOGY & DRUG DESIGN, 2019, 卷号: 94, 期号: 6, 页码: 2013-2022
作者:
Yang, Xiuyan
;
Deng, Meng
;
Zhang, Xi
;
Wang, Yi
;
Song, Kun
收藏
  |  
浏览/下载:75/0
  |  
提交时间:2020/07/01
PI3K alpha inhibitors
proliferation inhibition
thieno[3
2-d]pyrimidine derivatives
Selective activation of TWIK-related acid-sensitive K+ 3 subunit-containing channels is analgesic in rodent models
期刊论文
SCIENCE TRANSLATIONAL MEDICINE, 2019, 卷号: 11, 期号: 519, 页码: 12
作者:
Liao, Ping
;
Qiu, Yunguang
;
Mo, Yiqing
;
Fu, Jie
;
Song, Zhenpeng
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2020/07/01
Effects of traditional Chinese medicine formula Le-Cao-Shi on hepatitis B: In vivo and in vitro studies
期刊论文
JOURNAL OF ETHNOPHARMACOLOGY, 2019, 卷号: 244, 页码: 10
作者:
Zhao, Qing
;
Ren, Xia
;
Chen, Min
;
Yue, Shi-Jun
;
Zhang, Meng-Qi
收藏
  |  
浏览/下载:43/0
  |  
提交时间:2020/07/01
Traditional Chinese medicine
Formula Le-Cao-Shi
Hepatitis B virus
Anti-Hepatitis B
GIAT4RA functions as a tumor suppressor in non-small cell lung cancer by counteracting Uchl3-mediated deubiquitination of LSH
期刊论文
ONCOGENE, 2019, 卷号: 38, 期号: 46, 页码: 7133-7145
作者:
Yang, Rui
;
Liu, Na
;
Chen, Ling
;
Jiang, Yiqun
;
Shi, Ying
收藏
  |  
浏览/下载:49/0
  |  
提交时间:2020/07/01
TRAIL-based gene delivery and therapeutic strategies
期刊论文
ACTA PHARMACOLOGICA SINICA, 2019, 卷号: 40, 期号: 11, 页码: 1373-1385
作者:
Zhong, Hui-hai
;
Wang, Hui-yuan
;
Li, Jian
;
Huang, Yong-zhuo
收藏
  |  
浏览/下载:115/0
  |  
提交时间:2020/07/01
TRAIL
gene delivery
gene therapy
DNA
drug delivery systems
non-viral vectors
cancer therapy
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