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科研机构
上海药物研究所 [95]
内容类型
期刊论文 [94]
学位论文 [1]
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2021 [6]
2020 [7]
2019 [3]
2018 [2]
2017 [9]
2016 [5]
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Chemistry [1]
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Synthesis and antiviral activity of 2 '-deoxy-6 '-substituted carbocyclic nucleosides
期刊论文
CHEMICAL BIOLOGY & DRUG DESIGN, 2021, 页码: 12
作者:
Xue, Haitao
;
Guo, Shuang
;
Hu, Tianwen
;
Wei, Daibao
;
Xie, Yuanchao
收藏
  |  
浏览/下载:39/0
  |  
提交时间:2022/01/18
2 '-deoxy carbocyclic nucleoside
antiviral activity
hepatitis B virus
Mitsunobu reaction
Discovery of an M-Substituted N-Cyclopropylmethyl-7 alpha-phenyl-6,14-endoethanotetrahydronorthebaine as a Selective, Potent, and Orally Active kappa-Opioid Receptor Agonist with an Improved Central Nervous System Safety Profile
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 16, 页码: 12414-12433
作者:
He, Qian
;
Wei, Yuanyuan
;
Liu, Xiao
;
Ye, Rongrong
;
Kong, Linghui
收藏
  |  
浏览/下载:88/0
  |  
提交时间:2021/11/04
Direct C4-Acetoxylation of Tryptophan and Tryptophan-Containing Peptides via Palladium(II)-Catalyzed C-H Activation
期刊论文
ORGANIC LETTERS, 2021, 卷号: 23, 期号: 12, 页码: 4699-4704
作者:
Zhang, Qiyu
;
Xie, Xiong
;
Peng, Jingjing
;
Chen, Feiyang
;
Ma, Jinyu
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2021/08/17
Rhodium-Catalyzed C-H Activation/Annulation Cascade of Aryl Oximes and Propargyl Alcohols to Isoquinoline N-Oxides
期刊论文
ADVANCED SYNTHESIS & CATALYSIS, 2021, 页码: 7
作者:
Li, Yuan
;
Fang, Feifei
;
Zhou, Jianhui
;
Li, Jiyuan
;
Wang, Run
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2021/08/17
Isoquinoline N-oxides
beta-hydroxy elimination
Rhodium
Secondary propargyl alcohols
Rh-Catalyzed cascade C-H activation/C-C cleavage/cyclization of carboxylic acids with cyclopropanols
期刊论文
CHEMICAL COMMUNICATIONS, 2021, 页码: 4
作者:
Wang, Siqi
;
Miao, Erfei
;
Wang, Hao
;
Song, Bichao
;
Huang, Wei
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2021/08/17
SYNTHESIS, CHARACTERIZATION, AND DRAK2 INHIBITORY ACTIVITIES OF HYDROXYAURONEDERIVATIVESURONE DERIVATIVES
期刊论文
HETEROCYCLES, 2021, 卷号: 102, 期号: 8, 页码: 1536-1551
作者:
Zhao, Mingsheng
;
Dai, Chengqiu
;
Li, Yi
;
Liu, Yinan
;
Li, Jing-Ya
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2022/01/04
Substitution Effect of the Trifluoromethyl Group on the Bioactivity in Medicinal Chemistry: Statistical Analysis and Energy Calculations
期刊论文
JOURNAL OF CHEMICAL INFORMATION AND MODELING, 2020, 卷号: 60, 期号: 12, 页码: 6242-6250
作者:
Abula, Amina
;
Xu, Zhijian
;
Zhu, Zhengdan
;
Peng, Cheng
;
Chen, Zhaoqiang
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  |  
浏览/下载:24/0
  |  
提交时间:2021/05/24
Rh(iii)-catalyzed tandem annulative redox-neutral arylation/amidation of aromatic tethered alkenes
期刊论文
CHEMICAL SCIENCE, 2020, 卷号: 11, 期号: 44, 页码: 12124-12129
作者:
Chen, Chao
;
Shi, Chen
;
Yang, Yaxi
;
Zhou, Bing
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2020/12/24
Crystallography-guided discovery of carbazole-based retinoic acid-related orphan receptor gamma-t (ROR gamma t) modulators: insights into different protein behaviors with "short" and "long" inverse agonists
期刊论文
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 11
作者:
Yu, Ming-cheng
;
Yang, Feng
;
Ding, Xiao-yu
;
Sun, Nan-nan
;
Jiang, Zheng-yuan
收藏
  |  
浏览/下载:85/0
  |  
提交时间:2020/12/24
RORγ
t
cocrystal structures
MD simulation
“
short”
inverse agonists
agonists
“
long”
inverse agonists
Ruthenium-Catalyzed C-H Activations for the Synthesis of Indole Derivatives
期刊论文
CATALYSTS, 2020, 卷号: 10, 期号: 11, 页码: 27
作者:
Zhu, Haoran
;
Zhao, Sen
;
Zhou, Yu
;
Li, Chunpu
;
Liu, Hong
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2021/05/24
ruthenium
C-H activation
indole
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