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科研机构
安徽大学 [7]
内容类型
期刊论文 [7]
发表日期
2019 [2]
2018 [4]
2015 [1]
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专题:安徽大学
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Discovery of N-phenyl)-2-phenyl)acetamide as a Potent FMS-like Tyrosine Kinase 3 Internal Tandem Duplication Mutant Selective Inhibitor for Acute Myeloid Leukemia
期刊论文
Journal of Medicinal Chemistry, 2019, 卷号: Vol.62 No.2, 页码: 875-892
作者:
Tingting Lu
;
Jian Ge
;
Tao Ren
;
Wenchao Wang
;
Junjie Wang
收藏
  |  
浏览/下载:36/0
  |  
提交时间:2019/04/24
Discovery of N-phenyl)-2-phenyl)acetamide as a Potent FMS-like Tyrosine Kinase 3 Internal Tandem Duplication Mutant Selective Inhibitor for Acute Myeloid Leukemia
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: Vol.62 No.2, 页码: 875-892
作者:
Wang, Beilei
;
Li, Feng
;
Liu, Qingwang
;
Hu, Zhenquan
;
Liang, Xiaofei
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2019/04/24
Discovery of (S)-2-amino-N-(5-(6-chloro-5-(3-methylphenylsulfonamido)pyridin-3-yl)-4-methylthiazol-2-yl)-3-methylbutanamide (CHMFL-PI3KD-317) as a potent and selective phosphoinositide 3-kinase delta (PI3Kδ) inhibitor
期刊论文
European Journal of Medicinal Chemistry, 2018, 卷号: Vol.156, 页码: 831-846
作者:
Zongru Jiang
;
Wenliang Wang
;
Fengming Zou
;
Jing Liu
;
Qingsong Liu
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2019/04/22
PI3Kδ
Kinase
inhibitor
Acute
myeloid
leukemia
Structure-activity
relationship
Discovery of (E)-N-(4-((4-methylpiperazin-1-yl)methyl)-3-(trifluoromethyl)phenyl)-3-((3-(2-(pyridin-2-yl)vinyl)-1H-indazol-6-yl)thio)propanamide (CHMFL-ABL-121) as a highly potent ABL kinase inhibitor capable of overcoming a variety of ABL mutants including T315I for chronic myeloid leukemia
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: Vol.160, 页码: 61-81
作者:
Liu, Xiaochuan
;
Wang, Beilei
;
Wang, Junjie
;
Zhang, Yicong
;
Jiang, Zongru
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  |  
浏览/下载:12/0
  |  
提交时间:2019/04/24
ABL kinase
Kinase inhibitor
ABL mutant
CML
Discovery of 4--4-amino) cyclohexyl)amino)pyridin-4-yl)thiazol-2-yl)amino)methyl) tetrahydro-2H-pyran-4-carbonitrile as a novel highly selective and potent CDK9 kinase inhibitor
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: Vol.158, 页码: 896-916
作者:
Wang, Beilei
;
Wu, Yun
;
Liu, Qingwang
;
Jiang, Zongru
;
Wu, Jiaxin
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2019/04/24
CDK9
Kinase
inhibitor
Structure-activity
relationship
Leukemia
Discovery of -2-amino-N-pyridin-3-yl)-4-methylthiazol-2-yl)-3-methylbutanamide as a potent and selective phosphoinositide 3-kinase delta inhibitor
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: Vol.156, 页码: 831-846
作者:
Liu, Xiaochuan
;
Jiang, Zongru
;
Li, Feng
;
Hu, Zhenquan
;
Ge, Juan
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2019/04/24
PI3K
delta
Kinase
inhibitor
Acute
myeloid
leukemia
Structure-activity
relationship
Robust expression of vault RNAs induced by influenza A virus plays a critical role in suppression of PKR-mediated innate immunity.
期刊论文
Nucleic Acids Res., 2015, 卷号: Vol.43 No.21, 页码: 10321-10337
作者:
Chen,Ji-Long
;
Gao,George Fu
;
Yan,Ruoxiang
;
Wang,Yi
;
Guo,Guijie
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2019/04/22
DOUBLE-STRANDED-RNA
LONG NONCODING RNA
PROTEIN-KINASE PKR
TRANSLATION INITIATION-FACTOR
NS1 PROTEIN
HOST FACTORS
CELLULAR INHIBITOR
VIRAL REPLICATION
RIG-I
INTERFERON
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