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上海药物研究所 [5]
山东大学 [4]
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期刊论文 [15]
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PARP14 inhibits microglial activation via LPAR5 to promote post-stroke functional recovery
期刊论文
AUTOPHAGY, 2021, 卷号: 17, 期号: 10, 页码: 2905-2922
作者:
Tang, Ying
;
Liu, Jinchang
;
Wang, Yu
;
Yang, Li
;
Han, Bing
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  |  
浏览/下载:43/0
  |  
提交时间:2022/01/04
Autophagy
functional recovery
ischemic stroke
lysophosphatidic acid receptor 5
microglial activation
poly (ADP-ribose) polymerase 14
BOS-93, a novel bromophenol derivative, induces apoptosis and autophagy in human A549 lung cancer cells via PI3K/Akt/mTOR and MAPK signaling pathway
期刊论文
EXPERIMENTAL AND THERAPEUTIC MEDICINE, 2019, 卷号: 17, 期号: 5, 页码: 3848-3858
作者:
Guo, Chuanlong
;
Wang, Lijun
;
Zhao, Yue
;
Jiang, Bo
;
Luo, Jiao
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  |  
浏览/下载:117/0
  |  
提交时间:2019/08/28
bromophenol
apoptosis
autophagy
phosphoinositide 3-kinase
protein kinase B
mechanistic target of rapamycin signaling
reactive oxygen species
Pharmacologic characterization of fluzoparib, a novel poly(ADP-ribose) polymerase inhibitor undergoing clinical trials
期刊论文
CANCER SCIENCE, 2019, 卷号: 110, 期号: 3, 页码: 1064-1075
作者:
Wang, Lei
;
Yang, Changyong
;
Xie, Chengying
;
Jiang, Jiahua
;
Gao, Mingzhao
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  |  
浏览/下载:22/0
  |  
提交时间:2020/07/01
antitumor activity
fluzoparib
pharmacokinetics
poly(ADP-ribose) polymerase
toxicity
Discovery of potent 2,4-difluoro-linker poly(ADP-ribose) polymerase 1 inhibitors with enhanced water solubility and in vivo anticancer efficacy
期刊论文
ACTA PHARMACOLOGICA SINICA, 2017, 卷号: 38, 期号: 11, 页码: 1521-1532
作者:
Chen, Wen-hua
;
Song, Shan-shan
;
Qi, Ming-hui
;
Huan, Xia-juan
;
Wang, Ying-qing
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  |  
浏览/下载:26/0
  |  
提交时间:2019/01/08
PARP-1 inhibitor
olaparib
breast cancer
BRCA-deficient tumors
Discovery, mechanism and metabolism studies of 2,3-difluorophenyl-linker-containing PARP1 inhibitors with enhanced in vivo efficacy for cancer therapy
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 138, 页码: 514-531
作者:
Chen, Wenhua
;
Guo, Ne
;
Qi, Minghui
;
Dai, Haiying
;
Hong, Minghuang
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  |  
浏览/下载:29/0
  |  
提交时间:2019/01/08
Antitumor drug
BRCA1/2
PARP inhibitors
Molecular docking
Mixed galactolipid anomers accentuate apoptosis of multiple myeloma cells by inducing DNA damage
期刊论文
CARBOHYDRATE RESEARCH, 2015, 卷号: 408, 页码: 114-118
作者:
Deng, Si-Si
;
Zhang, Chao
;
Wang, Huan
;
Zang, Yi
;
Li, Jia
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  |  
浏览/下载:16/0
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提交时间:2019/01/08
Multiple myeloma
Glycolipid
Anomer
Synergism
Apoptosis
XRCC1 rs25487 polymorphism is associated with lung cancer risk in epidemiologically susceptible Chinese people
期刊论文
GENETICS AND MOLECULAR RESEARCH, 2015, 卷号: 14, 期号: 4
作者:
Wang, X.
;
Ma, K. W.
;
Zhao, Y. G.
;
Wang, G. J.
;
Li, W.
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  |  
浏览/下载:9/0
  |  
提交时间:2019/12/05
Base excision repair
Lung cancer
8-Oxoguanine DNA glycosylase rs1052133
poly(ADP-ribose) polymerase 1 rs1136410
Single nucleotide polymorphisms
X-ray repair cross-complementing group 1 rs25487
Voltage-Gated Potassium Channel Kv13 Is Highly Expressed in Human Osteosarcoma and Promotes Osteosarcoma Growth
期刊论文
http://dx.doi.org/10.3390/ijms140919245, 2013
Wu, Jin
;
Zhong, Daixing
;
Wu, Xinyu
;
Sha, Mo
;
Kang, Liangqi
;
Ding, Zhenqi
;
吴进
;
吴欣宇
;
沙漠
;
康两期
;
丁真奇
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2015/07/22
ION CHANNELS
CELL-PROLIFERATION
INDUCED APOPTOSIS
EWINGS-SARCOMA
BREAST-CANCER
K+ CHANNELS
LYMPHOCYTES
METASTASIS
THERAPY
ROLES
Cellular NAD depletion and decline of SIRT1 activity play critical roles in PARP-1-mediated acute epileptic neuronal death in vitro
期刊论文
Brain research, 2013, 页码: 14-23
作者:
Wang,S.
;
Yang,X.
;
Lin,Y.
;
Qiu,X.
;
Li,H.
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2019/12/23
Apoptosis-inducing factor
Epilepsy
NAD
Neuronal death
Poly(ADP-ribose)polymerase-1
SIRT1
Cellular NAD depletion and decline of SIRT1 activity play critical roles in PARP-1-mediated acute epileptic neuronal death in vitro
期刊论文
BRAIN RESEARCH, 2013, 卷号: 1535, 页码: 14-23
作者:
Wang, Shengjun
;
Yang, Xue
;
Lin, Youting
;
Qiu, Xiaoxue
;
Li, Hui
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2019/12/23
Poly(ADP-ribose)polymerase-1
NAD
Apoptosis-inducing factor
SIRT1
Epilepsy
Neuronal death
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