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Discovery and Development of a Potent, Selective, and Orally Bioavailable CHK1 Inhibitor Candidate: 5-((4-((3-Amino-3-methylbutyl)amino)-5-(trifluoromethyl)pyrimidin-2-yl)amino)picolinonitrile 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 20, 页码: 15069-15090
作者:  Jin, Tingting;  Xu, Lei;  Wang, Peipei;  Hu, Xiaobei;  Zhang, Runyuan
收藏  |  浏览/下载:20/0  |  提交时间:2022/01/04
Rational Design and Development of Novel CDK9 Inhibitors for the Treatment of Acute Myeloid Leukemia 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 19, 页码: 14647-14663
作者:  Han, Xu;  Song, Ning;  Saidahmatov, Abdusaid;  Wang, Peipei;  Wang, Yong
收藏  |  浏览/下载:15/0  |  提交时间:2021/12/16
Discovery of thalidomide-based PROTAC small molecules as the highly efficient SHP2 degraders 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 218, 页码: 14
作者:  Yang, Xiangbo;  Wang, Zhijia;  Pei, Yuan;  Song, Ning;  Xu, Lei
收藏  |  浏览/下载:37/0  |  提交时间:2021/08/17
Discovery of (R)-5-((5-(1-methyl-1H-pyrazol-4-yl)-4-(methylamino) pyrimidin-2-yl)amino)-3-(piperidin-3-yloxy)picolinonitrile, a novel CHK1 inhibitor for hematologic malignancies 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 173, 页码: 44-62
作者:  Tong, Lexian;  Song, Pinrao;  Jiang, Kailong;  Xu, Lei;  Jin, Tingting
收藏  |  浏览/下载:19/0  |  提交时间:2020/07/01
PM2.5 induced pulmonary fibrosis in vivo and in vitro 期刊论文
ECOTOXICOLOGY AND ENVIRONMENTAL SAFETY, 2019, 卷号: 171
作者:  Xu, Zihan;  Li, Zilin;  Liao, Ziyi;  Gao, Sumeng;  Hua, Li
收藏  |  浏览/下载:13/0  |  提交时间:2019/12/05
CagA increases DNA methylation and decreases PTEN expression in human gastric cancer 期刊论文
MOLECULAR MEDICINE REPORTS, 2019, 卷号: 19, 期号: 1
作者:  Zhang, Baogui;  Zhang, Xiaobei;  Jin, Meng;  Hu, Lei;  Zang, Mingde
收藏  |  浏览/下载:27/0  |  提交时间:2019/12/05
Effects of end surface and angle coupling on mode splitting and suppression in a cylindrical microcavity 期刊论文
APPLIED OPTICS, 2019, 卷号: 58, 页码: 1752-1756
作者:  Yan, Ming[1];  Zhang, Xiaobei[2];  Wang, Jiawei[3];  Hou, Fengyu[4];  Yang, Lei[5]
收藏  |  浏览/下载:3/0  |  提交时间:2019/04/22
Asymmetric Total Synthesis of -Strychnine 期刊论文
Organic Letters, 2019, 卷号: Vol.21 No.1, 页码: 252-255
作者:  Liping He;  Xiaobei Wang;  Xiaoqing Wu;  Zhaoxiang Meng;  Xin Peng
收藏  |  浏览/下载:10/0  |  提交时间:2019/02/25
Thermodynamic design and performance calculation of the thermochemical reformers (Open Access) 期刊论文
Energies, 2019, 卷号: 12, 期号: 19
作者:  Pan, Fumin;  Cheng, Xiaobei;  Wu, Xin;  Wang, Xin;  Gong, Jingfeng
收藏  |  浏览/下载:4/0  |  提交时间:2019/12/05
TFAP2C-Activated MALAT1 Modulates the Chemoresistance of Docetaxel-Resistant Lung Adenocarcinoma Cells. 期刊论文
Molecular therapy. Nucleic acids, 2019, 卷号: Vol.14, 页码: 567-582
作者:  Jing Chen;  Xiaobei Liu;  Yichen Xu;  Kai Zhang;  Jiayuan Huang
收藏  |  浏览/下载:28/0  |  提交时间:2019/12/13


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