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"One-Pot" Synthesis of Molnupiravir from Cytidine 期刊论文
ORGANIC PROCESS RESEARCH & DEVELOPMENT, 2022, 卷号: 26, 期号: 2, 页码: 358-364
作者:  Hu, TW (Hu, Tianwen) [1] , [2];  Xie, YC (Xie, Yuanchao) [3];  Zhu, FQ (Zhu, Fuqiang) [4];  Gong, XD (Gong, Xudong) [4];  Liu, Y (Liu, Yin) [2] , [3]
收藏  |  浏览/下载:124/0  |  提交时间:2022/03/23
Design, synthesis, in vitro evaluation of a new pyrrolo[1,2-a]thiazolo[5,4-d]pyrimidinone derivatives as cholinesterase inhibitors against Alzheimer's disease 期刊论文
JOURNAL OF HETEROCYCLIC CHEMISTRY, 2022, 卷号: 59, 期号: 6, 页码: 1086-1101
作者:  Zeng, Y (Zeng, Yan) [1] , [2];  Nie, LF (Nie, Lifei) [1];  Liu, L (Liu, Liu) [1];  Niu, C (Niu, Chao) [1] , [2];  Li, Y (Li, Yi) [1] , [2]
收藏  |  浏览/下载:20/0  |  提交时间:2022/06/21
A novel synthesis of tetrahydrocortisone 3-glucuronide 期刊论文
JOURNAL OF CARBOHYDRATE CHEMISTRY, 2022, 卷号: 41, 期号: 1, 页码: 18-27
作者:  Zhang, Y (Zhang, Yan) [1] , [2] , [3];  Zhang, SQ (Zhang, Suqing) [4];  Li, R (Li, Rui) [5];  Shen, JS (Shen, Jingshan) [3] , [4];  Jiang, XR (Jiang, Xiangrui) [3] , [4]
收藏  |  浏览/下载:22/0  |  提交时间:2022/04/07
Weinreb Amide Approach to the Practical Synthesis of a Key Remdesivir Intermediate 期刊论文
The Journal of organic chemistry, 2021, 卷号: 86, 期号: 7, 页码: 5065-5072
作者:  Xie, Yuanchao;  Hu, Tianwen;  Zhang, Yan;  Wei, Daibao;  Zheng, Wei
收藏  |  浏览/下载:31/0  |  提交时间:2021/05/06
Potency and pharmacokinetics of GS-441524 derivatives against SARS-CoV-2 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2021, 卷号: 46, 期号: 9, 页码: 1-12
作者:  Wei, DB (Wei, Daibao);  Hu, TW (Hu, Tianwen);  Zhang, YM (Zhang, Yumin);  Zheng, W (Zheng, Wei);  Xue, HT (Xue, Haitao)
收藏  |  浏览/下载:28/0  |  提交时间:2021/10/14
Synthesis of CBD and Its Derivatives Bearing Various C4 '-Side Chains with a Late-Stage Diversification Method 期刊论文
JOURNAL OF ORGANIC CHEMISTRY, 2020, 卷号: 85, 期号: 4, 页码: 2704-2715
作者:  Gong, XD (Gong, Xudong)[ 2,3 ];  Sun, CL (Sun, Changliang)[ 4 ];  Abame, MA (Abame, Melkamu Alemu)[ 1 ];  Shi, WQ (Shi, Wenqiang)[ 1 ];  Xie, YC (Xie, Yuanchao)[ 1 ]
收藏  |  浏览/下载:31/0  |  提交时间:2020/04/16
Pharmacokinetics-Driven Optimization of 4(3H)-Pyrimidinones as Phosphodiesterase Type 5 Inhibitors Leading to TPN171, a Clinical Candidate for the Treatment of Pulmonary Arterial Hypertension 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 10, 页码: 4979-4990
作者:  Wang, Z (Wang, Zhen)[ 1 ];  Jiang, XR (Jiang, Xiangrui)[ 1 ];  Zhang, XL (Zhang, Xianglei)[ 1,2 ];  Tian, GH (Tian, Guanghui)[ 3 ];  Yang, RL (Yang, Rulei)[ 3 ]
收藏  |  浏览/下载:137/0  |  提交时间:2019/06/28
Biological Activities of Artemisinin Derivatives Beyond Malaria 期刊论文
CURRENT TOPICS IN MEDICINAL CHEMISTRY, 2019, 卷号: 19, 期号: 3, 页码: 205-222
作者:  Liu, XY (Liu, Xiaoyan)[ 1,2 ];  Cao, JG (Cao, Jianguo)[ 2 ];  Huang, GZ (Huang, Guozheng)[ 2,3 ];  Zhao, QJ (Zhao, Qingjie)[ 1 ];  Shen, JS (Shen, Jingshan)[ 1 ]
收藏  |  浏览/下载:60/0  |  提交时间:2019/05/16
Industry-Oriented Route Evaluation and Process Optimization for the Preparation of Brexpiprazole 期刊论文
ORGANIC PROCESS RESEARCH & DEVELOPMENT, 2019, 卷号: 23, 期号: 5, 页码: 852-857
作者:  Chen, WM (Chen, Weiming)[ 1,2 ];  Suo, J (Suo, Jin)[ 3 ];  Liu, YJ (Liu, Yongjian)[ 4 ];  Xie, YC (Xie, Yuanchao)[ 3 ];  Wu, MJ (Wu, Mingjun)[ 4 ]
收藏  |  浏览/下载:29/0  |  提交时间:2020/04/03
A Facile Epoxide Aminolysis Promoted by (t-BuO)(2)Mg and Its Application to the Synthesis of Efinaconazole 期刊论文
ORGANIC PROCESS RESEARCH & DEVELOPMENT, 2018, 卷号: 22, 期号: 5, 页码: 625-632
作者:  Zhu, FQ (Zhu, Fuqiang);  Xie, YC (Xie, Yuanchao);  Zhang, J (Zhang, Jian);  Tian, GH (Tian, Guanghui);  Qin, HJ (Qin, Hongjian)
收藏  |  浏览/下载:58/0  |  提交时间:2018/06/20


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