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C3-Arylation of indoles with aryl ketones via C-C/C-H activations 期刊论文
CHEMICAL COMMUNICATIONS, 2021, 页码: 4
作者:  Guo, Zi-Qiong;  Xu, Hui;  Wang, Xing;  Wang, Zhen-Yu;  Ma, Biao
收藏  |  浏览/下载:44/0  |  提交时间:2021/11/04
Affinity Mass Spectrometry-Based Fragment Screening Identified a New Negative Allosteric Modulator of the Adenosine A(2A) Receptor Targeting the Sodium Ion Pocket 期刊论文
ACS CHEMICAL BIOLOGY, 2021, 卷号: 16, 期号: 6, 页码: 991-1002
作者:  Lu, Yan;  Liu, Hongyue;  Yang, Dehua;  Zhong, Li;  Xin, Ye
收藏  |  浏览/下载:25/0  |  提交时间:2021/08/17
Ligand-Promoted Alkynylation of Aryl Ketones: A Practical Tool for Structural Diversity in Drugs and Natural Products 期刊论文
ACS CATALYSIS, 2021, 卷号: 11, 期号: 3, 页码: 1758-1764
作者:  Xu, Hui;  Ma, Biao;  Fu, Zunyun;  Li, Han-Yuan;  Wang, Xing
收藏  |  浏览/下载:16/0  |  提交时间:2021/05/24
Ligand-induced activation of ERK1/2 signaling by constitutively active G(s)-coupled 5-HT receptors 期刊论文
ACTA PHARMACOLOGICA SINICA, 2019, 卷号: 40, 期号: 9, 页码: 1157-1167
作者:  Liu, Ping;  Yin, Yu-ling;  Wang, Ting;  Hou, Li;  Wang, Xiao-xi
收藏  |  浏览/下载:19/0  |  提交时间:2020/07/01
5-HT4R  5-HT6R  5-HT7AR  5-HT  ERK1/2  G(s)  beta-arrestin  Fyn  Src  
N-glycosylation of the beta(2) adrenergic receptor regulates receptor function by modulating dimerization 期刊论文
FEBS JOURNAL, 2017, 卷号: 284, 期号: 13, 页码: 2004-2018
作者:  Li, Xiaona;  Zhou, Mang;  Huang, Wei;  Yang, Huaiyu
收藏  |  浏览/下载:13/0  |  提交时间:2019/01/08
Androgen receptor: structure, role in prostate cancer and drug discovery 期刊论文
ACTA PHARMACOLOGICA SINICA, 2015, 卷号: 36, 期号: 1, 页码: 3-23
作者:  Tan, M. H. Eileen;  Li, Jun;  Xu, H. Eric;  Melcher, Karsten;  Yong, Eu-leong
收藏  |  浏览/下载:22/0  |  提交时间:2019/01/08
A bufadienolide derived androgen receptor antagonist with inhibitory activities against prostate cancer cells 期刊论文
CHEMICO-BIOLOGICAL INTERACTIONS, 2014, 卷号: 207, 页码: 16-22
作者:  Tian, Hai-Yan;  Yuan, Xiao-Feng;  Jin, Lu;  Li, Juan;  Luo, Cheng
收藏  |  浏览/下载:21/0  |  提交时间:2019/01/08
Molecular Modeling of the 3D Structure of 5-HT1AR: Discovery of Novel 5-HT1AR Agonists via Dynamic Pharmacophore-Based Virtual Screening 期刊论文
JOURNAL OF CHEMICAL INFORMATION AND MODELING, 2013, 卷号: 53, 期号: 12, 页码: 3202-3211
作者:  Xu, Lili;  Zhou, Shanglin;  Yu, Kunqian;  Gao, Bo;  Jiang, Hualiang
收藏  |  浏览/下载:14/0  |  提交时间:2019/01/08
Effects of HO-/MeO-PBDEs on Androgen Receptor: In Vitro Investigation and Helix 12-Involved MD Simulation 期刊论文
ENVIRONMENTAL SCIENCE & TECHNOLOGY, 2013, 卷号: 47, 期号: 20, 页码: 11802-11809
作者:  Wang, Xiaoxiang;  Yang, Huaiyu;  Hu, Xinxin;  Zhang, Xiaowei;  Zhang, Qiansen
收藏  |  浏览/下载:12/0  |  提交时间:2019/01/08
Mapping the Functional Binding Sites of Cholesterol in beta(2)-Adrenergic Receptor by Long-Time Molecular Dynamics Simulations 期刊论文
JOURNAL OF PHYSICAL CHEMISTRY B, 2013, 卷号: 117, 期号: 4, 页码: 1085-1094
作者:  Cang, Xiaohui;  Du, Yun;  Mao, Yanyan;  Wang, Yuanyuan;  Yang, Huaiyu
收藏  |  浏览/下载:8/0  |  提交时间:2019/01/08


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