CORC

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Discovery of High-Affinity Inhibitors of the BPTF Bromodomain 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 16, 页码: 12075-12088
作者:  Lu, Tian;  Lu, Haibo;  Duan, Zhe;  Wang, Jun;  Han, Jie
收藏  |  浏览/下载:38/0  |  提交时间:2021/11/04
Recent Progress and Clinical Development of Inhibitors that Block MDM4/p53 Protein-Protein Interactions 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 15, 页码: 10621-10640
作者:  Zhang, Shiyan;  Lou, Jianfeng;  Li, Yafang;  Zhou, Feilong;  Yan, Ziqin
收藏  |  浏览/下载:63/0  |  提交时间:2021/11/04
Structure-Guided Development of Small-Molecule PRC2 Inhibitors Targeting EZH2-EED Interaction 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 12, 页码: 8194-8207
作者:  Du, Daohai;  Xu, Dandan;  Zhu, Licheng;  Stazi, Giulia;  Zwergel, Clemens
收藏  |  浏览/下载:74/0  |  提交时间:2021/08/17
Phage-Display Based Discovery and Characterization of Peptide Ligands against WDR5 期刊论文
MOLECULES, 2021, 卷号: 26, 期号: 5, 页码: 12
作者:  Cao, Jiawen;  Fan, Tiantian;  Li, Yanlian;  Du, Zhiyan;  Chen, Lin
收藏  |  浏览/下载:70/0  |  提交时间:2021/05/24
Kinetics-Driven Drug Design Strategy for Next-Generation Acetylcholinesterase Inhibitors to Clinical Candidate 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 4, 页码: 1844-1855
作者:  Zhou, Yu;  Fu, Yan;  Yin, Wanchao;  Li, Jian;  Wang, Wei
收藏  |  浏览/下载:21/0  |  提交时间:2021/05/24
Cocrystals to tune oily vitamin E into crystal vitamin E 期刊论文
INTERNATIONAL JOURNAL OF PHARMACEUTICS, 2021, 卷号: 592, 页码: 8
作者:  Zhu, Bingqing;  Zhang, Qi;  Lu, Liye;  Bao, Junjie;  Rong, Xiaoyi
收藏  |  浏览/下载:133/0  |  提交时间:2021/05/24
Crystallography-guided discovery of carbazole-based retinoic acid-related orphan receptor gamma-t (ROR gamma t) modulators: insights into different protein behaviors with "short" and "long" inverse agonists 期刊论文
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 11
作者:  Yu, Ming-cheng;  Yang, Feng;  Ding, Xiao-yu;  Sun, Nan-nan;  Jiang, Zheng-yuan
收藏  |  浏览/下载:85/0  |  提交时间:2020/12/24
Machine-Learning-Guided Cocrystal Prediction Based on Large Data Base 期刊论文
CRYSTAL GROWTH & DESIGN, 2020, 卷号: 20, 期号: 10, 页码: 6610-6621
作者:  Wang, Dingyan;  Yang, Zeen;  Zhu, Bingqing;  Mei, Xuefeng;  Luo, Xiaomin
收藏  |  浏览/下载:12/0  |  提交时间:2020/12/24
Tunable Mechanical and Optoelectronic Properties of Organic Cocrystals by Unexpected Stacking Transformation from H- to J- and X-Aggregation 期刊论文
ACS NANO, 2020, 卷号: 14, 期号: 8, 页码: 10704-10715
作者:  Ji, Wei;  Xue, Bin;  Bera, Santu;  Guerin, Sarah;  Liu, Yanqing
收藏  |  浏览/下载:12/0  |  提交时间:2020/10/30
The axial chirality hidden in vitamin D and its application in cocrystal prediction 期刊论文
CRYSTENGCOMM, 2020, 卷号: 22, 期号: 18, 页码: 3095-3099
作者:  Guo, Mengfei;  Zhang, Zaiyong;  Chen, Zhaoqiang;  Ding, Qiaoce;  Lu, Liye
收藏  |  浏览/下载:33/0  |  提交时间:2020/07/01


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