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科研机构
上海药物研究所 [51]
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期刊论文 [51]
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2021 [4]
2020 [3]
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Conformational polymorphs of isotretinoin and their impact on physicochemical and biological properties
期刊论文
INTERNATIONAL JOURNAL OF PHARMACEUTICS, 2021, 卷号: 610, 页码: 10
作者:
Cheng, Yinxiang
;
Rong, Xiaoyi
;
Xia, Mengyuan
;
Zhang, Zaiyong
;
Wang, Jian-Rong
收藏
  |  
浏览/下载:54/0
  |  
提交时间:2022/01/04
Polymorph
Isotretinoin
Stability
Solubility
Bioavailability
Solidification of volatile D-Limonene by cyclodextrin metal-organic framework for pulmonary delivery via dry powder inhalers: In vitro and in vivo evaluation
期刊论文
INTERNATIONAL JOURNAL OF PHARMACEUTICS, 2021, 卷号: 606, 页码: 9
作者:
Zhou, Yong
;
Zhang, Meijuan
;
Wang, Caifen
;
Ren, Xiaohong
;
Guo, Tao
收藏
  |  
浏览/下载:98/0
  |  
提交时间:2021/11/04
D-Limonene
gamma-cyclodextrin metal-organic framework
Dry powder inhaler
Solidification
Aerosolization
Bioavailability
Design, Synthesis, and Biological Evaluation of Orally Bioavailable CHK1 Inhibitors Active against Acute Myeloid Leukemia
期刊论文
CHEMMEDCHEM, 2021, 页码: 12
作者:
Jin, Tingting
;
Wang, Peipei
;
Long, Xiubing
;
Jiang, Kailong
;
Song, Pinrao
收藏
  |  
浏览/下载:133/0
  |  
提交时间:2021/05/24
CHK1 inhibitor
diaminopyrimidine
DNA damage response
oral bioavailability
Cocrystals to tune oily vitamin E into crystal vitamin E
期刊论文
INTERNATIONAL JOURNAL OF PHARMACEUTICS, 2021, 卷号: 592, 页码: 8
作者:
Zhu, Bingqing
;
Zhang, Qi
;
Lu, Liye
;
Bao, Junjie
;
Rong, Xiaoyi
收藏
  |  
浏览/下载:133/0
  |  
提交时间:2021/05/24
Cocrystal
Vitamin E
Solidification
Stability
Bioavailability
Biodistribution and immunomodulatory activities of a proteoglycan isolated from Ganoderma lucidum
期刊论文
JOURNAL OF FUNCTIONAL FOODS, 2020, 卷号: 74, 页码: 13
作者:
Teng, Yilong
;
Liang, Haohui
;
Zhang, Zeng
;
He, Yanming
;
Pan, Yanna
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  |  
浏览/下载:132/0
  |  
提交时间:2020/12/21
Proteoglycan
Ganoderma lucidum
Bioavailability
Macrophage
Immunoregulation
Enhanced oral bioavailability and bioefficacy of phloretin using mixed polymeric modified self-nanoemulsions
期刊论文
FOOD SCIENCE & NUTRITION, 2020, 页码: 14
作者:
Wang, Yiling
;
Li, Dongli
;
Lin, Huiqiong
;
Jiang, Sen
;
Han, Lei
收藏
  |  
浏览/下载:138/0
  |  
提交时间:2020/07/01
anti-inflammatory
bioavailability
pharmacokinetics
phloretin
self-nanoemulsions
solubility
Activation of a gamma-cyclodextrin-based metal-organic framework using supercritical carbon dioxide for high-efficient delivery of honokiol
期刊论文
CARBOHYDRATE POLYMERS, 2020, 卷号: 235, 页码: 10
作者:
He, Yuanzhi
;
Hou, Xuefeng
;
Guo, Jingwen
;
He, Zehui
;
Guo, Teng
收藏
  |  
浏览/下载:149/0
  |  
提交时间:2020/07/01
gamma-cyclodextrin metal-organic framework
Activation
Honokiol
Supercritical carbon dioxide
Bioavailability
MOF Capacitates Cyclodextrin to Mega-Load Mode for High-Efficient Delivery of Valsartan
期刊论文
PHARMACEUTICAL RESEARCH, 2019, 卷号: 36, 期号: 8, 页码: 13
作者:
Zhang, Wei
;
Guo, Tao
;
Wang, Caifen
;
He, Yuanzhi
;
Zhang, Xi
收藏
  |  
浏览/下载:123/0
  |  
提交时间:2020/07/01
Bioavailability
cyclodextrin
metal-organic framework
solubility
valsartan
Supersaturated polymeric micelles for oral silybin delivery: the role of the Soluplus-PVPVA complex
期刊论文
ACTA PHARMACEUTICA SINICA B, 2019, 卷号: 9, 期号: 1, 页码: 107-117
作者:
Zhu, Chunliu
;
Gong, Shuang
;
Ding, Jinsong
;
Yu, Miaorong
;
Ahmad, Ejaj
收藏
  |  
浏览/下载:130/0
  |  
提交时间:2020/07/01
Silybin
Soluplus
PVPVA
Complex
Supersaturated drug delivery system
Oral bioavailability
Drug nanoclusters formed in confined nano-cages of CD-MOF: dramatic enhancement of solubility and bioavailability of azilsartan
期刊论文
ACTA PHARMACEUTICA SINICA B, 2019, 卷号: 9, 期号: 1, 页码: 97-106
作者:
He, Yuanzhi
;
Zhang, Wei
;
Guo, Tao
;
Zhang, Guoqing
;
Qin, Wei
收藏
  |  
浏览/下载:104/0
  |  
提交时间:2020/07/01
gamma-Cyclodextrin metal organic framework
Nanoclusterization
Azilsartan
Mechanism
Solubility
Bioavailability
Molecular modeling
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