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上海药物研究所 [5]
广州生物医药与健康研... [2]
暨南大学 [2]
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期刊论文 [9]
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2021 [2]
2020 [1]
2018 [2]
2015 [4]
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Chemistry [2]
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Discovery of a novel third-generation EGFR inhibitor and identification of a potential combination strategy to overcome resistance (vol 19, 90, 2020)
期刊论文
MOLECULAR CANCER, 2021, 卷号: 20, 期号: 1, 页码: 1
作者:
Zhang, Tao
;
Qu, Rong
;
Chan, Shingpan
;
Lai, Mengzhen
;
Tong, Linjiang
收藏
  |  
浏览/下载:57/0
  |  
提交时间:2021/11/04
Correction to: Discovery of a novel third-generation EGFR inhibitor and identification of a potential combination strategy to overcome resistance
期刊论文
Molecular Cancer, 2021, 卷号: 20, 期号: 1
作者:
Zhang,Tao
;
Qu,Rong
;
Chan,Shingpan
;
Lai,Mengzhen
;
Tong,Linjiang
收藏
  |  
浏览/下载:41/0
  |  
提交时间:2021/11/04
Discovery of a novel third-generation EGFR inhibitor and identification of a potential combination strategy to overcome resistance
期刊论文
MOLECULAR CANCER, 2020, 卷号: 19, 期号: 1, 页码: 15
作者:
Zhang, Tao
;
Qu, Rong
;
Chan, Shingpan
;
Lai, Mengzhen
;
Tong, Linjiang
收藏
  |  
浏览/下载:39/0
  |  
提交时间:2020/07/01
Non-small cell lung cancer (NSCLC)
EGFR T790M
Small-molecule inhibitor
Drug resistance
Ack1
Discovery of JND3229 as a New EGFR(C797S) Mutant Inhibitor with In Vivo Monodrug Efficacy
期刊论文
ACS MEDICINAL CHEMISTRY LETTERS, 2018, 卷号: 9, 期号: 11, 页码: 1123-1127
作者:
Lu, Xiaoyun
;
Zhang, Tao
;
Zhu, Su-Jie
;
Xun, Qiuju
;
Tong, Lingjiang
收藏
  |  
浏览/下载:107/0
  |  
提交时间:2019/01/08
EGFR(C797s)
Clinical resistance
Fourth-generation nhibitors
Monodrug efficacy
Discovery of JND3229 as a New EGFR(C797S) Mutant Inhibitor with In Vivo Monodrug Efficacy
期刊论文
2018, 卷号: 9, 期号: 11, 页码: 1123
作者:
Lu, Xiaoyun[1]
;
Zhang, Tao[2,6,7]
;
Zhu, Su-Jie[3,4]
;
Xun, Qiuju[5]
;
Tong, Lingjiang[2]
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2019/12/23
2,4-Diarylamino-pyrimidines as kinase inhibitors co-targeting IGF1R and EGFR(L858R/T790M)
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2015, 卷号: 25, 期号: 19, 页码: 4277-4281
作者:
Chan, Shingpan
;
Han, Kun
;
Qu, Rong
;
Tong, Linjiang
;
Li, Yingjun
收藏
  |  
浏览/下载:47/0
  |  
提交时间:2019/01/08
EGFR
IGF1R
NSCLC
Dual inhibitor
2,4-Diarylamino-pyrimidines as kinase inhibitors co-targeting IGF1R and EGFR(L858R/T790M)
期刊论文
2015, 卷号: 25, 期号: [db:dc_citation_issue], 页码: 4277
作者:
Chan, Shingpan[1,2]
;
Han, Kun[3]
;
Qu, Rong[2,3]
;
Tong, Linjiang[3]
;
Li, Yingjun[1,2]
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2019/12/03
2,4-Diarylamino-pyrimidines as kinase inhibitors co-targeting IGF1R and EGFR(L858R/T790M)
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2015, 卷号: 25, 期号: 19, 页码: 4277-4281
Chan, Shingpan
;
Han, Kun
;
Qu, Rong
;
Tong, Linjiang
;
Li, Yingjun
;
Zhang, Zhang
;
Cheng, Huimin
;
Lu, Xiaoyun
;
Patterson, Adam
;
Smaill, Jeff
;
Ren, Xiaomei
;
Ding, Jian
;
Xie, Hua
;
Ding, Ke
收藏
  |  
浏览/下载:246/0
  |  
提交时间:2016/12/16
2,4-Diarylamino-pyrimidines as kinase inhibitors co-targeting IGF1R and EGFR(L858R/T790M)
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2015, 卷号: 25, 期号: 19, 页码: 4277-4281
作者:
Smaill, Jeff
;
Lu, Xiaoyun
;
Cheng, Huimin
;
Zhang, Zhang
;
Li, Yingjun
收藏
  |  
浏览/下载:48/0
  |  
提交时间:2018/12/13
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