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Natural Product Albiziabioside A Conjugated with Pyruvate Dehydrogenase Kinase Inhibitor Dichloroacetate To Induce Apoptosis-Ferroptosis-M2-TAMs Polarization for Combined Cancer Therapy
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 19, 页码: 8760-8772
作者:
Wei, Gaofei
;
Sung, Jiahong
;
Luan, Weijing
;
Hou, Zhuang
;
Wang, Shuai
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2020/07/01
Dichloroacetate Ameliorates Cardiac Dysfunction Caused by Ischemic Insults Through AMPK Signal PathwayNot Only Shifts Metabolism
期刊论文
TOXICOLOGICAL SCIENCES, 2019, 卷号: 167, 期号: 2
作者:
Quan, Nanhu
;
Li, Xuan
;
Liu, Jia
;
Hu, Haiyan
;
Lu, Shaoxin
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2019/12/05
ischemia-reperfusion
dichloroacetate
AMP-activated protein kinase
metabolism
Sodium Dichloroacetate Stimulates Angiogenesis by Improving Endothelial Precursor Cell Function in an AKT/GSK-3 beta/Nrf2 Dependent Pathway in Vascular Dementia Rats
期刊论文
FRONTIERS IN PHARMACOLOGY, 2019, 卷号: 10
作者:
Zhao, Hui
;
Mao, Junqin
;
Yuan, Yuan
;
Feng, Jingjing
;
Cheng, Hao
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2019/12/06
sodium dichloroacetate
endothelial progenitor cells
reactive oxygen species
angiogenesis
vascular dementia
Synthesis, Characterization, and Antifungal Property of Hydroxypropyltrimethyl Ammonium Chitosan Halogenated Acetates
期刊论文
MARINE DRUGS, 2018, 卷号: 16, 期号: 9, 页码: 315
作者:
Mi, Yingqi
;
Tan, Wenqiang
;
Zhang, Jingjing
;
Wei, Lijie
;
Chen, Yuan
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2020/07/08
hydroxypropyltrimethyl ammonium chloride chitosan
halogenated acetate
antifungal activity
electronegativity
Synthesis of Quaternary Ammonium Salts of Chitosan Bearing Halogenated Acetate for Antifungal and Antibacterial Activities
期刊论文
POLYMERS, 2018, 卷号: 10, 期号: 5, 页码: 530
作者:
Zhang, Jingjing
;
Tan, Wenqiang
;
Luan, Fang
;
Yin, Xiuli
;
Dong, Fang
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2020/07/08
quaternary ammonium salts of chitosan
halogenated acetate
characterization
antifungal activity
antibacterial activity
Activation of Pyruvate Dehydrogenase by Sodium Dichloroacetate Shifts Metabolic Consumption from Amino Acids to Glucose in IPEC-J2 Cells and Intestinal Bacteria in Pigs
期刊论文
Journal of Agricultural and Food Chemistry, 2018, 卷号: 66, 期号: 15, 页码: 3793-3800
作者:
An, Rui
;
Tang, Zhiru
;
Li, Yunxia
;
Li, Tiejun
;
Xu, Qingqing
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2019/12/27
-glutamate
glucose
oxidative metabolism
pyruvate dehydrogenase
sodium dichloroacetate
Development of the First Generation of Disulfide-Based Subtype Selective and Potent Covalent Pyruvate Dehydrogenase Kinase 1 (PDK1) Inhibitors
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 6, 页码: 2227-2244
作者:
Liu, Yifu
;
Xie, Zuoquan
;
Zhao, Dan
;
Zhu, Jin
;
Mao, Fei
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2019/01/08
Synthesis, NMR and computational studies on tautomerism of dichloroacetate of hydroxyanthraquinone
期刊论文
JOURNAL OF MOLECULAR STRUCTURE, 2017, 卷号: 1141, 页码: 462-468
作者:
Zhu, Li
;
Wang, Wenfeng
;
Miao, Junwei
;
Yin, Xu
;
Hu, Xiufang
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2019/11/21
Nucleophilicity
Tautomerism
NMR
Computation
Hydroxyanthraquinone
2-Methoxyestradiol enhances radiosensitivity in radioresistant melanoma MDA-MB-435R cells by regulating glycolysis via HIF-1 alpha/PDK1 axis
期刊论文
INTERNATIONAL JOURNAL OF ONCOLOGY, 2017, 卷号: 50, 期号: 5
作者:
Zhao, Hong
;
Jiang, Huangang
;
Li, Zheng
;
Zhuang, Yafei
;
Liu, Yinyin
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2019/12/05
melanoma
HIF-1 alpha
glycolysis
radiosensitivity
2-MeOE2
dichloroacetate
metabolism
Synthesis, characterization, and antifungal property of chitosan ammonium salts with halogens
期刊论文
INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES, 2016, 卷号: 92, 页码: 293-298
作者:
Tan, WQ
;
Li, Q
;
Dong, F
;
Wei, LJ
;
Guo, ZY
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2016/12/18
Chitosan ammonium salts
Antifungal activity
Group electronegativity
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