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科研机构
北京大学 [39]
内容类型
期刊论文 [38]
其他 [1]
发表日期
2017 [3]
2016 [5]
2015 [2]
2014 [4]
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2012 [5]
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专题:北京大学
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Cryo-EM structures of the 80S ribosomes from human parasites Trichomonas vaginalis and Toxoplasma gondii
期刊论文
CELL RESEARCH, 2017
Li, Zhifei
;
Guo, Qiang
;
Zheng, Lvqin
;
Ji, Yongsheng
;
Xie, Yi-Ting
;
Lai, De-Hua
;
Lun, Zhao-Rong
;
Suo, Xun
;
Gao, Ning
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2017/12/03
cryo-electron microscopy
ribosome
translation
Trichomonas vaginalis
Toxoplasma gondii
RNA
TRANSLATION INITIATION COMPLEX
PEPTIDYL-TRANSFERASE CENTER
NEIGHBOR-JOINING METHOD
N-TERMINAL EXTENSION
EUKARYOTIC RIBOSOME
MITOCHONDRIAL RIBOSOME
70S RIBOSOME
ANGSTROM RESOLUTION
ELECTRON-MICROSCOPY
PROTEIN-SYNTHESIS
Antiamyloidogenic Activity of A beta 42-Binding Peptoid in Modulating Amyloid Oligomerization
期刊论文
SMALL, 2017
Zhao, Zijian
;
Zhu, Ling
;
Li, Haiyun
;
Cheng, Peng
;
Peng, Jiaxi
;
Yin, Yudan
;
Yang, Yang
;
Wang, Chen
;
Hu, Zhiyuan
;
Yang, Yanlian
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2017/12/04
aggregation,amyloid oligomerization,antiamyloidogenic,inhibitor,peptoids
GAMMA-SECRETASE INHIBITORS
SMALL-MOLECULE INHIBITORS
ALZHEIMERS-DISEASE
BETA-PEPTIDE
FIBRIL FORMATION
PROTEIN AGGREGATION
MOUSE MODEL
MECHANISM
NEUROTOXICITY
CONFORMATION
Rational Design of Selective Allosteric Inhibitors of PHGDH and Serine Synthesis with Anti-tumor Activity
期刊论文
CELL CHEMICAL BIOLOGY, 2017
Wang, Qian
;
Liberti, Maria V.
;
Liu, Pei
;
Deng, Xiaobing
;
Liu, Ying
;
Locasale, Jason W.
;
Lai, Luhua
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2017/12/03
PHOSPHOGLYCERATE DEHYDROGENASE
CANCER METABOLISM
SYNTHESIS PATHWAY
ACCURATE DOCKING
BINDING-SITES
DRUG DESIGN
BIOSYNTHESIS
DISCOVERY
CELLS
COMBINATION
A Hybrid Chalcone Combining the Trimethoxyphenyl and Isatinyl Groups Targets Multiple Oncogenic Proteins and Pathways in Hepatocellular Carcinoma Cells
期刊论文
PLOS ONE, 2016
Cao, Lili
;
Zhang, Lijun
;
Zhao, Xiang
;
Zhang, Ye
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2017/12/04
CANCER-CELLS
TUBULIN POLYMERIZATION
BIOLOGICAL EVALUATION
MUTATIONAL LANDSCAPE
MOLECULAR THERAPIES
ANTITUBULIN AGENTS
IN-VIVO
NUCLEOLIN
KINASE
IDENTIFICATION
The cap-binding site of influenza virus protein PB2 as a drug target
期刊论文
ACTA CRYSTALLOGRAPHICA SECTION D-STRUCTURAL BIOLOGY, 2016
Severin, Chelsea
;
de Moura, Tales Rocha
;
Liu, Yong
;
Li, Keqin
;
Zheng, Xiaofeng
;
Luo, Ming
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2017/12/03
antiviral
inhibitor
drug design
broad spectrum
SUBUNIT
DOMAIN
1ST-IN-CLASS
INHIBITOR
MECHANISM
REVEALS
VX-787
De novo design of helical peptides to inhibit tumor necrosis factor-alpha by disrupting its trimer formation
期刊论文
MEDCHEMCOMM, 2016
Shen, Qi
;
Zhang, Changsheng
;
Liu, Hongbo
;
Liu, Yuting
;
Cao, Junyue
;
Zhang, Xiaolin
;
Liang, Yuan
;
Zhao, Meiping
;
Lai, Luhua
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2017/12/03
SMALL-MOLECULE INHIBITORS
TNF-ALPHA
FACTOR ANTAGONISTS
BINDING
OLIGOMERIZATION
SUPERFAMILY
RECEPTORS
DISCOVERY
DOMAIN
Chiral Sulfoxide-Induced Single Turn Peptide alpha-Helicity
期刊论文
SCIENTIFIC REPORTS, 2016
Zhang, Qingzhou
;
Jiang, Fan
;
Zhao, Bingchuan
;
Lin, Huacan
;
Tian, Yuan
;
Xie, Mingsheng
;
Bai, Guoyun
;
Gilbert, Adam M.
;
Goetz, Gilles H.
;
Liras, Spiros
;
Mathiowetz, Alan A.
;
Price, David A.
;
Song, Kun
;
Tu, Meihua
;
Wu, Yujie
;
Wang, Tao
;
Flanagan, Mark E.
;
Wu, Yun-Dong
;
Li, Zigang
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2017/12/03
PROTEIN-PROTEIN INTERACTIONS
SMALL-MOLECULE INHIBITORS
RING-CLOSING METATHESIS
STAPLED PEPTIDES
DRUG DISCOVERY
STABILIZATION
HELIX
MODEL
WATER
NUCLEATION
Natural Product Kongensin A is a Non-Canonical HSP90 Inhibitor that Blocks RIP3-dependent Necroptosis
期刊论文
Cell Chemical Biology, 2016
Li, Dianrong
;
Li, Chao
;
Li, Lin
;
Chen, She
;
Wang, Lei
;
Li, Qiang
;
Wang, Xiaodong
;
Lei, Xiaoguang
;
Shen, Zhirong
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2017/12/04
MIXED LINEAGE KINASE
DOMAIN-LIKE PROTEIN
CELL-DEATH
PROGRAMMED NECROSIS
BIOORTHOGONAL LIGATION
MOLECULAR CHAPERONE
RIP3
CANCER
MLKL
COMPLEX
Small-Molecule-Driven Direct Reprogramming of Mouse Fibroblasts into Functional Neurons
期刊论文
CELL STEM CELL, 2015
Li, Xiang
;
Zuo, Xiaohan
;
Jing, Junzhan
;
Ma, Yantao
;
Wang, Jiaming
;
Liu, Defang
;
Zhu, Jialiang
;
Du, Xiaomin
;
Xiong, Liang
;
Du, Yuanyuan
;
Xu, Jun
;
Xiao, Xiong
;
Wang, Jinlin
;
Chai, Zhen
;
Zhao, Yang
;
Deng, Hongkui
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2017/12/03
DOPAMINERGIC-NEURONS
CELL FATE
CONVERSION
PLURIPOTENCY
IDENTIFICATION
EXPRESSION
GENERATION
INHIBITORS
GENES
Ainsliadimer A selectively inhibits IKK alpha/beta by covalently binding a conserved cysteine
期刊论文
NATURE COMMUNICATIONS, 2015
Dong, Ting
;
Li, Chao
;
Wang, Xing
;
Dian, Longyang
;
Zhang, Xiuguo
;
Li, Lin
;
Chen, She
;
Cao, Ran
;
Li, Li
;
Huang, Niu
;
He, Sudan
;
Lei, Xiaoguang
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2017/12/03
NF-KAPPA-B
BIOMIMETIC SYNTHESES
ALLOSTERIC SITE
CANCER-THERAPY
BCL-X
ACTIVATION
PHOSPHORYLATION
INFLAMMATION
KINASE
UBIQUITINATION
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