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科研机构
上海药物研究所 [20]
内容类型
期刊论文 [20]
发表日期
2020 [20]
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发表日期:2020
专题:上海药物研究所
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1-Phenyl-N-(benzothiazol-2-yl)methanimine derivatives as Middle East respiratory syndrome coronavirus inhibitors
期刊论文
RSC ADVANCES, 2020, 卷号: 10, 期号: 71, 页码: 43299-43311
作者:
Hu, Min-Qi
;
Li, Heng
;
Lin, Ying
;
Zhang, Ying
;
Tang, Jie
收藏
  |  
浏览/下载:51/0
  |  
提交时间:2021/05/24
Identification of SARS-CoV-2 entry inhibitors among already approved drugs
期刊论文
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 7
作者:
Yang, Li
;
Pei, Rong-juan
;
Li, Heng
;
Ma, Xin-na
;
Zhou, Yu
收藏
  |  
浏览/下载:42/0
  |  
提交时间:2020/12/24
COVID-19
SARS-CoV-2
virus entry inhibitors
high throughput screening assay
approved drug library
histamine receptor antagonists
clemastine
Chemical Constituents from Citrus changshan-huyou and Their Anti-Inflammatory Activities
期刊论文
CHEMISTRY & BIODIVERSITY, 2020, 页码: 10
作者:
Hu, Yu-Hong
;
Liu, Jin
;
Li, Heng
;
Tang, Wei
;
Li, Xu-Wen
收藏
  |  
浏览/下载:36/0
  |  
提交时间:2020/12/21
Citrus changshan-huyou
limonoids
structure modification
anti-inflammation
Manipulating the Click Reactivity of Dibenzoazacyclooctynes: From Azide Click Component to Caged Acylation Reagent by Silver Catalysis
期刊论文
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2020, 页码: 6
作者:
Shi, Wei
;
Tang, Feng
;
Ao, Jiwei
;
Yu, Qun
;
Liu, Junjie
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2020/12/21
acylation
click chemistry
peptides
rearrangements
silver
Extracellular Vesicle-Mediated Delivery of Circular RNA SCMH1 Promotes Functional Recovery in Rodent and Nonhuman Primate Ischemic Stroke Models
期刊论文
CIRCULATION, 2020, 卷号: 142, 期号: 6, 页码: 556-574
作者:
Yang, Li
;
Han, Bing
;
Zhang, Zhiting
;
Wang, Shuguo
;
Bai, Ying
收藏
  |  
浏览/下载:86/0
  |  
提交时间:2020/12/24
circular RNA
extracellular vesicles
MeCP2 protein
neuronal plasticity
primate
stroke
The artemisinin analog SM934 alleviates dry eye disease in rodent models by regulating TLR4/NF-kappa B/NLRP3 signaling
期刊论文
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 11
作者:
Yang, Fang-ming
;
Fan, Di
;
Yang, Xiao-qian
;
Zhu, Feng-hua
;
Shao, Mei-juan
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2020/12/24
dry eye disease
artemisinin derivative
beta-aminoarteether maleate
inflammation
macrophages
TLR4
inflammasome
Anti-SARS-CoV-2 activities in vitro of Shuanghuanglian preparations and bioactive ingredients
期刊论文
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 11
作者:
Su, Hai-xia
;
Yao, Sheng
;
Zhao, Wen-feng
;
Li, Min-jun
;
Liu, Jia
收藏
  |  
浏览/下载:115/0
  |  
提交时间:2020/12/24
SARS-CoV-2
3CL protease
traditional Chinese medicines
Shuanghuanglian oral liquid
baicalin
baicalein
Capsaicin derivatives with nitrothiophene substituents: Design, synthesis and antibacterial activity against multidrug-resistant S. aureus
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 198, 页码: 11
作者:
Wang, Zhi-Cheng
;
Wei, Bingyan
;
Pei, Fang-Ning
;
Yang, Teng
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2020/12/24
Capsaicin
Nitrothiophene
Multidrug-resistant S. aureus
Antibacterial agent
Selective Inhibition of STRN3-Containing PP2A Phosphatase Restores Hippo Tumor-Suppressor Activity in Gastric Cancer
期刊论文
CANCER CELL, 2020, 卷号: 38, 期号: 1, 页码: 115-+
作者:
Tang, Yang
;
Fang, Gemin
;
Guo, Fenghua
;
Zhang, Hui
;
Chen, Xiaoxu
收藏
  |  
浏览/下载:93/0
  |  
提交时间:2020/12/24
DC591017, a phosphodiesterase-4 (PDE4) inhibitor with robust anti-inflammation through regulating PKA-CREB signaling
期刊论文
BIOCHEMICAL PHARMACOLOGY, 2020, 卷号: 177, 页码: 15
作者:
Li, Heng
;
Li, Jian
;
Zhang, Xianglei
;
Feng, Chunlan
;
Fan, Chen
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2020/12/24
DC591017
PDE4
Inflammation
Macrophages
Dendritic cells
Psoriasis
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