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科研机构
上海药物研究所 [4]
厦门大学 [3]
北京大学 [1]
内容类型
期刊论文 [8]
发表日期
2017 [2]
2015 [1]
2014 [2]
2009 [2]
2008 [1]
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Marine-derived chromopeptide A, a novel class I HDAC inhibitor, suppresses human prostate cancer cell proliferation and migration
期刊论文
ACTA PHARMACOLOGICA SINICA, 2017, 卷号: 38, 期号: 4, 页码: 551-560
作者:
Sun, Jing-ya
;
Wang, Ji-dong
;
Wang, Xin
;
Liu, Hong-chun
;
Zhang, Min-min
收藏
  |  
浏览/下载:42/0
  |  
提交时间:2019/01/08
HDAC
chromopeptide A
FK228
human prostate cancer
cell cycle arrest
apoptosis
cancer cell migration
PC3 xenograft model
marinederivedchromopeptideaanovelclassihdacinhibitorsuppresseshumanprostatecancercellproliferationandmigration
期刊论文
actapharmacologicasinica, 2017, 卷号: 38, 期号: 4, 页码: 551
作者:
Sun Jingya
;
Wang Jidong
;
Wang Xin
;
Liu Hongchun
;
Zhang Minmin
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2020/07/01
HISTONE DEACETYLASE INHIBITORS
ANDROGEN DEPRIVATION THERAPY
ROMIDEPSIN
VORINOSTAT
EXPRESSION
RESISTANCE
TRIAL
DEPSIPEPTIDE
MITOXANTRONE
ABIRATERONE
HDAC
chromopeptide A
FK228
human prostate cancer
cell cycle arrest
apoptosis
cancer cell migration
PC3 xenograft model
Design, synthesis and biological evaluation of isoquinoline-based derivatives as novel histone deacetylase inhibitors
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2015, 卷号: 23, 期号: 17, 页码: 5881-5890
作者:
Yang, Wei
;
Li, Lixuan
;
Wang, Yulan
;
Wu, Xiaowei
;
Li, Tingting
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2019/01/08
HDACs
HDACs inhibitor
Hydroxamic acid
Isoquinoline
Design, synthesis and biological evaluation of 4-anilinothieno[2,3-d]pyrimidine-based hydroxamic acid derivatives as novel histone deacetylase inhibitors
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2014, 卷号: 22, 期号: 21, 页码: 6146-6155
作者:
Yang, Wei
;
Li, Lixuan
;
Ji, Xun
;
Wu, Xiaowei
;
Su, Mingbo
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2019/01/08
HDACs
HDACs inhibitor
Hydroxamic acid
Thieno[2,3-d]pyrimidines
Targeting Histone Deacetylases for Cancer Therapy: From Molecular Mechanisms to Clinical Implications
期刊论文
international journal of biological sciences, 2014
Li, Zhiming
;
Zhu, Wei-Guo
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  |  
浏览/下载:8/0
  |  
提交时间:2015/11/11
HDAC
HDAC inhibitor
epigenetic therapy
cancer
DNA-DAMAGE RESPONSE
HYPOXIA-INDUCIBLE FACTOR-1-ALPHA
TO-MESENCHYMAL TRANSITION
AUTOPHAGIC CELL-DEATH
INHIBITOR DEPSIPEPTIDE
GENE-EXPRESSION
VALPROIC ACID
CHROMATIN-STRUCTURE
MEDIATED APOPTOSIS
HDAC INHIBITOR
FACILE SYNTHESES OF THREE AHP-TYPE BUILDING BLOCKS WITH COMPLEMENTARY REACTIVITIES
期刊论文
http://dx.doi.org/10.3987/COM-08-S(D)35, 2009
Chen, W
;
Zheng, X
;
Ruan, YP
;
Huang, PQ
;
黄培强
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  |  
浏览/下载:2/0
  |  
提交时间:2013/12/12
CYANOBACTERIUM MICROCYSTIS-AERUGINOSA
N-ACYLIMINIUM IONS
ASYMMETRIC-SYNTHESIS
CYCLIC DEPSIPEPTIDE
OSCILLATORIA-AGARDHII
MICROPEPTIN T-20
AMINO-ACIDS
STEREOSELECTIVE-SYNTHESIS
CHYMOTRYPSIN INHIBITOR
ALPHA-AMIDOALKYLATION
FACILE SYNTHESES OF THREE AHP-TYPE BUILDING BLOCKS WITH COMPLEMENTARY REACTIVITIES
期刊论文
http://dx.doi.org/10.3987/COM-08-S(D)35, 2009
Chen,W
;
Huang,PQ
;
Ruan,YP
;
Zheng,X
;
郑啸
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2013/12/12
CYANOBACTERIUM MICROCYSTIS-AERUGINOSA
N-ACYLIMINIUM IONS
ASYMMETRIC-SYNTHESIS
CYCLIC DEPSIPEPTIDE
OSCILLATORIA-AGARDHII
MICROPEPTIN T-20
AMINO-ACIDS
STEREOSELECTIVE-SYNTHESIS
CHYMOTRYPSIN INHIBITOR
ALPHA-AMIDOALKYLATION
Phenylhexyl isothiocyanate has dual function as histone deacetylase inhibitor and hypomethylating agent and can inhibit myeloma cell growth by targeting critical pathways
期刊论文
http://dx.doi.org/10.1186/1756-8722-1-6, 2008
Lu, Quanyi
;
Lin, Xianghua
;
Feng, Jean
;
Zhao, Xiangmin
;
Gallagher, Ruth
;
Lee, Marietta Y.
;
Chiao, Jen-Wei
;
Liu, Delong
;
鹿全意
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2015/07/22
SUBEROYLANILIDE HYDROXAMIC ACID
HUMAN MULTIPLE-MYELOMA
PROSTATE-CANCER CELLS
MYELODYSPLASTIC SYNDROMES
DEPSIPEPTIDE FR901228
PLASMA-CELLS
P16 GENE
IN-VIVO
METHYLATION
APOPTOSIS
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