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Targeting epigenetic machinery: Emerging novel allosteric inhibitors 期刊论文
PHARMACOLOGY & THERAPEUTICS, 2019, 卷号: 204, 页码: 24
作者:  Ye, Fei;  Huang, Jing;  Wang, Hongbo;  Luo, Cheng;  Zhao, Kehao
收藏  |  浏览/下载:20/0  |  提交时间:2020/07/01
C10ORF12 modulates PRC2 histone methyltransferase activity and H3K27me3 levels 期刊论文
ACTA PHARMACOLOGICA SINICA, 2019, 卷号: 40, 期号: 11, 页码: 1457-1465
作者:  Shi, Yi;  Ma, Hong-lei;  Zhuang, You-wen;  Wang, Xiao-xi;  Jiang, Yi
收藏  |  浏览/下载:35/0  |  提交时间:2020/07/01
Aptamer functionalized magnetic graphene oxide nanocomposites for highly selective capture of histones 期刊论文
ELECTROPHORESIS, 2019, 卷号: 40, 期号: 16-17, 页码: 2135-2141
作者:  Chen, Yuanbo;  Jiang, Bo;  Hu, Yechen;  Deng, Nan;  Zhao, Baofeng
收藏  |  浏览/下载:80/0  |  提交时间:2019/12/02
Inhibition of G9a by a small molecule inhibitor, UNC0642, induces apoptosis of human bladder cancer cells 期刊论文
ACTA PHARMACOLOGICA SINICA, 2019, 卷号: 40, 期号: 8, 页码: 1076-1084
作者:  Cao, Yue-peng;  Sun, Jing-ya;  Li, Mei-qian;  Dong, Yu;  Zhang, Yuan-heng
收藏  |  浏览/下载:17/0  |  提交时间:2020/07/01
Design and Synthesis of Potent, Selective Inhibitors of Protein Arginine Methyltransferase 4 against Acute Myeloid Leukemia 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 11, 页码: 5414-5433
作者:  Guo, Zuhao;  Zhang, Zhuqing;  Yang, Hong;  Cao, Danyan;  Xu, Xiaowei
收藏  |  浏览/下载:16/0  |  提交时间:2020/07/01
Stella protein facilitates DNA demethylation by disrupting the chromatin association of the RING finger-type E3 ubiquitin ligase UHRF1 期刊论文
JOURNAL OF BIOLOGICAL CHEMISTRY, 2019, 卷号: 294, 期号: 22, 页码: 8907-8917
作者:  Du, Wenlong;  Dong, Qiang;  Zhang, Zhuqiang;  Liu, Baodong;  Zhou, Ting
收藏  |  浏览/下载:18/0  |  提交时间:2020/10/21
Inhibition of Ezh2 In Vitro and the Decline of Ezh2 in Developing Midbrain Promote Dopaminergic Neurons Differentiation Through Modifying H3K27me3 期刊论文
STEM CELLS AND DEVELOPMENT, 2019, 卷号: 28, 期号: 10, 页码: 649-658
作者:  Hong, Feng;  Zhao, Mengxue;  Zhang, Lei;  Feng, Linyin
收藏  |  浏览/下载:23/0  |  提交时间:2020/07/01
The dynamic conformational landscape of the protein methyltransferase SETD8 期刊论文
ELIFE, 2019, 卷号: 8, 页码: 76
作者:  Chen, Shi;  Wiewiora, Rafal P.;  Meng, Fanwang;  Babault, Nicolas;  Ma, Anqi
收藏  |  浏览/下载:11/0  |  提交时间:2020/07/01
Epigenetic changes: An emerging potential pharmacological target in allergic rhinitis 期刊论文
INTERNATIONAL IMMUNOPHARMACOLOGY, 2019, 卷号: 71
作者:  Yang, Jingpu;  Zhong, Wei;  Xue, Kai;  Wang, Zonggui
收藏  |  浏览/下载:17/0  |  提交时间:2019/12/05
Genome-wide target interactome profiling reveals a novel EEF1A1 epigenetic pathway for oncogenic lncRNA MALAT1 in breast cancer 期刊论文
AMERICAN JOURNAL OF CANCER RESEARCH, 2019, 卷号: 9, 期号: 4
作者:  Wang, Cong;  Li, Wei;  Hu, Ji-Fan;  Cui, Jiuwei;  Hoffman, Andrew R.
收藏  |  浏览/下载:27/0  |  提交时间:2019/12/05


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