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Identification of Betulinic Acid Derivatives as Potent TGR5 Agonists with Antidiabetic Effects via Humanized TGR5(H88Y) Mutant Mice 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 16, 页码: 12181-12199
作者:  Yun, Ying;  Zhang, Chenlu;  Guo, Shimeng;  Liang, Xiaoying;  Lan, Yuan
收藏  |  浏览/下载:40/0  |  提交时间:2021/11/04
A novel bile acid analog, A17, ameliorated non-alcoholic steatohepatitis in high-fat diet-fed hamsters 期刊论文
TOXICOLOGY AND APPLIED PHARMACOLOGY, 2020, 卷号: 404, 页码: 14
作者:  Wang, Ying;  Zhu, Yao;  Niu, Junxing;  Deng, Qiangqiang;  Guo, Shimeng
收藏  |  浏览/下载:59/0  |  提交时间:2020/12/21
Design of G-protein-coupled bile acid receptor 1 (GPBAR1, TGR5) soft drugs with reduced gallbladder-filling effects 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 203, 页码: 12
作者:  Han, Fanghui;  Ning, Mengmeng;  Cao, Hua;  Ye, Yangliang;  Feng, Ying
收藏  |  浏览/下载:32/0  |  提交时间:2020/12/21
Structural basis of GPBAR activation and bile acid recognition 期刊论文
NATURE, 2020, 页码: 29
作者:  Yang, Fan;  Mao, Chunyou;  Guo, Lulu;  Lin, Jingyu;  Ming, Qianqian
收藏  |  浏览/下载:44/0  |  提交时间:2020/12/24
TGR5 agonist ameliorates insulin resistance in skeletal muscles and improves glucose homeostasis in diabetic mice 期刊论文
METABOLISM-CLINICAL AND EXPERIMENTAL, 2019, 卷号: 99, 页码: 45-56
作者:  Huang, Suling;  Ma, Shanyao;  Ning, Mengmeng;  Yang, Wenji;  Ye, Yangliang
收藏  |  浏览/下载:24/0  |  提交时间:2020/07/01
Targeting Bile Acid-Activated Receptors in Bariatric Surgery. 期刊论文
Handbook of experimental pharmacology, 2019
作者:  Ding Lili;  Fang Zhipeng;  Liu Yanjun;  Zhang Eryun;  Huang Tracy
收藏  |  浏览/下载:48/0  |  提交时间:2019/12/05
胆汁酸膜受体TGR5在代谢性疾病中作用的研究进展 期刊论文
中国临床新医学, 2019, 期号: 1
作者:  吴晓贤;  王晓柠
收藏  |  浏览/下载:7/0  |  提交时间:2019/12/05
胆汁酸膜受体TGR5在代谢性疾病中作用的研究进展 期刊论文
中国临床新医学, 2019, 卷号: 12, 期号: 1
作者:  王晓柠;  吴晓贤
收藏  |  浏览/下载:3/0  |  提交时间:2019/12/05
Metabolite-Sensing G Protein Coupled Receptor TGR5 Protects Host From Viral Infection Through Amplifying Type I Interferon Responses 期刊论文
FRONTIERS IN IMMUNOLOGY, 2018, 卷号: 9
作者:  Xiong, Qingqing;  Huang, Hongjun;  Wang, Ning;  Chen, Ruoyu;  Chen, Naiyang
收藏  |  浏览/下载:2/0  |  提交时间:2019/12/06
Metabolite-Sensing G Protein Coupled Receptor TGR5 Protects Host From Viral Infection Through Amplifying Type I Interferon Responses 期刊论文
FRONTIERS IN IMMUNOLOGY, 2018, 卷号: Vol.9
作者:  Xiong, Qingqing;  Huang, Hongjun;  Wang, Ning;  Chen, Ruoyu;  Chen, Naiyang
收藏  |  浏览/下载:5/0  |  提交时间:2019/12/26


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