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科研机构
上海药物研究所 [27]
内容类型
期刊论文 [27]
发表日期
2020 [2]
2018 [5]
2017 [7]
2016 [4]
2015 [1]
2014 [4]
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Anti-proliferative cassane-type diterpenoids from the seeds of Caesalpinia minax
期刊论文
NATURAL PRODUCT RESEARCH, 2020, 页码: 10
作者:
Xu, Yunshao
;
Shi, Wei
;
Feng, Lu
;
Cao, Jun
;
Feng, Zheling
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2021/05/24
Caesalpinia minax
Fabaceae
cassane diterpenoids
cytotoxic activity
An antibody-drug conjugate targeting a GSTA glycosite-signature epitope of MUC1 expressed by non-small cell lung cancer
期刊论文
CANCER MEDICINE, 2020, 页码: 12
作者:
Pan, Deng
;
Tang, Yubo
;
Tong, Jiao
;
Xie, Chengmei
;
Chen, Jiaxi
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2020/12/24
A novel tumor-targeting treatment strategy uses energy restriction via co-delivery of albendazole and nanosilver
期刊论文
NANO RESEARCH, 2018, 卷号: 11, 期号: 9, 页码: 4507-4523
作者:
Liang, Jianming
;
Li, Ruixiang
;
He, Yuwei
;
Ling, Chengli
;
Wang, Qi
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2019/01/08
albendazole
nano silver
co-delivery
tumor targeting
energy metabolism
Current Strategies and Applications for Precision Drug Design
期刊论文
FRONTIERS IN PHARMACOLOGY, 2018, 卷号: 9
作者:
Wang, Chen
;
Xu, Pan
;
Zhang, Luyu
;
Huang, Jing
;
Zhu, Kongkai
收藏
  |  
浏览/下载:47/0
  |  
提交时间:2019/01/08
precision medicine
precision drug design
computational modeling
deep learning
antibody-drug conjugates
ligand-targeted conjugates
Self-assembly of Fluorescent Dehydroberberine Enhances Mitochondria-Dependent Antitumor Efficacy
期刊论文
CHEMISTRY-A EUROPEAN JOURNAL, 2018, 卷号: 24, 期号: 39, 页码: 9812-9819
作者:
An, Ruibing
;
Gu, Zhanni
;
Sun, Haifeng
;
Hu, Yuxuan
;
Yan, Runqi
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2019/01/08
antitumor
cell imaging
dehydroberberine
mitochondria
self-assembly
Epitopes of MUC1 Tandem Repeats in Cancer as Revealed by Antibody Crystallography: Toward Glycopeptide Signature-Guided Therapy
期刊论文
MOLECULES, 2018, 卷号: 23, 期号: 6
作者:
Zhou, Dapeng
;
Xu, Lan
;
Huang, Wei
;
Tonn, Torsten
收藏
  |  
浏览/下载:68/0
  |  
提交时间:2019/01/08
MUC1
tandem repeat
antibodies
glycopeptide
co-crystal
Identification and Characterizations of Novel, Selective Histone Methyltransferase SET7 Inhibitors by Scaffold Hopping- and 2D-Molecular Fingerprint-Based Similarity Search
期刊论文
MOLECULES, 2018, 卷号: 23, 期号: 3
作者:
Ding, Hong
;
Lu, Wen Chao
;
Hu, Jun Chi
;
Liu, Yu-Chih
;
Zhang, Chen Hua
收藏
  |  
浏览/下载:50/0
  |  
提交时间:2019/01/08
SET7
inhibitor
similarity search
ligand-based drug design
chemical biology probe
Dihydroartemisinin selectively inhibits PDGFR alpha-positive ovarian cancer growth and metastasis through inducing degradation of PDGFR alpha protein
期刊论文
CELL DISCOVERY, 2017, 卷号: 3
作者:
Li, Xiaoguang
;
Ba, Qian
;
Liu, Yanling
;
Yue, Qingxi
;
Chen, Peizhan
收藏
  |  
浏览/下载:43/0
  |  
提交时间:2019/01/08
Dihydroartemisinin
Epithelial-mesenchymal transition
metastasis
ovarian cancer
PDGFR alpha
Discovery of potent 2,4-difluoro-linker poly(ADP-ribose) polymerase 1 inhibitors with enhanced water solubility and in vivo anticancer efficacy
期刊论文
ACTA PHARMACOLOGICA SINICA, 2017, 卷号: 38, 期号: 11, 页码: 1521-1532
作者:
Chen, Wen-hua
;
Song, Shan-shan
;
Qi, Ming-hui
;
Huan, Xia-juan
;
Wang, Ying-qing
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2019/01/08
PARP-1 inhibitor
olaparib
breast cancer
BRCA-deficient tumors
Discovery, mechanism and metabolism studies of 2,3-difluorophenyl-linker-containing PARP1 inhibitors with enhanced in vivo efficacy for cancer therapy
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 138, 页码: 514-531
作者:
Chen, Wenhua
;
Guo, Ne
;
Qi, Minghui
;
Dai, Haiying
;
Hong, Minghuang
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2019/01/08
Antitumor drug
BRCA1/2
PARP inhibitors
Molecular docking
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