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Adaptive resistance to PI3K alpha-selective inhibitor CYH33 is mediated by genomic and transcriptomic alterations in ESCC cells 期刊论文
CELL DEATH & DISEASE, 2021, 卷号: 12, 期号: 1, 页码: 13
作者:  Wang, Yu-xiang;  Zhang, Xu;  Ma, Qing-yang;  Hu, Lan-dian;  Zhang, Xi
收藏  |  浏览/下载:47/0  |  提交时间:2021/05/24
Emerging roles of class I PI3K inhibitors in modulating tumor microenvironment and immunity 期刊论文
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 8
作者:  Sun, Pu;  Meng, Ling-hua
收藏  |  浏览/下载:39/0  |  提交时间:2020/12/21
Endosulfan promotes cell migration via PTP4A3-mediated signaling pathways in HUVECs 期刊论文
ECOTOXICOLOGY AND ENVIRONMENTAL SAFETY, 2020, 卷号: 192, 页码: 1-9
作者:  Li, Heng;  Liu, Shiqi;  Hu, Yumeng;  Zhao, Bin;  Sun, Yeqing
收藏  |  浏览/下载:24/0  |  提交时间:2021/09/14
Chemical Composition and Biological Activities of Endophytic Fungus Talaromyces Wortmannii LGT-4, Cultured in CYM Medium 期刊论文
IRANIAN JOURNAL OF PHARMACEUTICAL RESEARCH, 2020, 卷号: 19, 期号: 2, 页码: 259-263
作者:  Yang, Zhong-Duo;  Zhang, Yu;  Zhao, Wei-Hua;  Shu, Zong-Mei
收藏  |  浏览/下载:7/0  |  提交时间:2022/03/01
Design, synthesis, and biological evaluation of thieno[3,2-d]pyrimidine derivatives as potential simplified phosphatidylinositol 3-kinase alpha inhibitors 期刊论文
CHEMICAL BIOLOGY & DRUG DESIGN, 2019, 卷号: 94, 期号: 6, 页码: 2013-2022
作者:  Yang, Xiuyan;  Deng, Meng;  Zhang, Xi;  Wang, Yi;  Song, Kun
收藏  |  浏览/下载:75/0  |  提交时间:2020/07/01
Wortmannine F and G, two new pyranones from Talaromyces wortmannii LGT-4, the endophytic fungus of Tripterygium wilfordii 期刊论文
PHYTOCHEMISTRY LETTERS, 2019, 卷号: 29, 页码: 115-118
作者:  Zhao, Jun-Wen;  Yang, Zhong-Duo;  Zhou, Shuan-Yan;  Yang, Li-Jun;  Sun, Jian-Hui
收藏  |  浏览/下载:7/0  |  提交时间:2019/11/15
Wortmannine F and G, two new pyranones from Talaromyces wortmannii LGT-4, the endophytic fungus of Tripterygium wilfordii 期刊论文
PHYTOCHEMISTRY LETTERS, 2019, 卷号: 29, 页码: 115-118
作者:  Zhao, Jun-Wen;  Yang, Zhong-Duo;  Zhou, Shuan-Yan;  Yang, Li-Jun;  Sun, Jian-Hui
收藏  |  浏览/下载:6/0  |  提交时间:2022/03/01
Structure‐based pharmacophore models to probe anticancer activity of inhibitors of protein kinase B‐beta (PKB β). 期刊论文
Chemical Biology & Drug Design, 2019, 卷号: Vol.93 No.3, 页码: 325-336
作者:  Akhtar, N.a;  Jabeen, I.a;  Jalal, N.b;  Antilla, J.b
收藏  |  浏览/下载:16/0  |  提交时间:2019/11/21
High-throughput screening campaigns against a PI3K alpha isoform bearing the H1047R mutation identified potential inhibitors with novel scaffolds 期刊论文
ACTA PHARMACOLOGICA SINICA, 2018, 卷号: 39, 期号: 11, 页码: 1816-1822
作者:  Wang, Jia;  Gong, Grace Qun;  Zhou, Yan;  Lee, Woo-Jeong;  Buchanan, Christina Maree
收藏  |  浏览/下载:84/0  |  提交时间:2019/01/08
Synthesis, biological evaluation and structure-activity relationship of a novel class of PI3K alpha H1047R mutant inhibitors 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 158, 页码: 707-719
作者:  Zhang, Ning;  Yu, Zhimei;  Yang, Xiaohong;  Zhou, Yan;  Wang, Jia
收藏  |  浏览/下载:84/0  |  提交时间:2019/01/08


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