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Constitutive signal bias mediated by the human GHRHR splice variant 1 期刊论文
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2021, 卷号: 118, 期号: 40, 页码: 10
作者:  Cong, Zhaotong
收藏  |  浏览/下载:24/0  |  提交时间:2021/12/01
Insights into agonist-elicited activation of the human glucose-dependent insulinotropic polypeptide receptor 期刊论文
BIOCHEMICAL PHARMACOLOGY, 2021, 卷号: 192, 页码: 16
作者:  Yuliantie, Elita;  van der Velden, Wijnand J. C.;  Labroska, Viktorija;  Dai, Antao;  Zhao, Fenghui
收藏  |  浏览/下载:43/0  |  提交时间:2021/11/04
Signaling profiles in HEK 293T cells co-expressing GLP-1 and GIP receptors 期刊论文
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 8
作者:  Wang, Yu-zhe;  Yang, De-hua;  Wang, Ming-wei
收藏  |  浏览/下载:19/0  |  提交时间:2021/11/04
Activation pathway of a G protein-coupled receptor uncovers conformational intermediates as targets for allosteric drug design 期刊论文
NATURE COMMUNICATIONS, 2021, 卷号: 12, 期号: 1, 页码: 15
作者:  Lu, Shaoyong;  He, Xinheng;  Yang, Zhao;  Chai, Zongtao;  Zhou, Shuhua
收藏  |  浏览/下载:34/0  |  提交时间:2021/11/04
The Two Formyl Peptide Receptors Differently Regulate GPR84-Mediated Neutrophil NADPH Oxidase Activity 期刊论文
JOURNAL OF INNATE IMMUNITY, 2021, 页码: 15
作者:  Martensson, Jonas;  Sundqvist, Martina;  Manandhar, Asmita;  Leremias, Loukas;  Zhang, Linjie
收藏  |  浏览/下载:40/0  |  提交时间:2021/05/24
Evaluation of biased agonism mediated by dual agonists of the GLP-1 and glucagon receptors 期刊论文
BIOCHEMICAL PHARMACOLOGY, 2020, 卷号: 180, 页码: 16
作者:  Darbalaei, Sanaz;  Yuliantie, Elita;  Dai, Antao;  Chang, Rulue;  Zhao, Peishen
收藏  |  浏览/下载:18/0  |  提交时间:2020/12/21
Pharmacological characterization of mono-, dual- and tri-peptidic agonists at GIP and GLP-1 receptors 期刊论文
BIOCHEMICAL PHARMACOLOGY, 2020, 卷号: 177, 页码: 13
作者:  Yuliantie, Elita;  Darbalaei, Sanaz;  Dai, Antao;  Zhao, Peishen;  Yang, Dehua
收藏  |  浏览/下载:21/0  |  提交时间:2020/12/24
Molecular mechanisms of fentanyl mediated beta-arrestin biased signaling 期刊论文
PLOS COMPUTATIONAL BIOLOGY, 2020, 卷号: 16, 期号: 4, 页码: 24
作者:  de Waal, Parker W.;  Shi, Jingjing;  You, Erli;  Wang, Xiaoxi;  Melcher, Karsten
收藏  |  浏览/下载:27/0  |  提交时间:2020/07/01
A complex structure of arrestin-2 bound to a G protein-coupled receptor 期刊论文
CELL RESEARCH, 2019, 卷号: 29, 期号: 12, 页码: 971-983
作者:  Yin, Wanchao;  Li, Zhihai;  Jin, Mingliang;  Yin, Yu-Ling;  de Waal, Parker W.
收藏  |  浏览/下载:84/0  |  提交时间:2020/07/01
Ligand-induced activation of ERK1/2 signaling by constitutively active G(s)-coupled 5-HT receptors 期刊论文
ACTA PHARMACOLOGICA SINICA, 2019, 卷号: 40, 期号: 9, 页码: 1157-1167
作者:  Liu, Ping;  Yin, Yu-ling;  Wang, Ting;  Hou, Li;  Wang, Xiao-xi
收藏  |  浏览/下载:19/0  |  提交时间:2020/07/01
5-HT4R  5-HT6R  5-HT7AR  5-HT  ERK1/2  G(s)  beta-arrestin  Fyn  Src  


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