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Kinetics-Driven Drug Design Strategy for Next-Generation Acetylcholinesterase Inhibitors to Clinical Candidate 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 4, 页码: 1844-1855
作者:  Zhou, Yu;  Fu, Yan;  Yin, Wanchao;  Li, Jian;  Wang, Wei
收藏  |  浏览/下载:21/0  |  提交时间:2021/05/24
[1,5]-Hydride Shift-Cyclization versus C(sp(2))-H Functionalization in the Knoevenagel-Cyclization Domino Reactions of 1,4-and 1,5-Benzoxazepines 期刊论文
MOLECULES, 2020, 卷号: 25, 期号: 6, 页码: 19
作者:  Vargane, Dora Szaloki;  Toth, Laszlo;  Buglyo, Balazs;  Kiss-Szikszai, Attila;  Mandi, Attila
收藏  |  浏览/下载:38/0  |  提交时间:2020/07/01
Discovery and Biological Evaluation of New Selective Acetylcholinesterase Inhibitors with Anti-A beta Aggregation Activity through Molecular Docking-Based Virtual Screening 期刊论文
CHEMICAL & PHARMACEUTICAL BULLETIN, 2020, 卷号: 68, 期号: 2, 页码: 161-166
作者:  Liu, Guangpu;  Jiao, Yang;  Lin, Yongqiang;  Hao, Haifang;  Dou, Yanli
收藏  |  浏览/下载:55/0  |  提交时间:2020/07/01
Donepezil, a drug for Alzheimer's disease, promotes oligodendrocyte generation and remyelination 期刊论文
ACTA PHARMACOLOGICA SINICA, 2019, 卷号: 40, 期号: 11, 页码: 1386-1393
作者:  Cui, Xue;  Guo, Yu-e;  Fang, Jia-hui;  Shi, Chang-jie;  Suo, Na
收藏  |  浏览/下载:70/0  |  提交时间:2020/07/01
Discovery of New Selective Butyrylcholinesterase (BChE) Inhibitors with Anti-A beta Aggregation Activity: Structure-Based Virtual Screening, Hit Optimization and Biological Evaluation 期刊论文
MOLECULES, 2019, 卷号: 24, 期号: 14, 页码: 21
作者:  Jiang, Cheng-Shi;  Ge, Yong-Xi;  Cheng, Zhi-Qiang;  Wang, Yin-Yin;  Tao, Hong-Rui
收藏  |  浏览/下载:14/0  |  提交时间:2020/07/01
Discovery of new multifunctional selective acetylcholinesterase inhibitors: structure-based virtual screening and biological evaluation 期刊论文
JOURNAL OF COMPUTER-AIDED MOLECULAR DESIGN, 2019, 卷号: 33, 期号: 5, 页码: 521-530
作者:  Jiang, Cheng-Shi;  Ge, Yong-Xi;  Cheng, Zhi-Qiang;  Song, Jia-Li;  Wang, Yin-Yin
收藏  |  浏览/下载:12/0  |  提交时间:2020/07/01
donepeziladrugforalzheimersdiseasepromotesoligodendrocytegenerationandremyelination 期刊论文
actapharmacologicasinica, 2019, 卷号: 40, 期号: 11, 页码: 1386
作者:  Cui Xue;  Guo Yue;  Fang Jiahui;  Shi Changjie;  Suo Na
收藏  |  浏览/下载:58/0  |  提交时间:2020/07/01
Reconsideration of Anticholinesterase Therapeutic Strategies against Alzheimer's Disease 期刊论文
ACS chemical neuroscience, 2018
作者:  Wang, Huan;  Zhang, Haiyan
收藏  |  浏览/下载:58/0  |  提交时间:2019/01/08
Molecular-docking-guided design and synthesis of new IAA-tacrine hybrids as multifunctional AChE/BChE inhibitors 期刊论文
Bioorganic chemistry, 2018, 卷号: 83, 页码: 277-288
作者:  Cheng, Zhi-Qiang;  Zhu, Kong-Kai;  Zhang, Juan;  Song, Jia-Li;  Muehlmann, Luis Alexandre
收藏  |  浏览/下载:49/0  |  提交时间:2019/01/08
Rational Design of Novel Selective Dual-Target Inhibitors of Acetylcholinesterase and Monoamine Oxidase B as Potential Anti-Alzheimer's Disease Agents 期刊论文
ACS chemical neuroscience, 2018
作者:  Xu, Yixiang;  Zhang, Jian;  Wang, Huan;  Mao, Fei;  Bao, Keting
收藏  |  浏览/下载:85/0  |  提交时间:2019/01/08


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