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Optimized HSP90 mediated fluorescent probes for cancer-specific bioimaging 期刊论文
JOURNAL OF MATERIALS CHEMISTRY B, 2020, 卷号: 8, 期号: 9, 页码: 1878-1896
作者:  Zhu, Shulei;  Li, Yalei;  Huang, Yushu;  Zhang, Minmin;  Gu, Xiaofan
收藏  |  浏览/下载:27/0  |  提交时间:2020/07/01
Design, Synthesis and Pharmacological Evaluation of Novel Hsp90N-terminal Inhibitors Without Induction of Heat Shock Response 期刊论文
CHEMISTRYOPEN, 2019, 卷号: 8, 期号: 3, 页码: 344-353
作者:  Liu, Peng;  Chen, Xiangling;  Zhu, Jianming;  Li, Bo;  Chen, Zhaoqiang
收藏  |  浏览/下载:33/0  |  提交时间:2020/07/01
Inhibition of HSP90 beta Improves Lipid Disorders by Promoting Mature SREBPs Degradation via the Ubiquitin-proteasome System 期刊论文
THERANOSTICS, 2019, 卷号: 9, 期号: 20, 页码: 5769-5783
作者:  Zheng, Zu-Guo;  Zhang, Xin;  Liu, Xiao-Xiao;  Jin, Xiu-Xiu;  Dai, Lunzhi
收藏  |  浏览/下载:17/0  |  提交时间:2020/07/01
Discovery of FS36 as a Novel Human Hsp90 Inhibitor 期刊论文
PROGRESS IN BIOCHEMISTRY AND BIOPHYSICS, 2018, 卷号: 45, 期号: 7, 页码: 736-744
作者:  Li Gen;  Lu Kai-Kai;  Li Jian;  Yin Xiu-Shan;  Zhao Dong
收藏  |  浏览/下载:21/0  |  提交时间:2019/01/08
Design, synthesis and pharmacological evaluation of ALK and Hsp90 dual inhibitors bearing resorcinol and 2,4-diaminopyrimidine motifs 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 152, 页码: 76-86
作者:  Geng, Kaijun;  Liu, Hongchun;  Song, Zilan;  Zhang, Chi;  Zhang, Minmin
收藏  |  浏览/下载:177/0  |  提交时间:2019/01/08
Identification and therapeutic intervention of coactivated anaplastic lymphoma kinase, fibroblast growth factor receptor 2, and ephrin type-A receptor 5 kinases in hepatocellular carcinoma 期刊论文
Hepatology (Baltimore, Md.), 2018
作者:  Wang, Xin;  Zhang, Minmin;  Ping, Fangfang;  Liu, Hongchun;  Sun, Jingya
收藏  |  浏览/下载:56/0  |  提交时间:2019/01/08
Dynamics revelation of conformational changes and binding modes of heat shock protein 90 induced by inhibitor associations 期刊论文
RSC ADVANCES, 2018, 卷号: 8, 期号: 45, 页码: 25456-25467
作者:  Chen, Jianzhong;  Wang, Jinan;  Lai, Fengbo;  Wang, Wei;  Pang, Laixue
收藏  |  浏览/下载:26/0  |  提交时间:2019/01/08
Design, synthesis and pharmacological evaluation of 4,5-diarylisoxazols bearing amino acid residues within the 3-amido motif as potent heat shock protein 90 (Hsp90) inhibitors 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 125, 页码: 315-326
作者:  Zhang, Chi;  Wang, Xin;  Liu, Hongchun;  Zhang, Minmin;  Geng, Meiyu
收藏  |  浏览/下载:51/0  |  提交时间:2019/01/08
Targeting Hsp90 with FS-108 circumvents gefitinib resistance in EGFR mutant non-small cell lung cancer cells 期刊论文
ACTA PHARMACOLOGICA SINICA, 2016, 卷号: 37, 期号: 12, 页码: 1587-1596
作者:  Wang, Yue-qin;  Shen, Ai-jun;  Sun, Jing-ya;  Wang, Xin;  Liu, Hong-chun
收藏  |  浏览/下载:31/0  |  提交时间:2019/01/08
Regulation of Ubiquitin-like with Plant Homeodomain and RING Finger Domain 1 (UHRF1) Protein Stability by Heat Shock Protein 90 Chaperone Machinery 期刊论文
JOURNAL OF BIOLOGICAL CHEMISTRY, 2016, 卷号: 291, 期号: 38, 页码: 20125-20135
作者:  Ding, Guangjin;  Chen, Peilin;  Zhang, Hui;  Huang, Xiaojie;  Zang, Yi
收藏  |  浏览/下载:15/0  |  提交时间:2019/01/08


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