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浏览/检索结果: 共7条，第1-7条 帮助 限定条件 发表日期：2020     已选(0)清除 条数/页：5101520253035404550556065707580859095100   排序方式：请选择作者升序作者降序题名升序题名降序发表日期升序发表日期降序提交时间升序提交时间降序 Design, synthesis, and biological evaluation of tetrahydroquinolin derivatives as potent inhibitors of CBP bromodomain 期刊论文 BIOORGANIC CHEMISTRY, 2020, 卷号: 101, 页码: 11 作者:  Chen, Yu;  Bi, Xiaoyang;  Zhang, Fengcai;  Sun, Zhongya;  Xu, Pan 收藏  |  浏览/下载：24/0  |  提交时间：2020/12/24 In silico screening  Drug design  CBP  Bromodomain  Inhibitor  Acute Myeloblastic Leukemia   USP28 and USP25 are downregulated by Vismodegib in vitro and in colorectal cancer cell lines 期刊论文 FEBS JOURNAL, 2020, 页码: 18 作者:  Wang, Hui;  Meng, Qian;  Ding, Yiluan;  Xiong, Muya;  Zhu, Mengying 收藏  |  浏览/下载：84/0  |  提交时间：2020/12/24 colorectal cancer  HDX-MS  inhibitor  USP25  USP28  Vismodegib   A new BET inhibitor, 171, inhibits tumor growth through cell proliferation inhibition more than apoptosis induction 期刊论文 INVESTIGATIONAL NEW DRUGS, 2020, 卷号: 38, 期号: 3, 页码: 700-713 作者:  Damaneh, Mohammadali Soleimani;  Hu, Jian-Ping;  Huan, Xia-Juan;  Song, Shan-Shan;  Tian, Chang-Qing 收藏  |  浏览/下载：35/0  |  提交时间：2020/07/01 BET inhibitor  Cell proliferation  Apoptosis  Anti-cancer agent   Discovery of novel CBP bromodomain inhibitors through TR-FRET-based high-throughput screening 期刊论文 ACTA PHARMACOLOGICA SINICA, 2020, 卷号: 41, 期号: 2, 页码: 286-292 作者:  Zhang, Feng-cai;  Sun, Zhong-ya;  Liao, Li-ping;  Zuo, Yu;  Zhang, Dan 收藏  |  浏览/下载：29/0  |  提交时间：2020/07/01 CBP bromodomain  small-molecule inhibitor  high-throughput screening  TR-FRET  molecular modeling  human leukemia MV4-11 cells   A patent review of BRD4 inhibitors (2013-2019) 期刊论文 EXPERT OPINION ON THERAPEUTIC PATENTS, 2020, 卷号: 30, 期号: 1, 页码: 57-81 作者:  Lu, Tian;  Lu, Wenchao;  Luo, Cheng 收藏  |  浏览/下载：18/0  |  提交时间：2020/07/01 Bromodomain-containing protein 4 (BRD4)  bromodomain and extra-terminal (BET) family  small molecule inhibitors  cancer  patent  therapeutic potential   discoveryofnovelcbpbromodomaininhibitorsthroughtrfretbasedhighthroughputscreening 期刊论文 actapharmacologicasinica, 2020, 卷号: 41, 期号: 2, 页码: 285 作者:  Zhang Fengcai;  Sun Zhongya;  Liao Liping;  Zuo Yu;  Zhang Dan 收藏  |  浏览/下载：35/0  |  提交时间：2020/07/01 CBP bromodomain  small-molecule inhibitor  high-throughput screening  TR-FRET  molecular modeling  human leukemia MV4-11 cells   Protein Kinase D3 promotes the cell proliferation by activating the ERK1/c-MYC axis in breast cancer 期刊论文 Journal of Cellular and Molecular Medicine, 2020, 卷号: 24, 期号: 3, 页码: 2135-2144 作者:  Y. Liu,H. Song,S. Y. Yu,K. H. Huang,X. X. Ma,Y. H. Zhou,S. Yu,J. Z. Zhang and L. M. Chen 收藏  |  浏览/下载：3/0  |  提交时间：2021/07/06