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Design and development of an oral remdesivir derivative VV116 against SARS-CoV-2 期刊论文
CELL RESEARCH, 2021, 页码: 3
作者:  Xie, Yuanchao;  Yin, Wanchao;  Zhang, Yumin;  Shang, Weijuan;  Wang, Zhen
收藏  |  浏览/下载:108/0  |  提交时间:2021/11/04
Identification of pyrogallol as a warhead in design of covalent inhibitors for the SARS-CoV-2 3CL protease 期刊论文
NATURE COMMUNICATIONS, 2021, 卷号: 12, 期号: 1, 页码: 12
作者:  Su, Haixia;  Yao, Sheng;  Zhao, Wenfeng;  Zhang, Yumin;  Liu, Jia
收藏  |  浏览/下载:30/0  |  提交时间:2021/08/17
Kinetics-Driven Drug Design Strategy for Next-Generation Acetylcholinesterase Inhibitors to Clinical Candidate 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 4, 页码: 1844-1855
作者:  Zhou, Yu;  Fu, Yan;  Yin, Wanchao;  Li, Jian;  Wang, Wei
收藏  |  浏览/下载:21/0  |  提交时间:2021/05/24
USP28 and USP25 are downregulated by Vismodegib in vitro and in colorectal cancer cell lines 期刊论文
FEBS JOURNAL, 2020, 页码: 18
作者:  Wang, Hui;  Meng, Qian;  Ding, Yiluan;  Xiong, Muya;  Zhu, Mengying
收藏  |  浏览/下载:84/0  |  提交时间:2020/12/24
Identification of Highly Selective Lipoprotein-Associated Phospholipase A2 (Lp-PLA2) Inhibitors by a Covalent Fragment-Based Approach 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 13, 页码: 7052-7065
作者:  Huang, Fubao;  Hu, Hangchen;  Wang, Kai;  Peng, Chengyuan;  Xu, Wenwei
收藏  |  浏览/下载:41/0  |  提交时间:2020/12/24
Natural product piperine alleviates experimental allergic encephalomyelitis in mice by targeting dihydroorotate dehydrogenase 期刊论文
BIOCHEMICAL PHARMACOLOGY, 2020, 卷号: 177, 页码: 15
作者:  Liu, Zehui;  Hu, Qian;  Wang, Wanyan;  Lu, Sisi;  Wu, Dang
收藏  |  浏览/下载:28/0  |  提交时间:2020/12/24
Structural basis for inhibition of the RNA-dependent RNA polymerase from SARS-CoV-2 by remdesivir 期刊论文
SCIENCE, 2020, 卷号: 368, 期号: 6498, 页码: 1499-+
作者:  Yin, Wanchao;  Mao, Chunyou;  Luan, Xiaodong;  Shen, Dan-Dan;  Shen, Qingya
收藏  |  浏览/下载:56/0  |  提交时间:2020/12/24
Structure-based design of antiviral drug candidates targeting the SARS-CoV-2 main protease 期刊论文
SCIENCE, 2020, 卷号: 368, 期号: 6497, 页码: 1331-+
作者:  Dai, Wenhao;  Zhang, Bing;  Jiang, Xia-Ming;  Su, Haixia;  Li, Jian
收藏  |  浏览/下载:30/0  |  提交时间:2020/12/24
Structure of M-pro from SARS-CoV-2 and discovery of its inhibitors 期刊论文
NATURE, 2020, 页码: 24
作者:  Jin, Zhenming;  Du, Xiaoyu;  Xu, Yechun;  Deng, Yongqiang;  Liu, Meiqin
收藏  |  浏览/下载:40/0  |  提交时间:2020/07/01
Structural basis of ligand binding modes at the human formyl peptide receptor 2 期刊论文
NATURE COMMUNICATIONS, 2020, 卷号: 11, 期号: 1, 页码: 9
作者:  Chen, Tong;  Xiong, Muya;  Zong, Xin;  Ge, Yunjun;  Zhang, Hui
收藏  |  浏览/下载:11/0  |  提交时间:2020/12/24


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