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Distal mutation V486M disrupts the catalytic activity of DPP4 by affecting the flap of the propeller domain 期刊论文
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 9
作者:  Li, Teng-teng;  Peng, Cheng;  Wang, Ji-qiu;  Xu, Zhi-jian;  Su, Ming-bo
收藏  |  浏览/下载:42/0  |  提交时间:2022/01/18
Structural insights into hormone recognition by the human glucose-dependent insulinotropic polypeptide receptor 期刊论文
ELIFE, 2021, 卷号: 10, 页码: 20
作者:  Zhao, Fenghui;  Zhang, Chao;  Zhou, Qingtong;  Hang, Kaini;  Zou, Xinyu
收藏  |  浏览/下载:36/0  |  提交时间:2021/08/17
Cryo-EM structure of an activated VIP1 receptor-G protein complex revealed by a NanoBiT tethering strategy 期刊论文
NATURE COMMUNICATIONS, 2020, 卷号: 11, 期号: 1, 页码: 10
作者:  Duan, Jia;  Shen, Dan-dan;  Zhou, X. Edward;  Bi, Peng;  Liu, Qiu-feng
收藏  |  浏览/下载:24/0  |  提交时间:2020/12/24
Anti-SARS-CoV-2 activities in vitro of Shuanghuanglian preparations and bioactive ingredients 期刊论文
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 11
作者:  Su, Hai-xia;  Yao, Sheng;  Zhao, Wen-feng;  Li, Min-jun;  Liu, Jia
收藏  |  浏览/下载:115/0  |  提交时间:2020/12/24
Structural basis of ligand recognition and self-activation of orphan GPR52 期刊论文
NATURE, 2020, 页码: 21
作者:  Lin, Xi;  Li, Mingyue;  Wang, Niandong;  Wu, Yiran;  Luo, Zhipu
收藏  |  浏览/下载:178/0  |  提交时间:2020/07/01
Structures of AMP-activated protein kinase bound to novel pharmacological activators in phosphorylated, non-phosphorylated, and nucleotide-free states 期刊论文
JOURNAL OF BIOLOGICAL CHEMISTRY, 2019, 卷号: 294, 期号: 3, 页码: 953-967
作者:  Yan, Yan;  Zhou, X. Edward;  Novick, Scott J.;  Shaw, Simon J.;  Li, Yingwu
收藏  |  浏览/下载:13/0  |  提交时间:2020/07/01
Structural basis for ligand recognition of the human thromboxane A(2) receptor 期刊论文
NATURE CHEMICAL BIOLOGY, 2019, 卷号: 15, 期号: 1, 页码: 27-+
作者:  Fan, Hengxin;  Chen, Shuanghong;  Yuan, Xiaojing;  Han, Shuo;  Zhang, Hui
收藏  |  浏览/下载:89/0  |  提交时间:2019/01/08
Discovery of Potent Irreversible Pan-Fibroblast Growth Factor Receptor (FGFR) Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 61, 期号: 20, 页码: 9085-9104
作者:  Wang, Yuming;  Li, Lijun;  Fan, Jun;  Dai, Yang;  Jiang, Alan
收藏  |  浏览/下载:30/0  |  提交时间:2019/01/08
Two distinct domains of the glucagon-like peptide-1 receptor control peptide-mediated biased agonism 期刊论文
JOURNAL OF BIOLOGICAL CHEMISTRY, 2018, 卷号: 293, 期号: 24, 页码: 9370-9387
作者:  Lei, Saifei;  Clydesdale, Lachlan;  Dai, Antao;  Cai, Xiaoqing;  Feng, Yang
收藏  |  浏览/下载:52/0  |  提交时间:2019/01/08
Species-Specific Involvement of Integrin alpha IIb beta 3 in a Monoclonal Antibody CH12 Triggers Off-Target Thrombocytopenia in Cynomolgus Monkeys 期刊论文
MOLECULAR THERAPY, 2018, 卷号: 26, 期号: 6, 页码: 1457-1470
作者:  Zhang, Yiting;  Sun, Jianhua;  Tan, Minjia;  Liu, Yongzhen;  Li, Qian
收藏  |  浏览/下载:44/0  |  提交时间:2019/01/08


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