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Synthesis and antiviral activity of 2 '-deoxy-6 '-substituted carbocyclic nucleosides 期刊论文
CHEMICAL BIOLOGY & DRUG DESIGN, 2021, 页码: 12
作者:  Xue, Haitao;  Guo, Shuang;  Hu, Tianwen;  Wei, Daibao;  Xie, Yuanchao
收藏  |  浏览/下载:39/0  |  提交时间:2022/01/18
Discovery of an M-Substituted N-Cyclopropylmethyl-7 alpha-phenyl-6,14-endoethanotetrahydronorthebaine as a Selective, Potent, and Orally Active kappa-Opioid Receptor Agonist with an Improved Central Nervous System Safety Profile 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 16, 页码: 12414-12433
作者:  He, Qian;  Wei, Yuanyuan;  Liu, Xiao;  Ye, Rongrong;  Kong, Linghui
收藏  |  浏览/下载:88/0  |  提交时间:2021/11/04
Direct C4-Acetoxylation of Tryptophan and Tryptophan-Containing Peptides via Palladium(II)-Catalyzed C-H Activation 期刊论文
ORGANIC LETTERS, 2021, 卷号: 23, 期号: 12, 页码: 4699-4704
作者:  Zhang, Qiyu;  Xie, Xiong;  Peng, Jingjing;  Chen, Feiyang;  Ma, Jinyu
收藏  |  浏览/下载:28/0  |  提交时间:2021/08/17
Rhodium-Catalyzed C-H Activation/Annulation Cascade of Aryl Oximes and Propargyl Alcohols to Isoquinoline N-Oxides 期刊论文
ADVANCED SYNTHESIS & CATALYSIS, 2021, 页码: 7
作者:  Li, Yuan;  Fang, Feifei;  Zhou, Jianhui;  Li, Jiyuan;  Wang, Run
收藏  |  浏览/下载:17/0  |  提交时间:2021/08/17
Rh-Catalyzed cascade C-H activation/C-C cleavage/cyclization of carboxylic acids with cyclopropanols 期刊论文
CHEMICAL COMMUNICATIONS, 2021, 页码: 4
作者:  Wang, Siqi;  Miao, Erfei;  Wang, Hao;  Song, Bichao;  Huang, Wei
收藏  |  浏览/下载:25/0  |  提交时间:2021/08/17
SYNTHESIS, CHARACTERIZATION, AND DRAK2 INHIBITORY ACTIVITIES OF HYDROXYAURONEDERIVATIVESURONE DERIVATIVES 期刊论文
HETEROCYCLES, 2021, 卷号: 102, 期号: 8, 页码: 1536-1551
作者:  Zhao, Mingsheng;  Dai, Chengqiu;  Li, Yi;  Liu, Yinan;  Li, Jing-Ya
收藏  |  浏览/下载:9/0  |  提交时间:2022/01/04
Substitution Effect of the Trifluoromethyl Group on the Bioactivity in Medicinal Chemistry: Statistical Analysis and Energy Calculations 期刊论文
JOURNAL OF CHEMICAL INFORMATION AND MODELING, 2020, 卷号: 60, 期号: 12, 页码: 6242-6250
作者:  Abula, Amina;  Xu, Zhijian;  Zhu, Zhengdan;  Peng, Cheng;  Chen, Zhaoqiang
收藏  |  浏览/下载:24/0  |  提交时间:2021/05/24
Rh(iii)-catalyzed tandem annulative redox-neutral arylation/amidation of aromatic tethered alkenes 期刊论文
CHEMICAL SCIENCE, 2020, 卷号: 11, 期号: 44, 页码: 12124-12129
作者:  Chen, Chao;  Shi, Chen;  Yang, Yaxi;  Zhou, Bing
收藏  |  浏览/下载:13/0  |  提交时间:2020/12/24
Crystallography-guided discovery of carbazole-based retinoic acid-related orphan receptor gamma-t (ROR gamma t) modulators: insights into different protein behaviors with "short" and "long" inverse agonists 期刊论文
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 11
作者:  Yu, Ming-cheng;  Yang, Feng;  Ding, Xiao-yu;  Sun, Nan-nan;  Jiang, Zheng-yuan
收藏  |  浏览/下载:85/0  |  提交时间:2020/12/24
Ruthenium-Catalyzed C-H Activations for the Synthesis of Indole Derivatives 期刊论文
CATALYSTS, 2020, 卷号: 10, 期号: 11, 页码: 27
作者:  Zhu, Haoran;  Zhao, Sen;  Zhou, Yu;  Li, Chunpu;  Liu, Hong
收藏  |  浏览/下载:7/0  |  提交时间:2021/05/24


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