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科研机构
上海药物研究所 [7]
上海大学 [1]
暨南大学 [1]
复旦大学上海医学院 [1]
合肥物质科学研究院 [1]
内容类型
期刊论文 [11]
发表日期
2018 [11]
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Pyrazolo[4,3-b]pyrimido[4,5-e][1,4]diazepine derivatives as new multi-targeted inhibitors of Aurora A/B and KDR
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 158, 页码: 428-441
作者:
Zhang, Qiumeng
;
Shen, Qianqian
;
Gao, Lixin
;
Tong, Linjiang
;
Li, Jia
收藏
  |  
浏览/下载:34/0
  |  
提交时间:2019/01/08
Aurora A
Aurora B
KDR
Multi-targeted
Anticancer
Heterocyclic
Design, Synthesis, and Biological Evaluation of Pyrimido[4,5-d]pyrimidine-2,4(1H,3H)-diones as Potent and Selective Epidermal Growth Factor Receptor (EGFR) Inhibitors against L858R/T790M Resistance Mutation
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 61, 期号: 13, 页码: 5609-5622
作者:
Hao, Yongjia
;
Lyu, Jiankun
;
Qu, Rong
;
Tong, Yi
;
Sun, Deheng
收藏
  |  
浏览/下载:61/0
  |  
提交时间:2019/01/08
Discovery of novel 2,4-diarylaminopyrimidine derivatives as potent and selective epidermal growth factor receptor (EGFR) inhibitors against L858R/T790M resistance mutation
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 152, 页码: 298-306
作者:
Yan, Qi
;
Chen, Yuzhe
;
Tang, Baiyou
;
Xiao, Qiang
;
Qu, Rong
收藏
  |  
浏览/下载:77/0
  |  
提交时间:2019/01/08
EGFR inhibitors
Pyrimidine derivatives
Mutant selective inhibitors
AZD9291
T790M
Discovery of 4,7-Diamino-5-(4-phenoxyphenyl)-6-methylene-pyrinnido[5,4-b]pyrrolizines as Novel Bruton's Tyrosine Kinase Inhibitors
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 61, 期号: 10, 页码: 4608-4627
作者:
Xue, Yu
;
Song, Peiran
;
Song, Zilan
;
Wang, Aoli
;
Tong, Linjiang
收藏
  |  
浏览/下载:32/0
  |  
提交时间:2019/08/23
Discovery of 4,7-Diamino-5-(4-phenoxyphenyl)-6-methylene-pyrinnido[5,4-b]pyrrolizines as Novel Bruton's Tyrosine Kinase Inhibitors
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 61, 期号: 10, 页码: 4608-4627
作者:
Xue, Yu
;
Song, Peiran
;
Song, Zilan
;
Wang, Aoli
;
Tong, Linjiang
收藏
  |  
浏览/下载:36/0
  |  
提交时间:2019/01/08
Design, Synthesis, and Structure-Activity Relationship Study of 2-Oxo-3,4-dihydropyrimido[4,5-d]pyrimidines as New Colony Stimulating Factor 1 Receptor (CSF1R) Kinase Inhibitors
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 61, 期号: 6, 页码: 2353-2371
作者:
Xun, Qiuju
;
Zhang, Zhang
;
Luo, Jinfeng
;
Tong, Linjiang
;
Huang, Minhao
收藏
  |  
浏览/下载:39/0
  |  
提交时间:2019/01/08
Discovery of novel 2,4-diarylaminopyrimidine derivatives as potent and selective epidermal growth factor receptor (EGFR) inhibitors against L858R/T790M resistance mutation
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 152
作者:
Yan, Qi
;
Chen, Yuzhe
;
Tang, Baiyou
;
Xiao, Qiang
;
Qu, Rong
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2019/12/05
EGFR inhibitors
Pyrimidine derivatives
Mutant selective inhibitors
AZD9291
T790M
Design, Synthesis, and Structure-Activity Relationship Study of 2-Oxo-3,4-dihydropyrimido[4,5-d]pyrimidines as New Colony Stimulating Factor 1 Receptor (CSF1R) Kinase Inhibitors
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 61, 页码: 2353-2371
作者:
Xun, Qiuju[1]
;
Zhang, Zhang[2]
;
Luo, Jinfeng[3]
;
Tong, Linjiang[4]
;
Huang, Minhao[5]
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2019/04/22
Design, Synthesis, and Structure-Activity Relationship Study of 2-Oxo-3,4-dihydropyrimido[4,5-d]pyrimidines as New Colony Stimulating Factor 1 Receptor (CSF1R) Kinase Inhibitors
期刊论文
2018, 卷号: 61, 期号: 6, 页码: 2353
作者:
Xun, Qiuju[1,2]
;
Zhang, Zhang[3]
;
Luo, Jinfeng[1]
;
Tong, Linjiang[6]
;
Huang, Minhao[1,2]
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2019/12/10
Synthesis and Biological Activities of Novel 2-Aminobenzimidazoles EGFR~(T790M) Inhibitors
期刊论文
Chinese Journal of Synthetic Chemistry, 2018, 卷号: 26, 期号: 9, 页码: 637-646
作者:
Duan Jingyi
;
Zhang Yinyong
;
Qian Anran
;
Tong Linjiang
;
Xie Hua
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2019/01/08
1-fluoro-2-nitroarene
trans-4-aminocyclohexanol hydrochloride
2-aminobenzimidazole
EGFR~(T790M) inhibitor
synthesis
biological activity
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