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Discovery of an Inhibitor for the TREK-1 Channel Targeting an Intermediate Transition State of Channel Gating 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 19, 页码: 10972-10983
作者:  Ma, Yuqin;  Luo, Qichao;  Fu, Jie;  Che, Yanxin;  Guo, Fei
收藏  |  浏览/下载:11/0  |  提交时间:2021/05/24
TREK Channel Family Activator with a Well-Defined Structure-Activation Relationship for Pain and Neurogenic Inflammation 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 7, 页码: 3665-3677
作者:  Qiu, Yunguang;  Huang, Lu;  Fu, Jie;  Han, Chenxia;  Fang, Jing
收藏  |  浏览/下载:43/0  |  提交时间:2020/07/01
A Small-Molecule Compound Selectively Activates K2P Channel TASK-3 by Acting at Two Distant Clusters of Residues 期刊论文
MOLECULAR PHARMACOLOGY, 2019, 卷号: 96, 期号: 1, 页码: 26-35
作者:  Tian, Fuyun;  Qiu, Yunguang;  Lan, Xi;  Li, Min;  Yang, Huaiyu
收藏  |  浏览/下载:18/0  |  提交时间:2020/07/01
Comparison of Therapeutic Effects of TREK1 Blockers and Fluoxetine on Chronic Unpredicted Mild Stress Sensitive Rats 期刊论文
ACS CHEMICAL NEUROSCIENCE, 2018
作者:  Qi, Xinyang;  Zhang, Zhijun;  Wang, Liping;  Xu, Hua
收藏  |  浏览/下载:19/0  |  提交时间:2019/01/31
Lig4-4 selectively inhibits TREK-1 and plays potent neuroprotective roles in vitro and in rat MCAO model 期刊论文
2018, 卷号: 671, 页码: 93-98
作者:  Wang, Weiping;  Liu, Dongmei;  Xiao, Qiong;  Cai, Jie;  Feng, Nan
收藏  |  浏览/下载:3/0  |  提交时间:2020/01/03
Bepridil a class IV antiarrhythmic agent can block TREK-1 potassium channel 会议论文
29th Great Wall International Congress of Cardiology (GW-ICC), China-Heart-Society, and Beijing-Society-of-Cardiology, OCT 11-14, 2018
作者:  Zhiyong, M. A.;  Fu, Zhijie;  Li, Na;  Huang, Shanying;  Li, Li
收藏  |  浏览/下载:3/0  |  提交时间:2019/12/31
An allosteric ligand-binding site in the extracellular cap of K2P channels 期刊论文
NATURE COMMUNICATIONS, 2017, 卷号: 8
作者:  Luo, Qichao;  Chen, Liping;  Cheng, Xi;  Ma, Yuqin;  Li, Xiaona
收藏  |  浏览/下载:17/0  |  提交时间:2019/01/08
甲亢性心脏病中T4对心磷脂合成及TREK-1和KCNQ1的影响 学位论文
2017, 2016
郭凡
收藏  |  浏览/下载:5/0  |  提交时间:2017/06/20
T4  心磷脂  TREK-1  KCNQ1  T4  Cardiolipin  TREK-1  KCNQ1  
Arachidonic acid has protective effects on oxygen-glucose deprived astrocytes mediated through enhancement of potassium channel TREK-1 activity 期刊论文
NEUROSCIENCE LETTERS, 2017, 卷号: 636, 页码: 241-247
作者:  Lu, L;  Zhang, GR;  Song, CL;  Wang, XX;  Qian, WN
收藏  |  浏览/下载:7/0  |  提交时间:2017/05/08
Over-expressed human TREK-1 inhibits CHO cell proliferation via inhibiting PKA and p38 MAPK pathways and subsequently inducing G(1) arrest 期刊论文
2016, 卷号: 37, 期号: 9, 页码: 1190-1198
作者:  Zhang, Man;  Yin, Hua-jing;  Wang, Wei-ping;  Li, Jiang;  Wang, Xiao-liang
收藏  |  浏览/下载:4/0  |  提交时间:2020/01/04


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