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科研机构
新疆理化技术研究所 [14]
内容类型
期刊论文 [14]
发表日期
2022 [3]
2021 [2]
2020 [1]
2019 [3]
2018 [3]
2017 [1]
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Chemistry [1]
Pharmacolo... [1]
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"One-Pot" Synthesis of Molnupiravir from Cytidine
期刊论文
ORGANIC PROCESS RESEARCH & DEVELOPMENT, 2022, 卷号: 26, 期号: 2, 页码: 358-364
作者:
Hu, TW (Hu, Tianwen) [1] , [2]
;
Xie, YC (Xie, Yuanchao) [3]
;
Zhu, FQ (Zhu, Fuqiang) [4]
;
Gong, XD (Gong, Xudong) [4]
;
Liu, Y (Liu, Yin) [2] , [3]
收藏
  |  
浏览/下载:124/0
  |  
提交时间:2022/03/23
molnupiravir
cytidine
one-pot synthesis
DMF-DMA
Design, synthesis, in vitro evaluation of a new pyrrolo[1,2-a]thiazolo[5,4-d]pyrimidinone derivatives as cholinesterase inhibitors against Alzheimer's disease
期刊论文
JOURNAL OF HETEROCYCLIC CHEMISTRY, 2022, 卷号: 59, 期号: 6, 页码: 1086-1101
作者:
Zeng, Y (Zeng, Yan) [1] , [2]
;
Nie, LF (Nie, Lifei) [1]
;
Liu, L (Liu, Liu) [1]
;
Niu, C (Niu, Chao) [1] , [2]
;
Li, Y (Li, Yi) [1] , [2]
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2022/06/21
A novel synthesis of tetrahydrocortisone 3-glucuronide
期刊论文
JOURNAL OF CARBOHYDRATE CHEMISTRY, 2022, 卷号: 41, 期号: 1, 页码: 18-27
作者:
Zhang, Y (Zhang, Yan) [1] , [2] , [3]
;
Zhang, SQ (Zhang, Suqing) [4]
;
Li, R (Li, Rui) [5]
;
Shen, JS (Shen, Jingshan) [3] , [4]
;
Jiang, XR (Jiang, Xiangrui) [3] , [4]
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2022/04/07
Cortisone acetate
Koenig-Knorr glycosylation
lithium tri-tert-butoxyaluminum hydride
tetrahydrocortisone 3-glucuronide
Weinreb Amide Approach to the Practical Synthesis of a Key Remdesivir Intermediate
期刊论文
The Journal of organic chemistry, 2021, 卷号: 86, 期号: 7, 页码: 5065-5072
作者:
Xie, Yuanchao
;
Hu, Tianwen
;
Zhang, Yan
;
Wei, Daibao
;
Zheng, Wei
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2021/05/06
Potency and pharmacokinetics of GS-441524 derivatives against SARS-CoV-2
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2021, 卷号: 46, 期号: 9, 页码: 1-12
作者:
Wei, DB (Wei, Daibao)
;
Hu, TW (Hu, Tianwen)
;
Zhang, YM (Zhang, Yumin)
;
Zheng, W (Zheng, Wei)
;
Xue, HT (Xue, Haitao)
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2021/10/14
Covid-19
SARS-CoV-2
GS-441524
Antiviral
Nucleoside
Prodrug
Isobutyrate
Synthesis of CBD and Its Derivatives Bearing Various C4 '-Side Chains with a Late-Stage Diversification Method
期刊论文
JOURNAL OF ORGANIC CHEMISTRY, 2020, 卷号: 85, 期号: 4, 页码: 2704-2715
作者:
Gong, XD (Gong, Xudong)[ 2,3 ]
;
Sun, CL (Sun, Changliang)[ 4 ]
;
Abame, MA (Abame, Melkamu Alemu)[ 1 ]
;
Shi, WQ (Shi, Wenqiang)[ 1 ]
;
Xie, YC (Xie, Yuanchao)[ 1 ]
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2020/04/16
Pharmacokinetics-Driven Optimization of 4(3H)-Pyrimidinones as Phosphodiesterase Type 5 Inhibitors Leading to TPN171, a Clinical Candidate for the Treatment of Pulmonary Arterial Hypertension
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 10, 页码: 4979-4990
作者:
Wang, Z (Wang, Zhen)[ 1 ]
;
Jiang, XR (Jiang, Xiangrui)[ 1 ]
;
Zhang, XL (Zhang, Xianglei)[ 1,2 ]
;
Tian, GH (Tian, Guanghui)[ 3 ]
;
Yang, RL (Yang, Rulei)[ 3 ]
收藏
  |  
浏览/下载:137/0
  |  
提交时间:2019/06/28
Biological Activities of Artemisinin Derivatives Beyond Malaria
期刊论文
CURRENT TOPICS IN MEDICINAL CHEMISTRY, 2019, 卷号: 19, 期号: 3, 页码: 205-222
作者:
Liu, XY (Liu, Xiaoyan)[ 1,2 ]
;
Cao, JG (Cao, Jianguo)[ 2 ]
;
Huang, GZ (Huang, Guozheng)[ 2,3 ]
;
Zhao, QJ (Zhao, Qingjie)[ 1 ]
;
Shen, JS (Shen, Jingshan)[ 1 ]
收藏
  |  
浏览/下载:60/0
  |  
提交时间:2019/05/16
Anticancer activity
Antiviral activity
Artemisinin
Artemisinin derivatives
Dimer
Trimer
Industry-Oriented Route Evaluation and Process Optimization for the Preparation of Brexpiprazole
期刊论文
ORGANIC PROCESS RESEARCH & DEVELOPMENT, 2019, 卷号: 23, 期号: 5, 页码: 852-857
作者:
Chen, WM (Chen, Weiming)[ 1,2 ]
;
Suo, J (Suo, Jin)[ 3 ]
;
Liu, YJ (Liu, Yongjian)[ 4 ]
;
Xie, YC (Xie, Yuanchao)[ 3 ]
;
Wu, MJ (Wu, Mingjun)[ 4 ]
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2020/04/03
brexpiprazole
route evaluation
process optimization
impurity control strategy
A Facile Epoxide Aminolysis Promoted by (t-BuO)(2)Mg and Its Application to the Synthesis of Efinaconazole
期刊论文
ORGANIC PROCESS RESEARCH & DEVELOPMENT, 2018, 卷号: 22, 期号: 5, 页码: 625-632
作者:
Zhu, FQ (Zhu, Fuqiang)
;
Xie, YC (Xie, Yuanchao)
;
Zhang, J (Zhang, Jian)
;
Tian, GH (Tian, Guanghui)
;
Qin, HJ (Qin, Hongjian)
收藏
  |  
浏览/下载:58/0
  |  
提交时间:2018/06/20
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