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Discovery of a novel DDRs kinase inhibitor XBLJ-13 for the treatment of idiopathic pulmonary fibrosis 期刊论文
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 11
作者:  Dong, Ying;  Tang, Bi-xi;  Wang, Qi;  Zhou, Li-wei;  Li, Cong
收藏  |  浏览/下载:77/0  |  提交时间:2022/01/04
DRAK2 aggravates nonalcoholic fatty liver disease progression through SRSF6-associated RNA alternative splicing 期刊论文
CELL METABOLISM, 2021, 卷号: 33, 期号: 10, 页码: 2004-+
作者:  Li, Yufeng;  Xu, Junyu;  Lu, Yuting;  Bian, Hua;  Yang, Lin
收藏  |  浏览/下载:23/0  |  提交时间:2022/01/18
Multi-omics characterization of WNT pathway reactivation to ameliorate BET inhibitor resistance in liver cancer cells 期刊论文
GENOMICS, 2021, 卷号: 113, 期号: 3, 页码: 1057-1069
作者:  Liu, Yuwei;  Xue, Mengzhu;  Cao, Danyan;  Qin, Lihuai;  Wang, Ying
收藏  |  浏览/下载:33/0  |  提交时间:2021/08/17
Phage-Display Based Discovery and Characterization of Peptide Ligands against WDR5 期刊论文
MOLECULES, 2021, 卷号: 26, 期号: 5, 页码: 12
作者:  Cao, Jiawen;  Fan, Tiantian;  Li, Yanlian;  Du, Zhiyan;  Chen, Lin
收藏  |  浏览/下载:70/0  |  提交时间:2021/05/24
Identification of SARS-CoV-2 entry inhibitors among already approved drugs 期刊论文
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 7
作者:  Yang, Li;  Pei, Rong-juan;  Li, Heng;  Ma, Xin-na;  Zhou, Yu
收藏  |  浏览/下载:43/0  |  提交时间:2020/12/24
Rational Design and Evaluation of 6-(Pyrimidin-2-ylamino)-3,4-dihydroquinoxalin-2(1H)-ones as Polypharmacological Inhibitors of BET and Kinases 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 17, 页码: 9787-9802
作者:  Lv, Kaikai;  Chen, Weicong;  Chen, Danqi;  Mou, Jie;  Zhang, Huijie
收藏  |  浏览/下载:12/0  |  提交时间:2020/12/21
Structural basis of ligand binding modes at the human formyl peptide receptor 2 期刊论文
NATURE COMMUNICATIONS, 2020, 卷号: 11, 期号: 1, 页码: 9
作者:  Chen, Tong;  Xiong, Muya;  Zong, Xin;  Ge, Yunjun;  Zhang, Hui
收藏  |  浏览/下载:11/0  |  提交时间:2020/12/24
Targeting Hsp90 with FS-108 circumvents gefitinib resistance in EGFR mutant non-small cell lung cancer cells (vol 37, pg 1587, 2020) 期刊论文
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 2
作者:  Wang, Yue-qin;  Shen, Ai-jun;  Sun, Jing-ya;  Wang, Xin;  Liu, Hong-chun
收藏  |  浏览/下载:12/0  |  提交时间:2020/07/01
Stewartiacids A-N, C-23 carboxylated triterpenoids from Chinese Stewartia and their inhibitory effects against ATP-citrate lyase and NF-kappa B 期刊论文
RSC ADVANCES, 2020, 卷号: 10, 期号: 6, 页码: 3343-3356
作者:  Wan, Jiang;  Zang, Yi;  Xiao, Dao-An;  Li, Na;  Li, Junmin
收藏  |  浏览/下载:22/0  |  提交时间:2020/07/01
Structure-Based Discovery and Development of a Series of Potent and Selective Bromodomain and Extra-Terminal Protein Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 18, 页码: 8642-8663
作者:  Hu, Jianping;  Tian, Chang-Qing;  Damaneh, Mohammadali Soleimani;  Li, Yanlian;  Cao, Danyan
收藏  |  浏览/下载:11/0  |  提交时间:2020/07/01


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