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上海药物研究所 [9]
复旦大学上海医学院 [4]
西安交通大学 [3]
东北农业大学 [3]
兰州大学 [2]
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期刊论文 [36]
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Synthesis of the analogs of plocabulin and their preliminary structure-activity relationship study
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2021, 卷号: 51, 页码: 5
作者:
Wang, Leiming
;
Li, Xin
;
Cui, Hong
;
Lei, Xinsheng
;
Liu, Hongchun
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2021/12/01
Marine nature products
Plocabulin
PM060184
Synthesis
Antiproliferation
Design, Synthesis and Antiproliferative Activity of Chrysin Derivatives Bearing Triazole Moieties
期刊论文
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2020, 卷号: 40, 期号: 2, 页码: 440-446
作者:
Luan Tian
;
Quan Zheshan
;
Fang Yingquan
;
Yang Hongjing
收藏
  |  
浏览/下载:38/0
  |  
提交时间:2021/02/02
INHIBITION
CELLS
chrysin
synthesis
triazole
derivatives
antiproliferation
Identification of new NIK inhibitors by discriminatory analysis-based molecular docking and biological evaluation
期刊论文
ARCHIV DER PHARMAZIE, 2019, 卷号: 352, 期号: 7, 页码: 9
作者:
Cheng, Gang
;
Mei, Xiao-Bing
;
Yan, You-You
;
Chen, Jing
;
Zhang, Bo
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2020/07/01
antiproliferation activity
inhibitors
NF-kappa B inducing kinase
virtual screen
Discovery of Novel PRMT5 Inhibitors by Virtual Screening and Biological Evaluations
期刊论文
CHEMICAL & PHARMACEUTICAL BULLETIN, 2019, 卷号: 67, 期号: 4, 页码: 382-388
作者:
Tao, Hongrui
;
Yan, Xue
;
Zhu, Kongkai
;
Zhang, Hua
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2020/07/01
virtual screening
epigenetic inhibitor
antiproliferation
molecular docking
A unified mitochondria mechanistic target of rapamycin acyl-coenzyme A dehydrogenase 10 signal relay modulation for metformin growth inhibition in human immortalized keratinocytes cells.
期刊论文
Journal of cellular biochemistry, 2019, 卷号: 120, 页码: 1773-1782
作者:
Wu Jiawen
;
Xiao Shengxiang
;
Ren Jianwen
;
Zhang Dingwei
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  |  
浏览/下载:15/0
  |  
提交时间:2019/11/19
antiproliferation, human immortalized keratinocytes
metformin
acyl-coenzyme A dehydrogenase 10 (ACAD10)
(HaCaT) cells
mitochondria mechanistic target of rapamycin 1 (mTORC1) signal
Synthesis and biological evaluation of benzomorpholine derivatives as novel EZH2 inhibitors for anti-non-small cell lung cancer activity.
期刊论文
Molecular diversity, 2019
作者:
Feng Qiang
;
He Hualong
;
Gao Tiantao
;
Zhang Qiangsheng
;
Liu Zhihao
收藏
  |  
浏览/下载:77/0
  |  
提交时间:2019/02/25
Antiproliferation
activity
Benzomorpholine
EZH2
inhibitor
Structure–activity
relationship
Subcritical water extraction, identification and antiproliferation ability on HepG2 of polyphenols from lotus seed epicarp
期刊论文
INDUSTRIAL CROPS AND PRODUCTS, 2019, 卷号: 129, 页码: 472-479
作者:
Yan, Zheng[1]
;
Luo, Xiaoping[2]
;
Cong, Jingli[3]
;
Zhang, Haihui[4]
;
Ma, Haile[5]
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2019/12/24
Polyphenols
Lotus seed epicarp
Subcritical water extraction
Identification
Quantification
Antiproliferation
Crystal structure-based comparison of two NAMPT inhibitors
期刊论文
ACTA PHARMACOLOGICA SINICA, 2018, 卷号: 39, 期号: 2, 页码: 294-301
作者:
Zhang, Sai-long
;
Xu, Tian-ying
;
Yang, Zhen-lin
;
Han, Shuo
;
Zhao, Qiang
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2019/01/08
nicotinamide phosphoribosyltransferase (NAMPT)
FK866
MS0
anticancer drugs
antiproliferation
crystal structure
binding mode
miRNA-34a decreases ovarian cancer cell proliferation and chemoresistance by targeting HDAC1
期刊论文
BIOCHEMISTRY AND CELL BIOLOGY, 2018, 卷号: 96, 期号: 5, 页码: 663-671
作者:
Lv, Teng
;
Song, Kejuan
;
Zhang, Lili
;
Li, Weihua
;
Chen, Yulong
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2019/12/11
miR-34a
ovarian cancer
antiproliferation
cisplatin resistance
HDAC1
Novel multi-kinase inhibitor, T03 inhibits Taxol-resistant breast cancer
期刊论文
2018, 卷号: 17, 期号: 2, 页码: 2373-2383
作者:
Li, Yan
;
Liu, Chunxia
;
Tang, Ke
;
Chen, Yan
;
Tian, Kang
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2020/01/03
multi-kinase inhibitor
T03
antiproliferation
breast cancer
Taxol-resistant breast cancer
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