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Pyrazolo[4,3-b]pyrimido[4,5-e][1,4]diazepine derivatives as new multi-targeted inhibitors of Aurora A/B and KDR 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 158, 页码: 428-441
作者:  Zhang, Qiumeng;  Shen, Qianqian;  Gao, Lixin;  Tong, Linjiang;  Li, Jia
收藏  |  浏览/下载:34/0  |  提交时间:2019/01/08
Design, Synthesis, and Biological Evaluation of Pyrimido[4,5-d]pyrimidine-2,4(1H,3H)-diones as Potent and Selective Epidermal Growth Factor Receptor (EGFR) Inhibitors against L858R/T790M Resistance Mutation 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 61, 期号: 13, 页码: 5609-5622
作者:  Hao, Yongjia;  Lyu, Jiankun;  Qu, Rong;  Tong, Yi;  Sun, Deheng
收藏  |  浏览/下载:61/0  |  提交时间:2019/01/08
Discovery of novel 2,4-diarylaminopyrimidine derivatives as potent and selective epidermal growth factor receptor (EGFR) inhibitors against L858R/T790M resistance mutation 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 152, 页码: 298-306
作者:  Yan, Qi;  Chen, Yuzhe;  Tang, Baiyou;  Xiao, Qiang;  Qu, Rong
收藏  |  浏览/下载:77/0  |  提交时间:2019/01/08
Discovery of 4,7-Diamino-5-(4-phenoxyphenyl)-6-methylene-pyrinnido[5,4-b]pyrrolizines as Novel Bruton's Tyrosine Kinase Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 61, 期号: 10, 页码: 4608-4627
作者:  Xue, Yu;  Song, Peiran;  Song, Zilan;  Wang, Aoli;  Tong, Linjiang
收藏  |  浏览/下载:32/0  |  提交时间:2019/08/23
Discovery of 4,7-Diamino-5-(4-phenoxyphenyl)-6-methylene-pyrinnido[5,4-b]pyrrolizines as Novel Bruton's Tyrosine Kinase Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 61, 期号: 10, 页码: 4608-4627
作者:  Xue, Yu;  Song, Peiran;  Song, Zilan;  Wang, Aoli;  Tong, Linjiang
收藏  |  浏览/下载:36/0  |  提交时间:2019/01/08
Design, Synthesis, and Structure-Activity Relationship Study of 2-Oxo-3,4-dihydropyrimido[4,5-d]pyrimidines as New Colony Stimulating Factor 1 Receptor (CSF1R) Kinase Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 61, 期号: 6, 页码: 2353-2371
作者:  Xun, Qiuju;  Zhang, Zhang;  Luo, Jinfeng;  Tong, Linjiang;  Huang, Minhao
收藏  |  浏览/下载:39/0  |  提交时间:2019/01/08
Discovery of novel 2,4-diarylaminopyrimidine derivatives as potent and selective epidermal growth factor receptor (EGFR) inhibitors against L858R/T790M resistance mutation 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 152
作者:  Yan, Qi;  Chen, Yuzhe;  Tang, Baiyou;  Xiao, Qiang;  Qu, Rong
收藏  |  浏览/下载:14/0  |  提交时间:2019/12/05
Design, Synthesis, and Structure-Activity Relationship Study of 2-Oxo-3,4-dihydropyrimido[4,5-d]pyrimidines as New Colony Stimulating Factor 1 Receptor (CSF1R) Kinase Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 61, 页码: 2353-2371
作者:  Xun, Qiuju[1];  Zhang, Zhang[2];  Luo, Jinfeng[3];  Tong, Linjiang[4];  Huang, Minhao[5]
收藏  |  浏览/下载:25/0  |  提交时间:2019/04/22
Design, Synthesis, and Structure-Activity Relationship Study of 2-Oxo-3,4-dihydropyrimido[4,5-d]pyrimidines as New Colony Stimulating Factor 1 Receptor (CSF1R) Kinase Inhibitors 期刊论文
2018, 卷号: 61, 期号: 6, 页码: 2353
作者:  Xun, Qiuju[1,2];  Zhang, Zhang[3];  Luo, Jinfeng[1];  Tong, Linjiang[6];  Huang, Minhao[1,2]
收藏  |  浏览/下载:16/0  |  提交时间:2019/12/10
Synthesis and Biological Activities of Novel 2-Aminobenzimidazoles EGFR~(T790M) Inhibitors 期刊论文
Chinese Journal of Synthetic Chemistry, 2018, 卷号: 26, 期号: 9, 页码: 637-646
作者:  Duan Jingyi;  Zhang Yinyong;  Qian Anran;  Tong Linjiang;  Xie Hua
收藏  |  浏览/下载:27/0  |  提交时间:2019/01/08


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