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上海药物研究所 [36]
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昆明植物研究所 [11]
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期刊论文 [157]
学位论文 [5]
会议论文 [1]
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2016 [163]
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Diversity-oriented one-pot multicomponent synthesis of spirooxindole derivatives and their biological evaluation for anticancer activities
期刊论文
TETRAHEDRON, 2016, 卷号: 72, 期号: 52, 页码: 8523-8536
作者:
Yang, Jun
;
Liu, Xiong-Wei
;
Wang, Dan-Dan
;
Tian, Min-Yi
;
Han, Shuo-Nan
收藏
  |  
浏览/下载:84/0
  |  
提交时间:2017/02/14
Five-membered carbocyclic spirooxindoles
One-pot multicomponent synthesis
Knoevenagel condensation/Michael/cyclization
Aminomethylation
Antitumor activity
Preclinical Efficacy and Safety Assessment of Artemisinin-Chemotherapeutic Agent Conjugates for Ovarian Cancer
期刊论文
EBIOMEDICINE, 2016, 卷号: 14, 页码: 44-54
作者:
Li, Xiaoguang
;
Zhou, Yu
;
Liu, Yanling
;
Zhang, Xu
;
Chen, Tao
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2019/01/08
Dihydroartemisinin
Drug conjugates
Cell cycle
Apoptosis
Metastasis
Ovarian cancer
Pterostilbene induces apoptosis and cell cycle arrest in diffuse large B-cell lymphoma cells
期刊论文
SCIENTIFIC REPORTS, 2016, 卷号: 6
作者:
Kong, Yuanyuan
;
Chen, Gege
;
Xu, Zhijian
;
Yang, Guang
;
Li, Bo
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2019/01/08
Metabolism-based structure optimization: Discovery of a potent and orally available tyrosine kinase ALK inhibitor bearing the tetracyclic benzo[b]carbazolone core
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2016, 卷号: 26, 期号: 22, 页码: 5399-5402
作者:
Han, Mei
;
Wang, Chengyan
;
Ji, Yinchun
;
Song, Zilan
;
Xing, Li
收藏
  |  
浏览/下载:66/0
  |  
提交时间:2019/01/08
EML4-ALK kinase
Oxidative metabolism
Benzo[b]carbazolone
hERG
Antitumor activity
Antitumor action of CDK inhibitor LS-007 as a single agent and in combination with ABT-199 against human acute leukemia cells
期刊论文
ACTA PHARMACOLOGICA SINICA, 2016, 卷号: 37, 期号: 11, 页码: 1481-1489
作者:
Xie, Shao
;
Jiang, Hui
;
Zhai, Xiao-wen
;
Wei, Fan
;
Wang, Shu-dong
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2019/01/08
acute leukemia
CDK9
LS-007
ABT-199
apoptosis
drug synergism
Optimization, characterization, sulfation and antitumor activity of neutral polysaccharides from the fruit of Borojoa sorbilis cuter
期刊论文
CARBOHYDRATE POLYMERS, 2016, 卷号: 151, 页码: 364-372
作者:
Xu, Fangfang
;
Liao, Kangsheng
;
Wu, Yunshan
;
Pan, Qi
;
Wu, Lilan
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2019/01/08
Borojoa sorbilis cuter
Polysaccharide
Structural characterization
Sulfation
Antitumor activity
Metabolic characterization of pyrotinib in humans by ultra-performance liquid chromatography/quadrupole time-of-flight mass spectrometry
期刊论文
Journal of chromatography b-analytical technologies in the biomedical and life sciences, 2016, 卷号: 1033, 页码: 117-127
作者:
Zhu, Yunting
;
Li, Liang
;
Zhang, Ge
;
Wan, Hong
;
Yang, Changyong
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  |  
浏览/下载:40/0
  |  
提交时间:2019/05/09
Pyrotinib
Uplc/q-tof ms
Metabolism
Human
Cyp3a4
Drug-drug interaction
Metabolic characterization of pyrotinib in humans by ultra-performance liquid chromatography/quadrupole time-of-flight mass spectrometry
期刊论文
JOURNAL OF CHROMATOGRAPHY B-ANALYTICAL TECHNOLOGIES IN THE BIOMEDICAL AND LIFE SCIENCES, 2016, 卷号: 1033, 页码: 117-127
作者:
Zhu, Yunting
;
Li, Liang
;
Zhang, Ge
;
Wan, Hong
;
Yang, Changyong
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2019/01/08
Pyrotinib
UPLC/Q-TOF MS
Metabolism
Human
CYP3A4
Drug-drug interaction
HER2-targeted antibody drug conjugates for ovarian cancer therapy
期刊论文
EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES, 2016, 卷号: 93, 页码: 274-286
作者:
Jiang, Jing
;
Dong, Lihou
;
Wang, Lei
;
Wang, Ling
;
Zhang, Jing
收藏
  |  
浏览/下载:52/0
  |  
提交时间:2019/01/08
Ovarian cancer
Antibody drug conjugates (ADCs)
HER2/ErbB2
Monomethyl auristatin E (MMAE)
Safety, pharmacokinetics, and antitumor properties of anlotinib, an oral multi-target tyrosine kinase inhibitor, in patients with advanced refractory solid tumors
期刊论文
JOURNAL OF HEMATOLOGY & ONCOLOGY, 2016, 卷号: 9
作者:
Sun, Yongkun
;
Niu, Wei
;
Du, Feng
;
Du, Chunxia
;
Li, Shuting
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  |  
浏览/下载:35/0
  |  
提交时间:2019/01/08
Anlotinib
Anti-angiogenesis
Phase I study
Advanced refractory solid tumors
Pharmacokinetics
Safety
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