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Design and synthesis of Atglistatin derivatives as adipose triglyceride lipase inhibitors 期刊论文
CHEMICAL BIOLOGY & DRUG DESIGN, 2017, 卷号: 90, 期号: 6, 页码: 1122-1133
作者:  Jin, Jiyu;  Huang, Suling
收藏  |  浏览/下载:20/0  |  提交时间:2019/01/08
Discovery of alkyl bis(oxy)dibenzimidamide derivatives as novel protein arginine methyltransferase 1 (PRMT1) inhibitors 期刊论文
CHEMICAL BIOLOGY & DRUG DESIGN, 2017, 卷号: 90, 期号: 6, 页码: 1260-1270
作者:  Zhang, Wei-yao;  Lu, Wen-chao;  Jiang, Hao;  Lv, Zheng-bing;  Xie, Yi-qian
收藏  |  浏览/下载:32/0  |  提交时间:2019/01/08
PI-273, a Substrate-Competitive, Specific Small-Molecule Inhibitor of PI4KII alpha, Inhibits the Growth of Breast Cancer Cells 期刊论文
CANCER RESEARCH, 2017, 卷号: 77, 期号: 22, 页码: 6253-6266
作者:  Li, Jiangmei;  Gao, Zhen;  Zhao, Dan;  Zhang, Lunfeng;  Qiao, Xinhua
收藏  |  浏览/下载:24/0  |  提交时间:2019/01/08
SIRT7 deacetylates DDB1 and suppresses the activity of the CRL4 E3 ligase complexes 期刊论文
FEBS JOURNAL, 2017, 卷号: 284, 期号: 21, 页码: 3619-3636
作者:  Mo, Yan;  Lin, Ran;  Liu, Peng;  Tan, Minjia;  Xiong, Yue
收藏  |  浏览/下载:28/0  |  提交时间:2019/01/08
Evaluation of in vitro and in vivo activity of a multityrosine kinase inhibitor, AL3810, against human thyroid cancer 期刊论文
ACTA PHARMACOLOGICA SINICA, 2017, 卷号: 38, 期号: 11, 页码: 1533-1542
作者:  Xie, Qin;  Chen, Hui;  Ai, Jing;  Gao, Ying-lei;  Geng, Mei-yu
收藏  |  浏览/下载:17/0  |  提交时间:2019/01/08
Discovery of a series of dihydroquinoxalin-2(1H)-ones as selective BET inhibitors from a dual PLK1-BRD4 inhibitor 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 137, 页码: 176-195
作者:  Hu, Jianping;  Wang, Yingqing;  Li, Yanlian;  Xu, Lin;  Cao, Danyan
收藏  |  浏览/下载:32/0  |  提交时间:2019/01/08
Selective targeting p53(WT) lung cancer cells harboring homozygous p53 Arg72 by an inhibitor of CypA 期刊论文
ONCOGENE, 2017, 卷号: 36, 期号: 33, 页码: 4719-4731
作者:  Lu, W.;  Cheng, F.;  Yan, W.;  Li, X.;  Yao, X.
收藏  |  浏览/下载:8/0  |  提交时间:2019/01/08
Selective ATP hydrolysis inhibition in F1Fo ATP synthase enhances radiosensitivity in non-small-cell lung cancer cells (A549) 期刊论文
ONCOTARGET, 2017, 卷号: 8, 页码: 53602-53612
作者:  Zhang, Hong;  Wang, Yupei;  Hou, Qinzheng;  Xiao, Guoqing;  Yang, Shifeng
收藏  |  浏览/下载:11/0  |  提交时间:2018/05/31
LX2343 alleviates cognitive impairments in AD model rats by inhibiting oxidative stress-induced neuronal apoptosis and tauopathy 期刊论文
ACTA PHARMACOLOGICA SINICA, 2017, 卷号: 38, 期号: 8, 页码: 1104-1119
作者:  Guo, Xiao-dan;  Sun, Guang-long;  Zhou, Ting-ting;  Wang, Yi-yang;  Xu, Xin
收藏  |  浏览/下载:36/0  |  提交时间:2019/01/08
A Fusion Protein of the p53 Transaction Domain and the p53-Binding Domain of the Oncoprotein MdmX as an Efficient System for High-Throughput Screening of MdmX Inhibitors 期刊论文
BIOCHEMISTRY, 2017, 卷号: 56, 期号: 25, 页码: 3273-3282
作者:  Qin, Lingyun;  Zhou, Jingjing;  Su, Zhengding;  Liu, Huili;  Huang, Yongqi
收藏  |  浏览/下载:32/0  |  提交时间:2017/12/06


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