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Repressing MYC by targeting BET synergizes with selective inhibition of PI3K alpha against B cell lymphoma 期刊论文
CANCER LETTERS, 2022, 卷号: 524, 页码: 206-218
作者:  Chen, Zi-qi;  Cao, Zhe-rui;  Wang, Yi;  Zhang, Xi;  Xu, Lan
收藏  |  浏览/下载:53/0  |  提交时间:2021/12/16
CYH33  MYC  P300  BET  B cell lymphoma  PI3K  
The discovery of a novel series of potential ERR alpha inverse agonists based on p-nitrobenzenesulfonamide template for triple-negative breast cancer in vivo 期刊论文
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 2022, 卷号: 37, 期号: 1, 页码: 125-134
作者:  Gao, Zhipei;  Wang, Tianxiao;  Li, Rui;  Du, Yongli;  Lv, Han
收藏  |  浏览/下载:39/0  |  提交时间:2022/01/18
LS-106, a novel EGFR inhibitor targeting C797S, exhibits antitumor activities both in vitro and in vivo 期刊论文
CANCER SCIENCE, 2021, 页码: 12
作者:  Liu, Yingqiang;  Lai, Mengzhen;  Li, Shan;  Wang, Yanan;  Feng, Fang
收藏  |  浏览/下载:61/0  |  提交时间:2022/01/18
A camptothecin-based, albumin-binding prodrug enhances efficacy and safety in vivo 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 226, 页码: 11
作者:  Cheng, Zhiyang;  Huang, Ying;  Shen, Qianqian;  Zhao, Yangrong;  Wang, Lei
收藏  |  浏览/下载:83/0  |  提交时间:2021/11/04
Acceptor engineering of small-molecule fluorophores for NIR-II fluorescence and photoacoustic imaging 期刊论文
JOURNAL OF MATERIALS CHEMISTRY B, 2021, 卷号: 9, 期号: 48, 页码: 9951-9960
作者:  Li, Yaxi;  Zhou, Hongli;  Bi, Renzhe;  Li, Xiuting;  Zha, Menglei
收藏  |  浏览/下载:36/0  |  提交时间:2022/01/04
Discovery of a novel DDRs kinase inhibitor XBLJ-13 for the treatment of idiopathic pulmonary fibrosis 期刊论文
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 11
作者:  Dong, Ying;  Tang, Bi-xi;  Wang, Qi;  Zhou, Li-wei;  Li, Cong
收藏  |  浏览/下载:73/0  |  提交时间:2022/01/04
NIR-II imaging of hepatocellular carcinoma based on a humanized anti-GPC3 antibody 期刊论文
RSC MEDICINAL CHEMISTRY, 2021, 页码: 8
作者:  Shi, Hui;  Huttad, Lakshmi Vageesh;  Tan, Mingdian;  Liu, Hongguang;  Chua, Mei-Sze
收藏  |  浏览/下载:20/0  |  提交时间:2022/01/04
New monoamine antidepressant, hypidone hydrochloride (YL-0919), enhances the excitability of medial prefrontal cortex in mice via a neural disinhibition mechanism 期刊论文
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 11
作者:  Zhang, Yong-Mei;  Ye, Lu-Yu;  Li, Tian-Yu;  Guo, Fan;  Guo, Fei
收藏  |  浏览/下载:19/0  |  提交时间:2022/01/04
Inner nuclear membrane protein TMEM201 promotes breast cancer metastasis by positive regulating TGF beta signaling 期刊论文
ONCOGENE, 2021, 页码: 10
作者:  Kong, Ya;  Zhang, Yutian;  Wang, Hanlin;  Kan, Weijuan;  Guo, Haoran
收藏  |  浏览/下载:50/0  |  提交时间:2022/01/04
Ainsliadimer C, a disesquiterpenoid isolated from Ainsliaea macrocephala, ameliorates inflammatory responses in adipose tissue via Sirtuin 1-NLRP3 inflammasome axis 期刊论文
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 13
作者:  Chen, Cheng;  Ren, Yong-mei;  Zhu, Jian-zhong;  Chen, Jia-li;  Feng, Zhe-ling
收藏  |  浏览/下载:56/0  |  提交时间:2022/01/04


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