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期刊论文 [29]
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Development of hedgehog pathway inhibitors by epigenetically targeting GLI through BET bromodomain for the treatment of medulloblastoma
期刊论文
ACTA PHARMACEUTICA SINICA B, 2021, 卷号: 11, 期号: 2, 页码: 488-504
作者:
Liu, Xiaohua
;
Zhang, Yu
;
Li, Yalei
;
Wang, Juan
;
Ding, Huaqian
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2021/05/24
Medulloblastoma
Hedgehog signaling
pathway
Drug resistance
GLI
BRD4
USP28 and USP25 are downregulated by Vismodegib in vitro and in colorectal cancer cell lines
期刊论文
FEBS JOURNAL, 2020, 页码: 18
作者:
Wang, Hui
;
Meng, Qian
;
Ding, Yiluan
;
Xiong, Muya
;
Zhu, Mengying
收藏
  |  
浏览/下载:84/0
  |  
提交时间:2020/12/24
colorectal cancer
HDX-MS
inhibitor
USP25
USP28
Vismodegib
Medulloblastoma: Molecular understanding, treatment evolution, and new developments
期刊论文
PHARMACOLOGY & THERAPEUTICS, 2020, 卷号: 210, 页码: 13
作者:
Liu, Xiaohua
;
Ding, Chunyong
;
Tan, Wenfu
;
Zhang, Ao
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2020/07/01
Medulloblastoma
Pediatric brain tumor
Oncogenic driver gene
Hedgehog pathway inhibitor
Smoothened receptor antagonist
Colocalization Strategy Unveils an Underside Binding Site in the Transmembrane Domain of Smoothened Receptor
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 21, 页码: 9983-9989
作者:
Zhou, Fang
;
Ding, Kang
;
Zhou, Yiqing
;
Liu, Yang
;
Liu, Xiaoyan
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2020/07/01
L-4, a Well-Tolerated and Orally Active Inhibitor of Hedgehog Pathway, Exhibited Potent Anti-tumor Effects Against Medulloblastoma in vitro and in vivo
期刊论文
FRONTIERS IN PHARMACOLOGY, 2019, 卷号: 10
作者:
Zhu, Mingfei
;
Wang, Hong
;
Wang, Chenglin
;
Fang, Yanfen
;
Zhu, Tong
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2019/12/05
L-4
hedgehog
Smo
medulloblastoma
D473H
Novel-smoothened inhibitors for therapeutic targeting of naive and drug-resistant hedgehog pathway-driven cancers
期刊论文
ACTA PHARMACOLOGICA SINICA, 2019, 卷号: 40, 期号: 2
作者:
Li, Qing-rou
;
Zhao, Hui
;
Zhang, Xue-sai
;
Lang, Henk
;
Yu, Ker
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2019/12/05
hedgehog
smoothened inhibitor
paracrine
acquired drug resistance
Biomimetic nanoparticles delivered hedgehog pathway inhibitor to modify tumour microenvironment and improved chemotherapy for pancreatic carcinoma
期刊论文
ARTIFICIAL CELLS NANOMEDICINE AND BIOTECHNOLOGY, 2018, 卷号: 46
作者:
Jiang, Ting
;
Zhang, Bo
;
Zhang, Long
;
Wu, Xuemei
;
Li, Haichun
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2019/12/05
Biomimetic nanoparticles
tumour microenvironment
cyclopamine
chemotherapy
pancreatic ductal adenocarcinomas
Cynanbungeigenin C and D, a pair of novel epimers from Cynanchum bungei, suppress hedgehog pathway-dependent medulloblastoma by blocking signaling at the level of Gli
期刊论文
CANCER LETTERS, 2018, 卷号: 420
作者:
Li, Xiao-Yu
;
Zhou, Li-Fei
;
Gao, Li-Juan
;
Wei, Yang
;
Xu, Shi-Fang
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2019/12/05
Hh pathway inhibitor
Gli inhibitor
Natural product
C-21 steroid
Medulloblastoma
Acquired resistance
Strategies to target the Hedgehog signaling pathway for cancer therapy
期刊论文
MEDICINAL RESEARCH REVIEWS, 2018, 卷号: 38, 页码: 870-913
作者:
Xin, Minhang
;
Ji, Xinyue
;
De La Cruz, Ladie Kimberly
;
Thareja, Suresh
;
Wang, Binghe
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2019/11/26
sonidegib
hedgehog signaling pathway
Hh inhibitor
basal cell carcinoma
vismodegib
CAT(3), a prodrug of 13a(S)-3-hydroxyl-6,7-dimethoxyphenanthro[9, 10-b]-indolizidine, circumvents temozolomide-resistant glioblastoma via the Hedgehog signaling pathway, independently of O-6-methylguanine DNA methyltransferase expression
期刊论文
2018, 卷号: 11, 页码: 3671-3684
作者:
Ji, Ming
;
Wang, Liyuan
;
Chen, Ju
;
Xue, Nina
;
Wang, Chunyang
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2020/01/03
Gli inhibitor
chemotherapy
lomeguatrib
xenograft tumor model
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