CORC

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Repressing MYC by targeting BET synergizes with selective inhibition of PI3K alpha against B cell lymphoma 期刊论文
CANCER LETTERS, 2022, 卷号: 524, 页码: 206-218
作者:  Chen, Zi-qi;  Cao, Zhe-rui;  Wang, Yi;  Zhang, Xi;  Xu, Lan
收藏  |  浏览/下载:53/0  |  提交时间:2021/12/16
CYH33  MYC  P300  BET  B cell lymphoma  PI3K  
SL010110, a lead compound, inhibits gluconeogenesis via SIRT2-p300-mediated PEPCK1 degradation and improves glucose homeostasis in diabetic mice 期刊论文
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 13
作者:  Ren, Yu-ran;  Ye, Yang-liang;  Feng, Ying;  Xu, Ti-fei;  Shen, Yu
收藏  |  浏览/下载:22/0  |  提交时间:2021/05/24
p300/CBP inhibitor A-485 alleviates acute liver injury by regulating macrophage activation and polarization 期刊论文
THERANOSTICS, 2019, 卷号: 9, 期号: 26, 页码: 8344-8361
作者:  Peng, Jinjin;  Li, Jiacheng;  Huang, Jing;  Xu, Pan;  Huang, Heming
收藏  |  浏览/下载:17/0  |  提交时间:2020/07/01
Discovery and biological evaluation of thiobarbituric derivatives as potent p300/CBP inhibitors 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2018, 卷号: 26, 期号: 20, 页码: 5397-5407
作者:  Lu, Wenchao;  Xiong, Huan;  Chen, Yu;  Wang, Chen;  Zhang, Hao
收藏  |  浏览/下载:139/0  |  提交时间:2019/01/08
Identification of novel inhibitors of histone acetyltransferase hMOF through high throughput screening 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 157, 页码: 867-876
作者:  Zhang, Rukang;  Wang, Jiang;  Zhao, Liang;  Liu, Shien;  Du, Daohai
收藏  |  浏览/下载:37/0  |  提交时间:2019/01/08
Discovery of 1,8-acridinedione derivatives as novel GCN5 inhibitors via high throughput screening 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 151, 页码: 740-751
作者:  Xiong, Huan;  Han, Jie;  Wang, Jun;  Lu, Wenchao;  Wang, Chen
收藏  |  浏览/下载:28/0  |  提交时间:2019/01/08
Comparative Proteomic Analysis of Lysine Acetylation in Fish CIK Cells Infected with Aquareovirus 期刊论文
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 2017, 卷号: 18, 期号: 11, 页码: 21
作者:  Guo, Hong;  Zhang, Jie;  Wang, Yaping;  Bu, Chen;  Zhou, Yanyan
收藏  |  浏览/下载:26/0  |  提交时间:2019/07/03
Hippo Signaling Suppresses Cell Ploidy and Tumorigenesis through Skp2 其他
2017-05-01
Shihao Zhang; 张世浩; Qinghua Chen; 陈青花; Qingxu Liu; 刘清许; Li Yuxi; 李玉席; Xiufeng Sun; 孙秀峰; Lixin Hong; Suyuan Ji; Chengyan Liu; Jing Geng; Weiji Zhang; Zhonglei Lu; ZhenYu Yin; Yuanyuan Zeng; Kwang-Huei Lin; Qiao Wu; Qiyuan Li; Keiko Nakayama; Keiich I.Nakayama; Xianming Deng; Randy L.Johnson; Liang Zhu; Daming Gao; Lanfen Chen; 陈兰芬; Dawang Zhou; 周大旺
收藏  |  浏览/下载:32/0  |  提交时间:2017/05/18
Tip60: Main Functions and Its Inhibitors 期刊论文
MINI-REVIEWS IN MEDICINAL CHEMISTRY, 2017, 卷号: 17, 期号: 8, 页码: 675-682
作者:  Zhang, Xiaoli;  Wu, Jiyong;  Luan, Yepeng
收藏  |  浏览/下载:7/0  |  提交时间:2019/12/11


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