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Site-specific protein modification by 3-n-butylphthalide in primary hepatocytes: Covalent protein adducts diminished by glutathione and N-acetylcysteine 期刊论文
LIFE SCIENCES, 2021, 卷号: 287, 页码: 14
作者:  Xue, Yaru;  Ren, Xuelian;  Zhu, Zhengdan;  Lei, Peng;  Liu, Mengling
收藏  |  浏览/下载:39/0  |  提交时间:2022/01/18
Covalent sortase A inhibitor ML346 prevents Staphylococcus aureus infection of Galleria mellonella 期刊论文
RSC MEDICINAL CHEMISTRY, 2021, 页码: 12
作者:  Guan, Xiang-Na;  Zhang, Tao;  Yang, Teng;  Dong, Ze;  Yang, Song
收藏  |  浏览/下载:21/0  |  提交时间:2021/12/16
A facile method for vancomycin C-terminus functionalization and derivatization through hydrazide 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2021, 卷号: 42, 页码: 6
作者:  Hu, Yu;  Zou, Xiangman;  Shi, Weiwei;  Ma, Chenhui;  Chen, Feifei
收藏  |  浏览/下载:17/0  |  提交时间:2021/08/17
Substitution Effect of the Trifluoromethyl Group on the Bioactivity in Medicinal Chemistry: Statistical Analysis and Energy Calculations 期刊论文
JOURNAL OF CHEMICAL INFORMATION AND MODELING, 2020, 卷号: 60, 期号: 12, 页码: 6242-6250
作者:  Abula, Amina;  Xu, Zhijian;  Zhu, Zhengdan;  Peng, Cheng;  Chen, Zhaoqiang
收藏  |  浏览/下载:25/0  |  提交时间:2021/05/24
Targeted Proteomics Combined with Affinity Mass Spectrometry Analysis Reveals Antagonist E7 Acts As an Intracellular Covalent Ligand of Orphan Receptor GPR52 期刊论文
ACS CHEMICAL BIOLOGY, 2020, 卷号: 15, 期号: 12, 页码: 3275-3284
作者:  Ma, Mengna;  Guo, Shimeng;  Lin, Xi;  Li, Shanshan;  Wu, Yiran
收藏  |  浏览/下载:16/0  |  提交时间:2021/05/24
Covalent Inhibitors Allosterically Block the Activation of Rho Family Proteins and Suppress Cancer Cell Invasion 期刊论文
ADVANCED SCIENCE, 2020, 页码: 13
作者:  Sun, Zhongya;  Zhang, Hao;  Zhang, Yuanyuan;  Liao, Liping;  Zhou, Wen
收藏  |  浏览/下载:107/0  |  提交时间:2020/07/01
2-Oxo-3,4-dihydropyrimido[4,5-d] pyrimidines as new reversible inhibitors of EGFR C797S (Cys797 to Ser797) mutant 期刊论文
CHINESE CHEMICAL LETTERS, 2020, 卷号: 31, 期号: 5, 页码: 1281-1287
作者:  Hu, Xianglong;  Xun, Qiuju;  Zhang, Tao;  Zhu, Su-Jie;  Li, Qian
收藏  |  浏览/下载:47/0  |  提交时间:2020/07/01
Xanthatin inhibits STAT3 and NF-kappa B signalling by covalently binding to JAK and IKK kinases 期刊论文
JOURNAL OF CELLULAR AND MOLECULAR MEDICINE, 2019, 卷号: 23, 期号: 6, 页码: 4301-4312
作者:  Liu, Man;  Xiao, Cheng-qian;  Sun, Ming-wei;  Tan, Min-jia;  Hu, Li-hong
收藏  |  浏览/下载:7/0  |  提交时间:2020/07/01
Parthenolide Inhibits STAT3 Signaling by Covalently Targeting Janus Kinases 期刊论文
MOLECULES, 2018, 卷号: 23, 期号: 6
作者:  Liu, Man;  Xiao, Chengqian;  Sun, Mingwei;  Tan, Minjia;  Hu, Lihong
收藏  |  浏览/下载:33/0  |  提交时间:2019/01/08
Discovery of 4,7-Diamino-5-(4-phenoxyphenyl)-6-methylene-pyrinnido[5,4-b]pyrrolizines as Novel Bruton's Tyrosine Kinase Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 61, 期号: 10, 页码: 4608-4627
作者:  Xue, Yu;  Song, Peiran;  Song, Zilan;  Wang, Aoli;  Tong, Linjiang
收藏  |  浏览/下载:36/0  |  提交时间:2019/01/08


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