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Metabolism-based structure optimization: Discovery of a potent and orally available tyrosine kinase ALK inhibitor bearing the tetracyclic benzo[b]carbazolone core (vol 26, pg 5399, 2016)
Han, Mei4; Wang, Chengyan2; Ji, Yinchun1; Song, Zilan5; Xing, Li5; Su, Yi1; Wang, Xisheng2; Zhang, Ao3,5; Ai, Jing1,3,5; Geng, Meiyu1,3,5
刊名BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
2020-02-15
卷号30期号:4页码:1
ISSN号0960-894X
DOI10.1016/j.bmcl.2019.126931
通讯作者Zhang, Ao(aozhang@simm.ac.cn) ; Ai, Jing(jai@simm.ac.cn) ; Geng, Meiyu(mygeng@simm.ac.cn)
WOS研究方向Pharmacology & Pharmacy ; Chemistry
语种英语
出版者PERGAMON-ELSEVIER SCIENCE LTD
WOS记录号WOS:000507987200032
内容类型期刊论文
源URL[http://119.78.100.183/handle/2S10ELR8/282454]  
专题中国科学院上海药物研究所
通讯作者Zhang, Ao; Ai, Jing; Geng, Meiyu
作者单位1.Chinese Acad Sci, SIMM, Div Antitumor Pharmacol, State Key Lab Drug Res, Shanghai 201203, Peoples R China
2.Univ Sci & Technol China, Nano Sci & Technol Inst, Suzhou 215123, Peoples R China
3.Univ Chinese Acad Sci, Beijing 100049, Peoples R China
4.Ocean Univ China, Sch Med & Pharm, Dept Pharmacol & Glycobiol, Qingdao 266003, Peoples R China
5.Chinese Acad Sci, SIMM, CAS Key Lab Receptor Res, Shanghai 201203, Peoples R China
推荐引用方式
GB/T 7714
Han, Mei,Wang, Chengyan,Ji, Yinchun,et al. Metabolism-based structure optimization: Discovery of a potent and orally available tyrosine kinase ALK inhibitor bearing the tetracyclic benzo[b]carbazolone core (vol 26, pg 5399, 2016)[J]. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS,2020,30(4):1.
APA Han, Mei.,Wang, Chengyan.,Ji, Yinchun.,Song, Zilan.,Xing, Li.,...&Geng, Meiyu.(2020).Metabolism-based structure optimization: Discovery of a potent and orally available tyrosine kinase ALK inhibitor bearing the tetracyclic benzo[b]carbazolone core (vol 26, pg 5399, 2016).BIOORGANIC & MEDICINAL CHEMISTRY LETTERS,30(4),1.
MLA Han, Mei,et al."Metabolism-based structure optimization: Discovery of a potent and orally available tyrosine kinase ALK inhibitor bearing the tetracyclic benzo[b]carbazolone core (vol 26, pg 5399, 2016)".BIOORGANIC & MEDICINAL CHEMISTRY LETTERS 30.4(2020):1.
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