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科研机构
上海药物研究所 [15]
新疆理化技术研究所 [1]
中国科学院大学 [1]
内容类型
期刊论文 [17]
发表日期
2021 [3]
2020 [2]
2019 [3]
2018 [2]
2017 [2]
2016 [5]
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Facile and Cost-Effective Route for the Synthesis of Simmerafil
期刊论文
ORGANIC PROCESS RESEARCH & DEVELOPMENT, 2021, 卷号: 25, 期号: 11, 页码: 2432-2437
作者:
Odilov, Abdullajon
;
Liu, Yin
;
Hu, Tianwen
;
Jiang, Xiangrui
;
Suo, Jin
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2022/01/18
simmerafil
PDE5 inhibitor
salicylamide
synthesis
TPN672: A Novel Serotonin-Dopamine Receptor Modulator for the Treatment of Schizophrenia
期刊论文
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 2021, 卷号: 378, 期号: 1, 页码: 20-30
作者:
Wang, Yu
;
He, Yang
;
Yang, Feipu
;
Abame, Melkamu Alemu
;
Wu, Chunhui
收藏
  |  
浏览/下载:37/0
  |  
提交时间:2021/11/04
SARS-CoV-2 envelope protein causes acute respiratory distress syndrome (ARDS)-like pathological damages and constitutes an antiviral target
期刊论文
CELL RESEARCH, 2021, 页码: 14
作者:
Xia, Bingqing
;
Shen, Xurui
;
He, Yang
;
Pan, Xiaoyan
;
Liu, Feng-Liang
收藏
  |  
浏览/下载:78/0
  |  
提交时间:2021/08/17
Automated design and optimization of multitarget schizophrenia drug candidates by deep learning
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 204, 页码: 16
作者:
Tan, Xiaoqin
;
Jiang, Xiangrui
;
He, Yang
;
Zhong, Feisheng
;
Li, Xutong
收藏
  |  
浏览/下载:35/0
  |  
提交时间:2020/12/21
Schizophrenia
Multitarget antipsychotic drugs
Recurrent neural network
Multitask deep neural network
Automated drug design
Synthesis and biological investigation of triazolopyridinone derivatives as potential multireceptor atypical antipsychotics
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2020, 卷号: 30, 期号: 8, 页码: 6
作者:
Shi, Wenqiang
;
Wang, Yu
;
Wu, Chunhui
;
Yang, Feipu
;
Zheng, Wei
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2020/07/01
Triazolopyridinone
Antipsychotic
Multireceptor
5-HT1A receptor
Synthesis and Biological Evaluation of Five-Atom-Linker-Based Arylpiperazine Derivatives with an Atypical Antipsychotic Profile
期刊论文
CHEMMEDCHEM, 2019, 页码: 11
作者:
Wu, Chunhui
;
Wang, Yu
;
Yang, Feipu
;
Shi, Wenqiang
;
Wang, Zhen
收藏
  |  
浏览/下载:32/0
  |  
提交时间:2020/07/01
D-2
5-HT1A
5-HT2A
serotonin
SERT
PCP-induced hyperactivity
Oxidative Aromatization of 3,4-Dihydroquinolin-2(1H)-ones to Quinolin-2(1H)-ones Using Transition-Metal-Activated Persulfate Salts
期刊论文
JOURNAL OF ORGANIC CHEMISTRY, 2019, 卷号: 84, 期号: 13, 页码: 8702-8709
作者:
Chen, Weiming
;
Sun, Changliang
;
Zhang, Yan
;
Hu, Tianwen
;
Zhu, Fuqiang
收藏
  |  
浏览/下载:45/0
  |  
提交时间:2020/07/01
Continuation of structure-activity relationship study of novel benzamide derivatives as potential antipsychotics
期刊论文
ARCHIV DER PHARMAZIE, 2019, 卷号: 352, 期号: 4, 页码: 13
作者:
Xu, Mingshuo
;
Guo, Shuang
;
Yang, Feipu
;
Wang, Yu
;
Wu, Chunhui
收藏
  |  
浏览/下载:43/0
  |  
提交时间:2020/07/01
5-HT1A
5-HT2A
catalepsy
D-2
PCP-induced hyperactivity
Synthesis and biological evaluation of a series of novel pyridinecarboxamides as potential multi-receptor antipsychotic drugs
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2018, 卷号: 28, 期号: 4, 页码: 606-611
作者:
Xu, Mingshuo
;
Wang, Yu
;
Yang, Feipu
;
Wu, Chunhui
;
Wang, Zhen
收藏
  |  
浏览/下载:51/0
  |  
提交时间:2019/01/08
Antipsychotic
Multi-receptor
Pyridinecarboxamide
5-HT1A receptor
PCP-induced hyperlocomotion
Synthesis and biological evaluation of a series of multi-target N-substituted cyclic imide derivatives with potential antipsychotic effect
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 145, 页码: 74-85
作者:
Xu, Mingshuo
;
Wang, Yu
;
Yang, Feipu
;
Wu, Chunhui
;
Wang, Zhen
收藏
  |  
浏览/下载:54/0
  |  
提交时间:2019/01/08
Antipsychotic
Cyclic imide
Multi-target
5-HT1A receptor
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