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Synthesis and biological evaluation of 2,5-diaryl-1,3,4-oxadiazole derivatives as novel Src homology 2 domain-containing protein tyrosine phosphatase 2 (SHP2) inhibitors 期刊论文
BIOORGANIC CHEMISTRY, 2021, 卷号: 116, 页码: 13
作者:  Meng, Xiang-Dong;  Gao, Li-Xin;  Wang, Zhi-Jia;  Feng, Bo;  Zhang, Chun
收藏  |  浏览/下载:30/0  |  提交时间:2021/12/01
Synthesis and Protein Tyrosine Phosphatase 1B (PTP1B) Inhibitory Activity Evaluation of Novel N-Acylhydrazone Derivatives Containing Carbazole and Aromatic Ring/Aromatic Fused Heterocycle 期刊论文
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2021, 卷号: 41, 期号: 9, 页码: 3593-3607
作者:  Li Yingjun;  Lin Ledi;  Liu Jihong;  Gao Lixin;  Sheng Li
收藏  |  浏览/下载:18/0  |  提交时间:2021/12/01
Rearranged Diels-Alder Adducts and Prenylated Flavonoids as Potential PTP1B Inhibitors from Morus nigra 期刊论文
JOURNAL OF NATURAL PRODUCTS, 2021, 卷号: 84, 期号: 8, 页码: 2303-2311
作者:  Qu, Ke-Jun;  Wang, Bin;  Jiang, Chang-Sheng;  Xie, Bao-Gang;  Liu, Ai-Hong
收藏  |  浏览/下载:41/0  |  提交时间:2021/11/04
Synthesis and Protein Tyrosine Phosphatase 1B (PTP1B) Inhibitory Activity Evaluation of Novel Arylaminoacetylhydrazone Derivatives Containing Carbazole Moiety 期刊论文
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2021, 卷号: 41, 期号: 8, 页码: 3157-3170
作者:  Li Yingjun;  Lin Ledi;  Jin Kun;  Gao Lixin;  Sheng Li
收藏  |  浏览/下载:19/0  |  提交时间:2021/11/04
The Two Formyl Peptide Receptors Differently Regulate GPR84-Mediated Neutrophil NADPH Oxidase Activity 期刊论文
JOURNAL OF INNATE IMMUNITY, 2021, 页码: 15
作者:  Martensson, Jonas;  Sundqvist, Martina;  Manandhar, Asmita;  Leremias, Loukas;  Zhang, Linjie
收藏  |  浏览/下载:41/0  |  提交时间:2021/05/24
SL010110, a lead compound, inhibits gluconeogenesis via SIRT2-p300-mediated PEPCK1 degradation and improves glucose homeostasis in diabetic mice 期刊论文
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 13
作者:  Ren, Yu-ran;  Ye, Yang-liang;  Feng, Ying;  Xu, Ti-fei;  Shen, Yu
收藏  |  浏览/下载:22/0  |  提交时间:2021/05/24
Synthesis and Protein Tyrosine Phosphatase 1B (PTP1B) Inhibitory Activity Evaluation of Novel Carbazole-Based Carbohydrazone Derivatives 期刊论文
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2020, 卷号: 40, 期号: 2, 页码: 478-488
作者:  Li, Yingjun;  Liu, Xuejie;  Liu, Jihong;  Gao, Lixin;  Jin, Kun
收藏  |  浏览/下载:44/0  |  提交时间:2020/07/01
Alleviation of Synovial Inflammation of Juanbi-Tang on Collagen-Induced Arthritis and TNF-Tg Mice Model 期刊论文
FRONTIERS IN PHARMACOLOGY, 2020, 卷号: 11, 页码: 17
作者:  Wang, Tengteng;  Jia, Qingyun;  Chen, Tao;  Yin, Hao;  Tian, Xiaoting
收藏  |  浏览/下载:31/0  |  提交时间:2020/07/01
Phytochemical and biological studies on rare and endangered plants endemic to China. Part XIV. Structurally diverse terpenoids from the twigs and needles of the endangered plant Picea brachytyla 期刊论文
PHYTOCHEMISTRY, 2020, 卷号: 169, 页码: 11
作者:  Jiang, Wei;  Xiong, Juan;  Zang, Yi;  Li, Junmin;  Osman, Ezzat E. A.
收藏  |  浏览/下载:83/0  |  提交时间:2020/07/01
3,6-二取代三唑并噻二唑衍生物的合成及其对细胞分裂周期25B磷酸酶和蛋白酪氨酸磷酸酶1B抑制活性评价 期刊论文
应用化学, 2020, 卷号: 37, 期号: 9, 页码: 994
作者:  李英俊;  杨鸿境;  曹欣;  高立信;  靳焜
收藏  |  浏览/下载:31/0  |  提交时间:2020/12/24


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