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Remodeling Tumor-Associated Macrophages and Neovascularization Overcomes EGFR(T790M)-Associated Drug Resistance by PD-L1 Nanobody-Mediated Codelivery 期刊论文
SMALL, 2018, 卷号: 14, 期号: 47
作者:  Yin, Weimin;  Yu, Xiaolu;  Kang, Xuejia;  Zhao, Yuge;  Zhao, Pengfei
收藏  |  浏览/下载:100/0  |  提交时间:2019/01/08
Identification of compound D2923 as a novel anti-tumor agent targeting CSF1R 期刊论文
ACTA PHARMACOLOGICA SINICA, 2018, 卷号: 39, 期号: 11, 页码: 1768-1776
作者:  Liu, Ying-Qiang;  Wang, Ya-Nan;  Lu, Xiao-Yun;  Tong, Lin-Jiang;  Li, Yan
收藏  |  浏览/下载:110/0  |  提交时间:2019/01/08
Discovery of Potent Irreversible Pan-Fibroblast Growth Factor Receptor (FGFR) Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 61, 期号: 20, 页码: 9085-9104
作者:  Wang, Yuming;  Li, Lijun;  Fan, Jun;  Dai, Yang;  Jiang, Alan
收藏  |  浏览/下载:29/0  |  提交时间:2019/01/08
The receptor tyrosine kinase HIR-1 coordinates HIF-independent responses to hypoxia and extracellular matrix injury 期刊论文
SCIENCE SIGNALING, 2018, 卷号: 11, 期号: 550, 页码: 12
作者:  Vozdek, Roman;  Long, Yong;  Ma, Dengke K.
收藏  |  浏览/下载:25/0  |  提交时间:2019/07/02
Backbone and side-chain chemical shift assignments of the kringle domain of human receptor tyrosine kinase-like orphan receptor 1 (ROR1) (vol 12, pg 145, 2018) 期刊论文
BIOMOLECULAR NMR ASSIGNMENTS, 2018, 卷号: 12, 期号: 2, 页码: 363-363
作者:  Ma, Xiaofang;  Zhang, Yingying;  Liu, Bin;  Yang, Jiahui;  Hu, Kaifeng
收藏  |  浏览/下载:30/0  |  提交时间:2018/10/07
Arsenic circumvents the gefitinib resistance by binding to P62 and mediating autophagic degradation of EGFR in non-small cell lung cancer 期刊论文
CELL DEATH & DISEASE, 2018, 卷号: 9
作者:  Mao, Jianhua;  Ma, Lie;  Shen, Yan;  Zhu, Kongkai;  Zhang, Ru
收藏  |  浏览/下载:49/0  |  提交时间:2019/01/08
Stable Cocrystals and Salts of the Antineoplastic Drug Apatinib with Improved Solubility in Aqueous Solution 期刊论文
CRYSTAL GROWTH & DESIGN, 2018, 卷号: 18, 期号: 8, 页码: 4701-4714
作者:  Zhu, Bin;  Wang, Jian-Rong;  Zhang, Qi;  Li, Meiqi;  Guo, Chunyang
收藏  |  浏览/下载:70/0  |  提交时间:2019/01/08
Current Strategies and Applications for Precision Drug Design 期刊论文
FRONTIERS IN PHARMACOLOGY, 2018, 卷号: 9
作者:  Wang, Chen;  Xu, Pan;  Zhang, Luyu;  Huang, Jing;  Zhu, Kongkai
收藏  |  浏览/下载:47/0  |  提交时间:2019/01/08
Design, Synthesis, and Biological Evaluation of Pyrimido[4,5-d]pyrimidine-2,4(1H,3H)-diones as Potent and Selective Epidermal Growth Factor Receptor (EGFR) Inhibitors against L858R/T790M Resistance Mutation 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 61, 期号: 13, 页码: 5609-5622
作者:  Hao, Yongjia;  Lyu, Jiankun;  Qu, Rong;  Tong, Yi;  Sun, Deheng
收藏  |  浏览/下载:61/0  |  提交时间:2019/01/08
Design, synthesis and biological evaluation of a series of novel 2-benzamide-4-(6-oxy-N-methyl-l-naphthamide)-pyridine derivatives as potent fibroblast growth factor receptor (FGFR) inhibitors 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 154, 页码: 9-28
作者:  Wei, Manman;  Peng, Xia;  Xing, Li;  Dai, Yang;  Huang, Ruimin
收藏  |  浏览/下载:63/0  |  提交时间:2019/01/08


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