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4-Oxo-1,4-dihydroquinoline-3-carboxamide Derivatives as New Axl Kinase Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 14, 页码: 6807-6825
Tan, Li; Zhang, Zhang; Gao, Dongylin; Luo, Jinfeng; Tu, Zheng-Chao; Li, Zhengqiu; Peng, Lijie; Ren, Xiaomei; Ding, Ke
收藏  |  浏览/下载:23/0  |  提交时间:2016/12/16
Structure-Based Design of Tetrahydroisoquinoline-7-carboxamides as Selective Discoidin Domain Receptor 1 (DDR1) Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 12, 页码: 5911-5916
Wang, Zhen; Bian, Huan; Bartual, Sergio G.; Du, Wenting; Luo, Jinfeng; Zhao, Hu; Zhang, Shasha; Mo, Cheng; Zhou, Yang; Xu, Yong; Tu, Zhengchao; Ren, Xiaomei; Lu, Xiaoyun; Brekken, Rolf A.; Yao, Libo; Bullock, Alex N.; Su, Jin; Ding, Ke
收藏  |  浏览/下载:50/0  |  提交时间:2016/12/16
Structure-Based Design of Tetrahydroisoquinoline-7-carboxamides as Selective Discoidin Domain Receptor 1 (DDR1) Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 12, 页码: 5911-5916
作者:  Yao, Libo;  Ding, Ke;  Su, Jin;  Bullock, Alex N.;  Brekken, Rolf A.
收藏  |  浏览/下载:32/0  |  提交时间:2018/12/13
4-Oxo-1,4-dihydroquinoline-3-carboxamide Derivatives as New Axl Kinase Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 14, 页码: 6807-6825
作者:  Tan, Li;  Zhang, Zhang;  Gao, Dongylin;  Luo, Jinfeng;  Tu, Zheng-Chao
收藏  |  浏览/下载:17/0  |  提交时间:2018/12/13
Small-Molecule BET Inhibitors in Clinical and Preclinical Development and Their Therapeutic Potential 期刊论文
CURRENT TOPICS IN MEDICINAL CHEMISTRY, 2015, 卷号: 15, 期号: 8, 页码: 776-794
Yu, Lei; Wang, Zhen; Zhang, Zhang; Ren, Xiaomei; Lu, Xiaoyun; Ding, Ke
收藏  |  浏览/下载:25/0  |  提交时间:2016/12/16
2,4-Diarylamino-pyrimidines as kinase inhibitors co-targeting IGF1R and EGFR(L858R/T790M) 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2015, 卷号: 25, 期号: 19, 页码: 4277-4281
Chan, Shingpan; Han, Kun; Qu, Rong; Tong, Linjiang; Li, Yingjun; Zhang, Zhang; Cheng, Huimin; Lu, Xiaoyun; Patterson, Adam; Smaill, Jeff; Ren, Xiaomei; Ding, Jian; Xie, Hua; Ding, Ke
收藏  |  浏览/下载:246/0  |  提交时间:2016/12/16
Hybrid pyrimidine alkynyls inhibit the clinically resistance related Bcr-Abl(T315I) mutant 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2015, 卷号: 25, 期号: 17, 页码: 3458-3463
作者:  Ding, Ke;  Pan, Xiaofeng;  Wang, Deping;  Zhuang, Xiaoxi;  Luo, Jingfeng
收藏  |  浏览/下载:22/0  |  提交时间:2018/12/13
2,4-Diarylamino-pyrimidines as kinase inhibitors co-targeting IGF1R and EGFR(L858R/T790M) 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2015, 卷号: 25, 期号: 19, 页码: 4277-4281
作者:  Smaill, Jeff;  Lu, Xiaoyun;  Cheng, Huimin;  Zhang, Zhang;  Li, Yingjun
收藏  |  浏览/下载:48/0  |  提交时间:2018/12/13
Small-Molecule BET Inhibitors in Clinical and Preclinical Development and Their Therapeutic Potential 期刊论文
CURRENT TOPICS IN MEDICINAL CHEMISTRY, 2015, 卷号: 15, 期号: 8, 页码: 776-794
作者:  Wang, Zhen;  Zhang, Zhang;  Ren, Xiaomei;  Lu, Xiaoyun;  Ding, Ke
收藏  |  浏览/下载:10/0  |  提交时间:2018/12/13
N-(3-Ethynyl-2,4-difluorophenyl)sulfonamide Derivatives as Selective Raf Inhibitors 期刊论文
ACS MEDICINAL CHEMISTRY LETTERS, 2015, 卷号: 6, 期号: 5, 页码: 543-547
作者:  Ding, Ke;  Cheng, Huimin;  Zhang, Zhang;  Zhuang, Xiaoxi;  Li, Yingjun
收藏  |  浏览/下载:18/0  |  提交时间:2018/12/13


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