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The discovery of novel and selective fatty acid binding protein 4 inhibitors by virtual screening and biological evaluation 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2016, 卷号: 24, 期号: 18, 页码: 4310-4317
作者:  Song, Ming;  Xu, Yong;  Zhang, Yan;  Nie, Tao;  Zhou, Yang
收藏  |  浏览/下载:22/0  |  提交时间:2018/12/13
Isolation of lingzhifuran A and lingzhilactones D-F from Ganoderma lucidum as specific Smad3 phosphorylation inhibitors and total synthesis of lingzhifuran 期刊论文
RSC ADVANCES, 2016, 卷号: 6, 期号: 81, 页码: 77887-77897
Ding, Wei-Yi; Ai, Jun; Wang, Xin-Long; Qiu, Fayang G.; Lv, Qing; Fang, Ping; Hou, Fan-Fan; Yan, Yong-Ming; Cheng, Yong-Xian
收藏  |  浏览/下载:19/0  |  提交时间:2016/12/16
Structure-Activity Relationship Study of Rakicidins: Overcoming Chronic Myeloid Leukemia Resistance to Imatinib with 4-Methylester-Rakicidin A 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 3, 页码: 1184-1196
作者:  Yang, Guang;  Zhang, Quan;  Chen, Yue;  Sang, Feng;  Ding, Yahui
收藏  |  浏览/下载:25/0  |  提交时间:2018/12/13
Discovery of Benzo[cd]indol-2(1H)-ones as Potent and Specific BET Bromodomain Inhibitors: Structure-Based Virtual Screening, Optimization, and Biological Evaluation 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 4, 页码: 1565-1579
作者:  Tu, Zhengchao;  Zhou, Yulai;  Ding, Ke;  Xu, Yong;  Xue, Xiaoqian
收藏  |  浏览/下载:25/0  |  提交时间:2018/12/13
Isolation of lingzhifuran A and lingzhilactones D-F from Ganoderma lucidum as specific Smad3 phosphorylation inhibitors and total synthesis of lingzhifuran 期刊论文
RSC ADVANCES, 2016, 卷号: 6, 期号: 81, 页码: 77887-77897
作者:  Hou, Fan-Fan;  Fang, Ping;  Lv, Qing;  Qiu, Fayang G.;  Wang, Xin-Long
收藏  |  浏览/下载:20/0  |  提交时间:2018/12/13
Discovery of Benzo[cd]indol-2(1H)-ones as Potent and Specific BET Bromodomain Inhibitors: Structure-Based Virtual Screening, Optimization, and Biological Evaluation 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 4, 页码: 1565-1579
Xue, Xiaoqian; Zhang, Yan; Liu, Zhaoxuan; Song, Ming; Xing, Yanli; Xiang, Qiuping; Wang, Zhen; Tu, Zhengchao; Zhou, Yulai; Ding, Ke; Xu, Yong
收藏  |  浏览/下载:21/0  |  提交时间:2016/12/16
The discovery of novel and selective fatty acid binding protein 4 inhibitors by virtual screening and biological evaluation 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2016, 卷号: 24, 期号: 18, 页码: 4310-4317
Zhou, Yang; Nie, Tao; Zhang, Yan; Song, Ming; Li, Kuai; Ding, Mengxiao; Ding, Ke; Wu, Donghai; Xu, Yong
收藏  |  浏览/下载:22/0  |  提交时间:2016/12/16
Structure-Activity Relationship Study of Rakicidins: Overcoming Chronic Myeloid Leukemia Resistance to Imatinib with 4-Methylester-Rakicidin A 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 3, 页码: 1184-1196
Sang, Feng; Ding, Yahui; Wang, Jinghan; Sun, Bingxia; Sun, Jianlei; Geng, Yan; Zhang, Zhang; Ding, Ke; Wu, Ling-Ling; Liu, Jian-Wei; Ba, Cuigai; Yang, Guang; Zhang, Quan; Li, Lu-Yuan; Chen, Yue
收藏  |  浏览/下载:46/0  |  提交时间:2016/12/16
Discovery and Optimization of 3-(2-(Pyrazolo[1,5-a]pyrimidin-6-yl)-ethynyl)benzamides as Novel Selective and Orally Bioavailable Discoidin Domain Receptor 1 (DDR1) Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2013, 卷号: 56, 期号: 8
作者:  Ding, Ke;  Ren, Xiaomei;  Xu, Yong;  Tu, Zhengchao;  Zhang, Zhang
收藏  |  浏览/下载:12/0  |  提交时间:2018/12/13
Discovery and Optimization of 3-(2-(Pyrazolo[1,5-a]pyrimidin-6-yl)-ethynyl)benzamides as Novel Selective and Orally Bioavailable Discoidin Domain Receptor 1 (DDR1) Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2013, 卷号: 56, 期号: 8
Gao, Mingshan; Duan, Lei; Luo, Jinfeng; Zhang, Lianwen; Lu, Xiaoyun; Zhang, Yan; Zhang, Zhang; Tu, Zhengchao; Xu, Yong; Ren, Xiaomei; Ding, Ke
收藏  |  浏览/下载:26/0  |  提交时间:2016/12/16


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