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Identification of 5-benzylidene-2-phenylthiazolones as potent PRMT5 inhibitors by virtual screening, structural optimization and biological evaluations 期刊论文
BIOORGANIC CHEMISTRY, 2018, 卷号: 81, 页码: 289-298
作者:  Zhu, Kongkai;  Tao, Hongrui;  Song, Jia-Li;  Jin, Lu;  Zhang, Yuanyuan
收藏  |  浏览/下载:129/0  |  提交时间:2019/01/08
Natural Breviscapin, Mangiferin, and a Modified Mangostin Present Inhibitory Effect on Dipeptidyl Peptidase-IV 期刊论文
CHEMISTRYSELECT, 2018, 卷号: 3, 期号: 39, 页码: 10864-10868
作者:  Hou, Bo;  Kuang, Meng-Ting;  Chi, Xiao-Qian;  Li, Jin-Yu;  Yang, Liu
收藏  |  浏览/下载:52/0  |  提交时间:2018/12/03
Pharmacophore modeling, molecular docking and molecular dynamics simulations toward identifying lead compounds for Chk1 期刊论文
COMPUTATIONAL BIOLOGY AND CHEMISTRY, 2018, 卷号: 76, 页码: 53-60
作者:  Li, Yaping;  Peng, Jiale;  Zhou, Yeheng;  Li, Penghua;  Li, Yingying
收藏  |  浏览/下载:29/0  |  提交时间:2018/11/12
Discovery of novel wee1 inhibitors via structure-based virtual screening and biological evaluation 期刊论文
JOURNAL OF COMPUTER-AIDED MOLECULAR DESIGN, 2018, 卷号: 32, 期号: 9, 页码: 901-915
作者:  Li, Yaping;  Pu, Yinglan;  Liu, Hui;  Zhang, Li;  Liu, Xingyong
收藏  |  浏览/下载:50/0  |  提交时间:2018/11/06
Identification of a novel selective small-molecule inhibitor of protein arginine methyltransferase 5 (PRMT5) by virtual screening, resynthesis and biological evaluations 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2018, 卷号: 28, 期号: 9, 页码: 1476-1483
作者:  Zhu, Kongkai;  Jiang, Chengshi;  Tao, Hongrui;  Liu, Jingqiu;  Zhang, Hua
收藏  |  浏览/下载:59/0  |  提交时间:2019/01/08
Computational chemical biology and drug design: Facilitating protein structure, function, and modulation studies 期刊论文
MEDICINAL RESEARCH REVIEWS, 2018, 卷号: 38, 期号: 3, 页码: 914-950
作者:  Zheng, Mingyue;  Zhao, Jihui;  Cui, Chen;  Fu, Zunyun;  Li, Xutong
收藏  |  浏览/下载:42/0  |  提交时间:2019/01/08
Discovery of Novel Inhibitors of Indoleamine 2,3-Dioxygenase 1 Through Structure-Based Virtual Screening 期刊论文
FRONTIERS IN PHARMACOLOGY, 2018, 卷号: 9
作者:  Zhang, Guoqing;  Xing, Jing;  Wang, Yulan;  Wang, Lihao;  Ye, Yan
收藏  |  浏览/下载:25/0  |  提交时间:2019/01/08
Computer-Aided Drug Design in Epigenetics 期刊论文
FRONTIERS IN CHEMISTRY, 2018, 卷号: 6
作者:  Lu, Wenchao;  Zhang, Rukang;  Jiang, Hao;  Zhang, Huimin;  Luo, Cheng
收藏  |  浏览/下载:26/0  |  提交时间:2019/01/08
Hit optimization studies of 3-hydroxy-indolin-2-one analogs as potential anti-HIV-1 agents 期刊论文
BIOORGANIC CHEMISTRY, 2018, 卷号: 79
作者:  Chander, Subhash;  Tang, Cheng-Run;  Penta, Ashok;  Wang, Ping;  Bhagwat, Deepak P.
收藏  |  浏览/下载:12/0  |  提交时间:2019/12/04
Structure-Based Virtual Screening, Compound Synthesis, and Bioassay for the Design of Chitinase Inhibitors 期刊论文
JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY, 2018, 卷号: 66, 页码: 3351-3357
作者:  Dong, Yawen;  Jiang, Xi;  Liu, Tian;  Ling, Yun;  Yang, Qing
收藏  |  浏览/下载:3/0  |  提交时间:2019/12/02


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